Flualprazolam (original) (raw)
Flualprazolam is a tranquilizer of the triazolobenzodiazepine (TBZD) class, which are benzodiazepines (BZDs) fused with a triazole ring. It was first synthesised in 1976, but was never marketed. It has subsequently been sold as a designer drug, first being definitively identified as such in Sweden in 2018. It can be described as the 2'-fluoro derivative of alprazolam or the fluoro instead of chloro analogue of triazolam, and has similar sedative and anxiolytic effects.
| Property | Value |
|---|---|
| dbo:abstract | Flualprazolam ist eine chemische Verbindung aus der Gruppe der Benzodiazepine, welches in den 1970er Jahren von (gehört heute zu Pfizer) entwickelt, aber niemals kommerziell vermarktet wurde. Es wird jedoch seit ca. 2018 als Designerdroge bzw. Legal-High über das Internet angeboten. Seit Januar 2021 wird es im BtMG aufgeführt. Man kann Flualprazolam als das 2'-Fluor-Derivat des Alprazolam sehen, oder als das Fluor- statt des Chlor-Analogons vom Triazolam. Es hat ähnlich wie dieses eine stark ausgeprägte hypnotische, sedative und anxiolytische Wirkung. Die geschätzte Äquivalenzdosis zu 10 mg Diazepam ist 0,25–0,5 mg. (de) Flualprazolam is a tranquilizer of the triazolobenzodiazepine (TBZD) class, which are benzodiazepines (BZDs) fused with a triazole ring. It was first synthesised in 1976, but was never marketed. It has subsequently been sold as a designer drug, first being definitively identified as such in Sweden in 2018. It can be described as the 2'-fluoro derivative of alprazolam or the fluoro instead of chloro analogue of triazolam, and has similar sedative and anxiolytic effects. (en) Il flualprazolam è uno psicofarmaco appartenente alla categoria delle che fu sintetizzato per la prima volta nel 1976, ma che non fu mai commercializzato. Successivamente è stato venduto come designer drug, identificato per la prima volta in Svezia in maniera definitiva nel 2018. Può essere considerato come il derivato 2'-fluoro dell'alprazolam e ha effetti sedativi simili ad altri ansiolitici. (it) O flualprazolam é um derivado da benzodiazepina que foi sintetizado pela primeira vez em 1976, mas nunca foi comercializado. Posteriormente foi vendido como um droga sintética, sendo identificado pela primeira vez na Suécia em 2018. Pode ser descrito como o derivado 2'-flúor do alprazolam, ou o flúor em vez do análogo do cloro do triazolam, e tem efeitos sedativos e ansiolíticos semelhantes. (pt) |
| dbo:casNumber | 28910-91-0 |
| dbo:fdaUniiCode | FWF5L8D2BE |
| dbo:pubchem | 10359044 |
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| dbp:h | 12 (xsd:integer) |
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| dbp:legalCa | Schedule IV (en) |
| dbp:legalDe | Anlage II (en) |
| dbp:legalStatus | Illegal in Sweden (en) |
| dbp:legalUk | PSA (en) |
| dbp:legalUn | P IV (en) |
| dbp:legalUs | Schedule I (en) |
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| dbp:pubchem | 10359044 (xsd:integer) |
| dbp:smiles | CC1=NN=C2N1C3=CCC4=CC=CC=C4F (en) |
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| rdfs:comment | Flualprazolam is a tranquilizer of the triazolobenzodiazepine (TBZD) class, which are benzodiazepines (BZDs) fused with a triazole ring. It was first synthesised in 1976, but was never marketed. It has subsequently been sold as a designer drug, first being definitively identified as such in Sweden in 2018. It can be described as the 2'-fluoro derivative of alprazolam or the fluoro instead of chloro analogue of triazolam, and has similar sedative and anxiolytic effects. (en) Il flualprazolam è uno psicofarmaco appartenente alla categoria delle che fu sintetizzato per la prima volta nel 1976, ma che non fu mai commercializzato. Successivamente è stato venduto come designer drug, identificato per la prima volta in Svezia in maniera definitiva nel 2018. Può essere considerato come il derivato 2'-fluoro dell'alprazolam e ha effetti sedativi simili ad altri ansiolitici. (it) O flualprazolam é um derivado da benzodiazepina que foi sintetizado pela primeira vez em 1976, mas nunca foi comercializado. Posteriormente foi vendido como um droga sintética, sendo identificado pela primeira vez na Suécia em 2018. Pode ser descrito como o derivado 2'-flúor do alprazolam, ou o flúor em vez do análogo do cloro do triazolam, e tem efeitos sedativos e ansiolíticos semelhantes. (pt) Flualprazolam ist eine chemische Verbindung aus der Gruppe der Benzodiazepine, welches in den 1970er Jahren von (gehört heute zu Pfizer) entwickelt, aber niemals kommerziell vermarktet wurde. Es wird jedoch seit ca. 2018 als Designerdroge bzw. Legal-High über das Internet angeboten. Seit Januar 2021 wird es im BtMG aufgeführt. (de) |
| rdfs:label | Flualprazolam (de) Flualprazolam (en) Flualprazolam (it) Flualprazolam (pt) |
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