Cytokine-dependent imatinib resistance in mouse BCR-ABL+, Arf-null lymphoblastic leukemia (original) (raw)
- Richard T. Williams1,
- Willem den Besten2,3, and
- Charles J. Sherr2,3,4
- 1 Department of Oncology, St. Jude Children’s Research Hospital, Memphis, Tennessee 38105, USA;
- 2 Department of Genetics and Tumor Cell Biology, St. Jude Children’s Research Hospital, Memphis, Tennessee 38105, USA;
- 3 Howard Hughes Medical Institute, St. Jude Children’s Research Hospital, Memphis, Tennessee 38105, USA
Abstract
Retroviral transduction of the BCR-ABL kinase into primary mouse bone marrow cells lacking the Arf tumor suppressor rapidly generates polyclonal populations of continuously self-renewing pre-B cells, virtually all of which have leukemic potential. Intravenous infusion of 20 such cells into healthy syngeneic mice induces rapidly fatal, transplantable lymphoblastic leukemias that resist imatinib therapy. Introduction of BCR-ABL into _Arf_-null severe combined immunodeficient (SCID) bone marrow progenitors lacking the cytokine receptor common γ-chain yields leukemogenic pre-B cells that exhibit greater sensitivity to imatinib in vivo. Hence, salutary cytokines in the hematopoietic microenvironment can facilitate leukemic proliferation and confer resistance to targeted therapy.
- BCR-ABL kinase
- Arf tumor suppressor
- imatinib (Gleevec)
- leukemia-initiating cells
- cytokines
- drug resistance
Footnotes
↵4 Corresponding author.
↵4 E-MAIL sherr{at}stjude.org; FAX (901) 495-2381.Supplemental material is available at http://www.genesdev.org.
Article published online ahead of print. Article and publication date are online at http://www.genesdev.org/cgi/doi/10.1101/gad.1588607
- Received June 29, 2007.
- Accepted July 25, 2007.
Freely available online through the Genes & Development Open Access option.
Copyright © 2007, Cold Spring Harbor Laboratory Press