Synthesis of New Thieno[b]azepinediones from α-Methylene Ketones (original) (raw)

Synthesis 2002(8): 1096-1100
DOI: 10.1055/s-2002-31963

PAPER

© Georg Thieme Verlag Stuttgart · New York

Evelyne Migianu, Gilbert Kirsch*
Laboratoire d’Ingénierie Moléculaire et Biochimie Pharmacologique, Faculté des Sciences, Université de Metz, Ile du Saulcy, 57045 Metz Cedex, France
Fax: +33(3)87315333; e-Mail: kirsch@sciences.univ-metz.fr;

Further Information

Publication History

Received 25 January 2002
Publication Date:
03 June 2002 (online)

• Abstract
• Full Text
• References

Abstract

New substituted 6,7-dihydro-4_H_-thieno[3,2-_b_]azepine-5,8-diones were synthesized in seven steps, starting from substituted α-methylene ketones, via 3-aminothiophene-2-carboxylic acid alkyl esters.

Key words

heterocycles - thieno[_b_]azepinediones - α-methylene ketones - 3-aminothiophene-2-carboxylic acid alkyl esters

References

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