| dbo:abstract |
ليفوكاباستين (بالإنجليزية: Levocabastine) هو دواء يُستعمل في علاج: * التهاب الملتحمة الحليمي العملاق (ar) Levocabastin ist ein Arzneistoff aus der Gruppe der H1-Antihistaminika der zweiten Generation. Es wird in Form von einer Suspension als Augentropfen und Nasenspray zur lokalen symptomatischen Behandlung allergischer Erkrankungen eingesetzt. (de) Levocabastine (trade name Livostin or Livocab, depending on the region) is a selective second-generation H1 receptor antagonist which was discovered at Janssen Pharmaceutica in 1979. It is used for allergic conjunctivitis. As well as acting as an antihistamine, levocabastine has also subsequently been found to act as a potent and selective antagonist for the neurotensin receptor NTS2, and was the first drug used to characterise the different neurotensin subtypes. This has made it a useful tool for the study of this receptor. The pharmaceutical drug Bilina is a combination of Levocabastine, benzalkonium chloride, and other components and is typically used in a 0.5 mg/ml suspension as eye-drops, dispensed in 4ml bottles for the treatment of allergic conjunctivitis or similar allergic ocular conditions. (en) La lévocabastine (R50547) est une substance chimique de la famille des cyclohexyl-3-méthylpipéridines qui possède des propriétés antihistaminiques H1. C'est une molécule utilisée dans le traitement des manifestations allergiques notamment oculaires conjonctivite. Il est commercialisé en France avec la spécialité Levophta. (fr) Levocabastina (nome comercial Livostin) é um seletivo de segunda geração o qual foi descoberto na Janssen Farmacêutica em 1979. É usado para conjuntivite alérgica. Além de atuar como anti-histamínico, levocabastina também foi encontrado como um antagonista potente e seletivo para o receptor de neurotensina , e foi a primeira droga utilizada para caracterizar os diferentes subtipos de neurotensina. Isso a tornou uma ferramenta útil para o estudo desse receptor. O medicamento Bilina é uma combinação de Levocabastina, cloreto de benzalcônio, e outros componentes e é tipicamente suada em suspensão a 0.5 mg/ml como um colírio, comercializada normalmente em frascos de 4ml para o tratamento de conjuntivite alérgica ou condições oculares alérgicas similares. (pt) |
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Livostin (en) |
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DB01106 |
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54385 |
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https://druginfo.nlm.nih.gov/drugportal/name/levocabastine%20hydrochloride https://druginfo.nlm.nih.gov/drugportal/rn/79516-68-0 |
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| rdfs:comment |
ليفوكاباستين (بالإنجليزية: Levocabastine) هو دواء يُستعمل في علاج: * التهاب الملتحمة الحليمي العملاق (ar) Levocabastin ist ein Arzneistoff aus der Gruppe der H1-Antihistaminika der zweiten Generation. Es wird in Form von einer Suspension als Augentropfen und Nasenspray zur lokalen symptomatischen Behandlung allergischer Erkrankungen eingesetzt. (de) La lévocabastine (R50547) est une substance chimique de la famille des cyclohexyl-3-méthylpipéridines qui possède des propriétés antihistaminiques H1. C'est une molécule utilisée dans le traitement des manifestations allergiques notamment oculaires conjonctivite. Il est commercialisé en France avec la spécialité Levophta. (fr) Levocabastine (trade name Livostin or Livocab, depending on the region) is a selective second-generation H1 receptor antagonist which was discovered at Janssen Pharmaceutica in 1979. It is used for allergic conjunctivitis. As well as acting as an antihistamine, levocabastine has also subsequently been found to act as a potent and selective antagonist for the neurotensin receptor NTS2, and was the first drug used to characterise the different neurotensin subtypes. This has made it a useful tool for the study of this receptor. (en) Levocabastina (nome comercial Livostin) é um seletivo de segunda geração o qual foi descoberto na Janssen Farmacêutica em 1979. É usado para conjuntivite alérgica. Além de atuar como anti-histamínico, levocabastina também foi encontrado como um antagonista potente e seletivo para o receptor de neurotensina , e foi a primeira droga utilizada para caracterizar os diferentes subtipos de neurotensina. Isso a tornou uma ferramenta útil para o estudo desse receptor. (pt) |
| rdfs:label |
ليفوكاباستين (ar) Levocabastin (de) Lévocabastine (fr) Levocabastine (en) Levocabastina (pt) |
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