| dbo:abstract |
تستولاكتون (بالإنجليزية: Testolactone) هو دواء يُستعمل في علاج: * سرطان الثدي (ar) Testolactone (INN, USAN) (brand name Teslac) is a non-selective, irreversible, steroidal aromatase inhibitor which is used as an antineoplastic drug to treat advanced-stage breast cancer.The drug was discontinued in 2008 and is no longer available for medical use. (en) Il Testolattone (17α-Oxa-D-omoandrosta-1,4-diene-3,17-dione) è un agente antineoplastico derivato del progesterone ed è utilizzato per trattare gli stadi avanzati del cancro al seno. È un antineoplastico sintetico strutturalmente distinto dagli androgeni steroidei poiché possiede un anello lattonico 6 atomi al posto del classico anello carbociclico a 5 atomi. (it) |
| dbo:alternativeName |
Teslac (en) |
| dbo:casNumber |
968-93-4 |
| dbo:chEBI |
9460 |
| dbo:chEMBL |
1571 |
| dbo:class |
dbr:Antiestrogen dbr:Aromatase_inhibitor |
| dbo:drugbank |
DB00894 |
| dbo:fdaUniiCode |
6J9BLA949Q |
| dbo:kegg |
D00153 |
| dbo:pubchem |
13769 |
| dbo:thumbnail |
wiki-commons:Special:FilePath/Testolactone.svg?width=300 |
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dbr:Liver |
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3 (xsd:integer) |
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C (en) |
| dbp:proteinBound |
~85% (en) |
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dbr:Oral_administration |
| dbp:smiles |
CC12CCC3CCCC4=CCC=CC34C (en) |
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Teslac (en) |
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| gold:hypernym |
dbr:Agent |
| rdf:type |
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| rdfs:comment |
تستولاكتون (بالإنجليزية: Testolactone) هو دواء يُستعمل في علاج: * سرطان الثدي (ar) Testolactone (INN, USAN) (brand name Teslac) is a non-selective, irreversible, steroidal aromatase inhibitor which is used as an antineoplastic drug to treat advanced-stage breast cancer.The drug was discontinued in 2008 and is no longer available for medical use. (en) Il Testolattone (17α-Oxa-D-omoandrosta-1,4-diene-3,17-dione) è un agente antineoplastico derivato del progesterone ed è utilizzato per trattare gli stadi avanzati del cancro al seno. È un antineoplastico sintetico strutturalmente distinto dagli androgeni steroidei poiché possiede un anello lattonico 6 atomi al posto del classico anello carbociclico a 5 atomi. (it) |
| rdfs:label |
تستولاكتون (ar) Testolattone (it) Testolactone (en) |
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freebase:Testolactone yago-res:Testolactone http://www4.wiwiss.fu-berlin.de/drugbank/resource/drugs/DB00894 wikidata:Testolactone dbpedia-ar:Testolactone dbpedia-cy:Testolactone dbpedia-it:Testolactone dbpedia-sh:Testolactone dbpedia-sr:Testolactone https://global.dbpedia.org/id/3g7E5 |
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wikipedia-en:Testolactone?oldid=1112041741&ns=0 |
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wiki-commons:Special:FilePath/Testolactone.svg |
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wikipedia-en:Testolactone |
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