Jan Mos - Academia.edu (original) (raw)

Papers by Jan Mos

Research paper thumbnail of Eltoprazine - a specific anti-aggressive drug (serenic) in animal aggression models

Aggressive Behavior, 1989

Research paper thumbnail of Ultrasonic vocalisation, rectal temperature and negative geotaxis: effects of benzodiazepine receptor ligands

Research paper thumbnail of Everill, B., Brain, P.F., Rustana, A., Mos, J. and Olivier, B. (1991). Ethoexperimental analysis of the impact of Chlordiazepoxide (CPD) on social interactions in three strains of mice. Behavioural Processes 25: 55-67

Research paper thumbnail of A motivational analysis of ambivalent actions in the agonistic behaviour of rats in tests used to study effects of drugs on aggression

Progress in clinical and biological research, 1984

Research paper thumbnail of A comparison of the full 5-HT1A agonist flesinoxan with other 5-HT1A agonists: Effects on behaviour and a quantification of (partial) agonism on cells

European Neuropsychopharmacology, 1996

Research paper thumbnail of Results and significance of the RIVM Strategic Research 2007-2010 : Prepared for the future

Dit rapport brengt verslag uit van vier jaar Strategisch Onderzoek RIVM (SOR), het eigen onderzoe... more Dit rapport brengt verslag uit van vier jaar Strategisch Onderzoek RIVM (SOR), het eigen onderzoeksbudget van het RIVM. Het SOR-budget is bedoeld voor onderzoek om het RIVM te voorzien van de benodigde expertise en kwaliteit, zodat het nu en in de toekomst taken voor opdrachtgevers adequaat kan uitvoeren. Het rapport geeft de inhoudelijke resultaten en toepassingsmogelijkheden weer van alle projecten over de periode 2007-2010. In totaal zijn in de onderzoeksperiode 86 projecten uitgevoerd, onderverdeeld in 6 strategische thema's. Ongeveer een derde deel van de projecten loopt nog door na 2011; de voorlopige resultaten van de lopende projecten zijn hier vermeld. De resultaten van dit SOR-programma bestaan uit een schat aan nieuw instrumentarium, nieuwe data en kennis, en verbetering van bestaand instrumentarium en bestaande kennis op het gebied van volksgezondheid en milieu. Deze resultaten dragen in belangrijke mate bij aan de uitvoering van de huidige kerntaken van het RIVM. Da...

Research paper thumbnail of Aggression Induced by Electrical-Stimulation in the Hypothalamus of Male and Female Rats

Research paper thumbnail of Serotonergic Modulation of Agonistic Behaviour

Topics in the Neurosciences, 1987

Over the last fifteen years several hypotheses have emerged concerning the neurochemical control ... more Over the last fifteen years several hypotheses have emerged concerning the neurochemical control of aggressive behaviour. A variety of single neurotransmitters were suggested to control. aggression e.g. the “aggressive monoamines” (Eichelman and Thoa 973), acetylcholine (Smith et a1. 1970) and serotonin (Valzelli and Garattini 1968). Later, the theories of single neurotransmitter control were extended to multi-transmitter modulation of aggressive behaviour (Avis 1974; Daruna 1978; Pradhan 1915; Reis 1974).

Research paper thumbnail of Ethopharmacological studies differentiate the effects of various serotonergic compounds on aggression in rats

Drug Development Research, 1992

ABSTRACT

Research paper thumbnail of Behavioural Pharmacology of the 5-HT1A Agonist Flesinoxan

Behavioural Pharmacology, 1992

Research paper thumbnail of Preclinical Characteristics of the Anti-Aggressive Actions of Eltoprazine

Clinical Neuropharmacology, 1992

Research paper thumbnail of A Comparison of Drug Responses by Male and Female Rats During Aggression Tests

The Development of Sex Differences and Similarities in Behavior, 1993

The scope of this chapter is to compare the differences and similarities of the neuropharmacology... more The scope of this chapter is to compare the differences and similarities of the neuropharmacology of male and female aggression in rats. Unfortunately such a task is far from easy because aggression research in the realm of neuropharmacology has mainly focussed on males, notably in rodents. The reasons for this choice are obvious and valid. With some exceptions, under many circumstances males are more aggressive than females. However, the generality of our conclusions ana our knowledge on brain-behavior relationships is severily limited by this bias to study male aggression. In contrast to the more etho-ecologically oriented studies, in most psycho-pharmacological experiments there is no emphasis on the function of the observed behavior, which may profoundly differ in males and females. Indeed the adaptive or survival value of aggression in rodents housed under laboratory conditions can only be extrapolated from their feral counterparts. However, to study the neuropharmacological organization under more ecologically relevant conditions is not very practical, not to say impossible. We therefore have to rely on extrapolations from the laboratory situation to more naturalistic situations and vice versa. A comparison of the neuropharmacology of male and female aggression is interesting for different reasons. First, it is important to understand the regulation of aggression within different genders of the same species where internal and external factors evoking aggression may differ profoundly. Is the basic neuropharmacology similar despite the diversity in the other regulatory mechanisms? Second, it is of interest to know whether drugs that modulate aggression in males are equally effective and selective in both sexes. Our work was to a large extent governed by the latter interest. Since we have discovered and developed drugs that exert unique anti-aggressive actions in animals, we wanted to know whether these drugs could be equally useful for treating (pathological) aggression in males and females. 205

Research paper thumbnail of Serotoninergic Function and Aggression in Animals

Serotonin (5-hydroxytryptamine; 5-HT) has for some time been implicated in the control of aggress... more Serotonin (5-hydroxytryptamine; 5-HT) has for some time been implicated in the control of aggression. Early work on 5-HT and aggression indicated that general 5-HT activation decreased aggression, whereas an overall inactivation of 5-HT by various means enhanced it (Valzelli, 1981).

Research paper thumbnail of Electrical Stimulation as a Tool to Trace Physiological Properties of the Hypothalamic Network in Aggression

The Biology of Aggression, 1981

ABSTRACT The aggressive responses during electrical stimulation in the hypothalamus may or may no... more ABSTRACT The aggressive responses during electrical stimulation in the hypothalamus may or may not derive from activation of a neural system especially subservient to aggression, for we do not know which neuronal elements mediate such effects. In order to identify these neurons one can try to define their location and to trace their anatomical connections. In addition it appears possible to estimate the physiological properties of the network involved, by threshold-intensity measurements at different preset parameters of the stimulating current. Such measurements may then provide a basis for comparison of the networks involved in stimulation-induced aggression and the networks involved in concomitant behavioral responses.

Research paper thumbnail of Concepts in Animal Models for Pathological Aggressive Behaviour in Humans

Animal models for psychiatric disorders should ideally fullfil the following criteria: the behavi... more Animal models for psychiatric disorders should ideally fullfil the following criteria: the behavioural abnormalities should be measurable in an appropriate context and the neurobiological causes for this deviant behaviour should be known. In case these criteria are met, these models might be called homologous, in a similar way as for instance used in functional morphology. It is clear that these conditions are not met by the current models for aggressive behaviour in animals.

Research paper thumbnail of 5HT 1A behavioural models

Pharmacochemistry Library

Publisher Summary 5-HT 1A receptor agonists have been tested in a wide variety of animal models i... more Publisher Summary 5-HT 1A receptor agonists have been tested in a wide variety of animal models indicative of CNS functions. These range from models for motion sickness and emesis to models predictive for antipsychotic drugs. In most of these tests, 5-HT 1A receptor agonists appear to be active, although the degree of specificity varies. 5-HT 1A receptor agonists influence the total serotonin neurotransmission by acting on the somatodendritic autoreceptor as well as by acting on postsynaptic receptors. From many behavioral effects of 5-HT 1A receptor agonists, the precise molecular mechanism of action remains elusive and it is quite conceivable that similar behavioral effects can be induced by various manipulations of the serotonin neurotransmission.

Research paper thumbnail of Measuring Behavior '96, International Workshop on Methods and Techniques in Behavioral Research (Utrecht, The Netherlands, 16-18 October 1996)

Research paper thumbnail of Etho-Experimental Studies of Similarities and Differences in Male and Female Agonistic Behaviour

Ethoexperimental Approaches to the Study of Behavior, 1989

Research paper thumbnail of Preclinical Evidence for the Role of Serotonin Receptors in Anxiety

Medical Science Symposia Series, 1993

Animal paradigms are important to detect anxiolytic properties of psychoactive compounds. Two ani... more Animal paradigms are important to detect anxiolytic properties of psychoactive compounds. Two animal anxiety paradigms are presented, ultrasonic distress vocalizations (USV) in rat pups and stress-induced hyperthermia (SIH) in mice, to describe the putative anxiolytic properties of serotonergic ligands. Both paradigms indicate that 5-HTAreceptor agonists are potent anxiolytics, whereas specific 5-HT reuptake blockers also exert some anxiolytic properties. 5-HT02antagonists may have some anxiogenic properties (in USV), whereas 5-HT, antagonists seem to be devoid of anxiolytic properties in the paradigms used.

Research paper thumbnail of Pro-Aggressive Actions of Benzodiazepines

Topics in the Neurosciences, 1987

The benzodiazepines (BDZ) are known for a wide variety of pharmacological effects, among which an... more The benzodiazepines (BDZ) are known for a wide variety of pharmacological effects, among which anxiolytic, hypnotic, sedatory, muscle relaxing and anticonvulsant actions are the most prominent. Much progress has been made in the elucidation of their mechanism of action by the discovery and characterization of high affinity binding sites for BDZ in the brain. However, not all complex behavioural actions are completely explained by the concepts derived from receptor binding. One such behavioural response is the intriguing question of the pro-aggressive action of low doses of benzodiazepines.

Research paper thumbnail of Eltoprazine - a specific anti-aggressive drug (serenic) in animal aggression models

Aggressive Behavior, 1989

Research paper thumbnail of Ultrasonic vocalisation, rectal temperature and negative geotaxis: effects of benzodiazepine receptor ligands

Research paper thumbnail of Everill, B., Brain, P.F., Rustana, A., Mos, J. and Olivier, B. (1991). Ethoexperimental analysis of the impact of Chlordiazepoxide (CPD) on social interactions in three strains of mice. Behavioural Processes 25: 55-67

Research paper thumbnail of A motivational analysis of ambivalent actions in the agonistic behaviour of rats in tests used to study effects of drugs on aggression

Progress in clinical and biological research, 1984

Research paper thumbnail of A comparison of the full 5-HT1A agonist flesinoxan with other 5-HT1A agonists: Effects on behaviour and a quantification of (partial) agonism on cells

European Neuropsychopharmacology, 1996

Research paper thumbnail of Results and significance of the RIVM Strategic Research 2007-2010 : Prepared for the future

Dit rapport brengt verslag uit van vier jaar Strategisch Onderzoek RIVM (SOR), het eigen onderzoe... more Dit rapport brengt verslag uit van vier jaar Strategisch Onderzoek RIVM (SOR), het eigen onderzoeksbudget van het RIVM. Het SOR-budget is bedoeld voor onderzoek om het RIVM te voorzien van de benodigde expertise en kwaliteit, zodat het nu en in de toekomst taken voor opdrachtgevers adequaat kan uitvoeren. Het rapport geeft de inhoudelijke resultaten en toepassingsmogelijkheden weer van alle projecten over de periode 2007-2010. In totaal zijn in de onderzoeksperiode 86 projecten uitgevoerd, onderverdeeld in 6 strategische thema's. Ongeveer een derde deel van de projecten loopt nog door na 2011; de voorlopige resultaten van de lopende projecten zijn hier vermeld. De resultaten van dit SOR-programma bestaan uit een schat aan nieuw instrumentarium, nieuwe data en kennis, en verbetering van bestaand instrumentarium en bestaande kennis op het gebied van volksgezondheid en milieu. Deze resultaten dragen in belangrijke mate bij aan de uitvoering van de huidige kerntaken van het RIVM. Da...

Research paper thumbnail of Aggression Induced by Electrical-Stimulation in the Hypothalamus of Male and Female Rats

Research paper thumbnail of Serotonergic Modulation of Agonistic Behaviour

Topics in the Neurosciences, 1987

Over the last fifteen years several hypotheses have emerged concerning the neurochemical control ... more Over the last fifteen years several hypotheses have emerged concerning the neurochemical control of aggressive behaviour. A variety of single neurotransmitters were suggested to control. aggression e.g. the “aggressive monoamines” (Eichelman and Thoa 973), acetylcholine (Smith et a1. 1970) and serotonin (Valzelli and Garattini 1968). Later, the theories of single neurotransmitter control were extended to multi-transmitter modulation of aggressive behaviour (Avis 1974; Daruna 1978; Pradhan 1915; Reis 1974).

Research paper thumbnail of Ethopharmacological studies differentiate the effects of various serotonergic compounds on aggression in rats

Drug Development Research, 1992

ABSTRACT

Research paper thumbnail of Behavioural Pharmacology of the 5-HT1A Agonist Flesinoxan

Behavioural Pharmacology, 1992

Research paper thumbnail of Preclinical Characteristics of the Anti-Aggressive Actions of Eltoprazine

Clinical Neuropharmacology, 1992

Research paper thumbnail of A Comparison of Drug Responses by Male and Female Rats During Aggression Tests

The Development of Sex Differences and Similarities in Behavior, 1993

The scope of this chapter is to compare the differences and similarities of the neuropharmacology... more The scope of this chapter is to compare the differences and similarities of the neuropharmacology of male and female aggression in rats. Unfortunately such a task is far from easy because aggression research in the realm of neuropharmacology has mainly focussed on males, notably in rodents. The reasons for this choice are obvious and valid. With some exceptions, under many circumstances males are more aggressive than females. However, the generality of our conclusions ana our knowledge on brain-behavior relationships is severily limited by this bias to study male aggression. In contrast to the more etho-ecologically oriented studies, in most psycho-pharmacological experiments there is no emphasis on the function of the observed behavior, which may profoundly differ in males and females. Indeed the adaptive or survival value of aggression in rodents housed under laboratory conditions can only be extrapolated from their feral counterparts. However, to study the neuropharmacological organization under more ecologically relevant conditions is not very practical, not to say impossible. We therefore have to rely on extrapolations from the laboratory situation to more naturalistic situations and vice versa. A comparison of the neuropharmacology of male and female aggression is interesting for different reasons. First, it is important to understand the regulation of aggression within different genders of the same species where internal and external factors evoking aggression may differ profoundly. Is the basic neuropharmacology similar despite the diversity in the other regulatory mechanisms? Second, it is of interest to know whether drugs that modulate aggression in males are equally effective and selective in both sexes. Our work was to a large extent governed by the latter interest. Since we have discovered and developed drugs that exert unique anti-aggressive actions in animals, we wanted to know whether these drugs could be equally useful for treating (pathological) aggression in males and females. 205

Research paper thumbnail of Serotoninergic Function and Aggression in Animals

Serotonin (5-hydroxytryptamine; 5-HT) has for some time been implicated in the control of aggress... more Serotonin (5-hydroxytryptamine; 5-HT) has for some time been implicated in the control of aggression. Early work on 5-HT and aggression indicated that general 5-HT activation decreased aggression, whereas an overall inactivation of 5-HT by various means enhanced it (Valzelli, 1981).

Research paper thumbnail of Electrical Stimulation as a Tool to Trace Physiological Properties of the Hypothalamic Network in Aggression

The Biology of Aggression, 1981

ABSTRACT The aggressive responses during electrical stimulation in the hypothalamus may or may no... more ABSTRACT The aggressive responses during electrical stimulation in the hypothalamus may or may not derive from activation of a neural system especially subservient to aggression, for we do not know which neuronal elements mediate such effects. In order to identify these neurons one can try to define their location and to trace their anatomical connections. In addition it appears possible to estimate the physiological properties of the network involved, by threshold-intensity measurements at different preset parameters of the stimulating current. Such measurements may then provide a basis for comparison of the networks involved in stimulation-induced aggression and the networks involved in concomitant behavioral responses.

Research paper thumbnail of Concepts in Animal Models for Pathological Aggressive Behaviour in Humans

Animal models for psychiatric disorders should ideally fullfil the following criteria: the behavi... more Animal models for psychiatric disorders should ideally fullfil the following criteria: the behavioural abnormalities should be measurable in an appropriate context and the neurobiological causes for this deviant behaviour should be known. In case these criteria are met, these models might be called homologous, in a similar way as for instance used in functional morphology. It is clear that these conditions are not met by the current models for aggressive behaviour in animals.

Research paper thumbnail of 5HT 1A behavioural models

Pharmacochemistry Library

Publisher Summary 5-HT 1A receptor agonists have been tested in a wide variety of animal models i... more Publisher Summary 5-HT 1A receptor agonists have been tested in a wide variety of animal models indicative of CNS functions. These range from models for motion sickness and emesis to models predictive for antipsychotic drugs. In most of these tests, 5-HT 1A receptor agonists appear to be active, although the degree of specificity varies. 5-HT 1A receptor agonists influence the total serotonin neurotransmission by acting on the somatodendritic autoreceptor as well as by acting on postsynaptic receptors. From many behavioral effects of 5-HT 1A receptor agonists, the precise molecular mechanism of action remains elusive and it is quite conceivable that similar behavioral effects can be induced by various manipulations of the serotonin neurotransmission.

Research paper thumbnail of Measuring Behavior '96, International Workshop on Methods and Techniques in Behavioral Research (Utrecht, The Netherlands, 16-18 October 1996)

Research paper thumbnail of Etho-Experimental Studies of Similarities and Differences in Male and Female Agonistic Behaviour

Ethoexperimental Approaches to the Study of Behavior, 1989

Research paper thumbnail of Preclinical Evidence for the Role of Serotonin Receptors in Anxiety

Medical Science Symposia Series, 1993

Animal paradigms are important to detect anxiolytic properties of psychoactive compounds. Two ani... more Animal paradigms are important to detect anxiolytic properties of psychoactive compounds. Two animal anxiety paradigms are presented, ultrasonic distress vocalizations (USV) in rat pups and stress-induced hyperthermia (SIH) in mice, to describe the putative anxiolytic properties of serotonergic ligands. Both paradigms indicate that 5-HTAreceptor agonists are potent anxiolytics, whereas specific 5-HT reuptake blockers also exert some anxiolytic properties. 5-HT02antagonists may have some anxiogenic properties (in USV), whereas 5-HT, antagonists seem to be devoid of anxiolytic properties in the paradigms used.

Research paper thumbnail of Pro-Aggressive Actions of Benzodiazepines

Topics in the Neurosciences, 1987

The benzodiazepines (BDZ) are known for a wide variety of pharmacological effects, among which an... more The benzodiazepines (BDZ) are known for a wide variety of pharmacological effects, among which anxiolytic, hypnotic, sedatory, muscle relaxing and anticonvulsant actions are the most prominent. Much progress has been made in the elucidation of their mechanism of action by the discovery and characterization of high affinity binding sites for BDZ in the brain. However, not all complex behavioural actions are completely explained by the concepts derived from receptor binding. One such behavioural response is the intriguing question of the pro-aggressive action of low doses of benzodiazepines.