Targeting tumor-associated macrophages with anti-CSF-1R antibody reveals a strategy for cancer therapy - PubMed (original) (raw)
. 2014 Jun 16;25(6):846-59.
doi: 10.1016/j.ccr.2014.05.016. Epub 2014 Jun 2.
Michael A Cannarile 2, Sabine Hoves 2, Jörg Benz 3, Katharina Wartha 2, Valeria Runza 2, Flora Rey-Giraud 2, Leon P Pradel 2, Friedrich Feuerhake 4, Irina Klaman 2, Tobin Jones 2, Ute Jucknischke 2, Stefan Scheiblich 2, Klaus Kaluza 2, Ingo H Gorr 2, Antje Walz 5, Keelara Abiraj 5, Philippe A Cassier 6, Antonio Sica 7, Carlos Gomez-Roca 8, Karin E de Visser 9, Antoine Italiano 10, Christophe Le Tourneau 11, Jean-Pierre Delord 8, Hyam Levitsky 12, Jean-Yves Blay 6, Dominik Rüttinger 2
Affiliations
- PMID: 24898549
- DOI: 10.1016/j.ccr.2014.05.016
Free article
Targeting tumor-associated macrophages with anti-CSF-1R antibody reveals a strategy for cancer therapy
Carola H Ries et al. Cancer Cell. 2014.
Free article
Abstract
Macrophage infiltration has been identified as an independent poor prognostic factor in several cancer types. The major survival factor for these macrophages is macrophage colony-stimulating factor 1 (CSF-1). We generated a monoclonal antibody (RG7155) that inhibits CSF-1 receptor (CSF-1R) activation. In vitro RG7155 treatment results in cell death of CSF-1-differentiated macrophages. In animal models, CSF-1R inhibition strongly reduces F4/80(+) tumor-associated macrophages accompanied by an increase of the CD8(+)/CD4(+) T cell ratio. Administration of RG7155 to patients led to striking reductions of CSF-1R(+)CD163(+) macrophages in tumor tissues, which translated into clinical objective responses in diffuse-type giant cell tumor (Dt-GCT) patients.
Trial registration: ClinicalTrials.gov NCT01494688.
Copyright © 2014 Elsevier Inc. All rights reserved.
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