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Papers by Jean-yves Mérour
ChemInform, Apr 4, 2006
ABSTRACT
Current Organic Chemistry, May 1, 2001
Abstract: The results of research into the chemistry of 7-azaindole during the last twenty years ... more Abstract: The results of research into the chemistry of 7-azaindole during the last twenty years are presented. New synthetic methods for the 7-azaindole structures are developed including palladium-catalysed cross-coupling reactions. Reactivity of 3-formyl-, 3-halogeno-and 2-...
Chemischer Informationsdienst, Dec 26, 1978
ChemInform, Dec 2, 2003
A new family of pyrrolo[1,2:1%,2%]azepino[5,6-b]indole derivatives 8,15 related to anthramycin sk... more A new family of pyrrolo[1,2:1%,2%]azepino[5,6-b]indole derivatives 8,15 related to anthramycin skeleton was prepared in good yield from indole-2-carboxylic acid and b-aminoesters 4 through intramolecular cyclisation.
ChemInform, Jan 14, 2003
Fused pyridine derivatives Fused pyridine derivatives R 0450 A Straightforward Synthesis of Oxazi... more Fused pyridine derivatives Fused pyridine derivatives R 0450 A Straightforward Synthesis of Oxazino[2,3,4-ij]quinoline Derivatives from 8-Hydroxyquinolines.-The reaction of hydroxyquinolines (I), (IV) and (VIII) and hydroxyisoquinoline (XI) with 2,3-dibromopropanoate (II) and related dibromo compounds (XIII) and (XV) is studied. In a variety of cases, tricyclic or tetracyclic derivatives (III), (IX) and (XIV) are obtained as the products.-(ARRAULT, A.;
ChemInform, Mar 27, 2007
A new route to the paullone scaffold was designed. The key step consisted in a free radical indol... more A new route to the paullone scaffold was designed. The key step consisted in a free radical indole formation from an o-alkenyl arylisonitrile followed by Stille coupling with N-Boc-o-iodoaniline. After deprotection and closure of the seven-membered ring by lactamisation, parent or cyano-substituted paullones were obtained in moderate to good yields.
ChemInform, Apr 4, 2006
ABSTRACT
Current Organic Chemistry, May 1, 2001
Abstract: The results of research into the chemistry of 7-azaindole during the last twenty years ... more Abstract: The results of research into the chemistry of 7-azaindole during the last twenty years are presented. New synthetic methods for the 7-azaindole structures are developed including palladium-catalysed cross-coupling reactions. Reactivity of 3-formyl-, 3-halogeno-and 2-...
Chemischer Informationsdienst, Dec 26, 1978
ChemInform, Dec 2, 2003
A new family of pyrrolo[1,2:1%,2%]azepino[5,6-b]indole derivatives 8,15 related to anthramycin sk... more A new family of pyrrolo[1,2:1%,2%]azepino[5,6-b]indole derivatives 8,15 related to anthramycin skeleton was prepared in good yield from indole-2-carboxylic acid and b-aminoesters 4 through intramolecular cyclisation.
ChemInform, Jan 14, 2003
Fused pyridine derivatives Fused pyridine derivatives R 0450 A Straightforward Synthesis of Oxazi... more Fused pyridine derivatives Fused pyridine derivatives R 0450 A Straightforward Synthesis of Oxazino[2,3,4-ij]quinoline Derivatives from 8-Hydroxyquinolines.-The reaction of hydroxyquinolines (I), (IV) and (VIII) and hydroxyisoquinoline (XI) with 2,3-dibromopropanoate (II) and related dibromo compounds (XIII) and (XV) is studied. In a variety of cases, tricyclic or tetracyclic derivatives (III), (IX) and (XIV) are obtained as the products.-(ARRAULT, A.;
ChemInform, Mar 27, 2007
A new route to the paullone scaffold was designed. The key step consisted in a free radical indol... more A new route to the paullone scaffold was designed. The key step consisted in a free radical indole formation from an o-alkenyl arylisonitrile followed by Stille coupling with N-Boc-o-iodoaniline. After deprotection and closure of the seven-membered ring by lactamisation, parent or cyano-substituted paullones were obtained in moderate to good yields.