Fátima Mota - Academia.edu (original) (raw)

Fátima Mota

Related Authors

cesar huamani

Marcela Gonzalez

Marcela Gonzalez

Universidad Nacional de Colombia (National University of Colombia)

Uploads

Papers by Fátima Mota

Research paper thumbnail of Calculation of drug-like molecules solubility using predictive activity coefficient models

Fluid Phase Equilibria, 2012

The A-UNIFAC, UNIFAC, and NRTL-SAC models are used to predict solubility in pure solvents of a se... more The A-UNIFAC, UNIFAC, and NRTL-SAC models are used to predict solubility in pure solvents of a set of drug-like molecules. To apply A-UNIFAC, a new set of residual interaction parameters between the ACOH group and six other groups had to be estimated. The solute model parameters of NRTL-SAC were also estimated for this set of molecules. NRTL-SAC showed better performance at 298.15 K, with an average absolute deviation of 37.6%. Solubility dependence with temperature was also studied: all models presented average deviations around 40%. In general, there is an improvement given by the A-UNIFAC over the UNIFAC in aqueous systems, proving the importance of taking association into account.

Research paper thumbnail of Calculation of drug-like molecules solubility using predictive activity coefficient models

Fluid Phase Equilibria, 2012

The A-UNIFAC, UNIFAC, and NRTL-SAC models are used to predict solubility in pure solvents of a se... more The A-UNIFAC, UNIFAC, and NRTL-SAC models are used to predict solubility in pure solvents of a set of drug-like molecules. To apply A-UNIFAC, a new set of residual interaction parameters between the ACOH group and six other groups had to be estimated. The solute model parameters of NRTL-SAC were also estimated for this set of molecules. NRTL-SAC showed better performance at 298.15 K, with an average absolute deviation of 37.6%. Solubility dependence with temperature was also studied: all models presented average deviations around 40%. In general, there is an improvement given by the A-UNIFAC over the UNIFAC in aqueous systems, proving the importance of taking association into account.

Log In