Vinyl sulfones as mechanism-based cysteine protease inhibitors - PubMed (original) (raw)
. 1995 Aug 18;38(17):3193-6.
doi: 10.1021/jm00017a002.
Affiliations
- PMID: 7650671
- DOI: 10.1021/jm00017a002
Vinyl sulfones as mechanism-based cysteine protease inhibitors
J T Palmer et al. J Med Chem. 1995.
No abstract available
Similar articles
- Synthesis of macrocyclic trypanosomal cysteine protease inhibitors.
Chen YT, Lira R, Hansell E, McKerrow JH, Roush WR. Chen YT, et al. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5860-3. doi: 10.1016/j.bmcl.2008.06.012. Epub 2008 Jun 10. Bioorg Med Chem Lett. 2008. PMID: 18585034 Free PMC article. - The design and synthesis of inhibitors of the cysteinyl protease, Der p I.
Billson J, Clark J, Conway SP, Hart T, Johnson T, Langston SP, Ramjee M, Quibell M, Scott RK. Billson J, et al. Bioorg Med Chem Lett. 1998 May 5;8(9):993-8. doi: 10.1016/s0960-894x(98)00151-6. Bioorg Med Chem Lett. 1998. PMID: 9871695 - Aspartic vinyl sulfones: inhibitors of a caspase-3-dependent pathway.
Glória PM, Coutinho I, Gonçalves LM, Baptista C, Soares J, Newton AS, Moreira R, Saraiva L, Santos MM. Glória PM, et al. Eur J Med Chem. 2011 Jun;46(6):2141-6. doi: 10.1016/j.ejmech.2011.02.067. Epub 2011 Mar 5. Eur J Med Chem. 2011. PMID: 21439692 - Synthesis and structure-activity relationship studies of cruzain and rhodesain inhibitors.
Rocha DA, Silva EB, Fortes IS, Lopes MS, Ferreira RS, Andrade SF. Rocha DA, et al. Eur J Med Chem. 2018 Sep 5;157:1426-1459. doi: 10.1016/j.ejmech.2018.08.079. Epub 2018 Aug 31. Eur J Med Chem. 2018. PMID: 30282318 Review. - Michael acceptors as cysteine protease inhibitors.
Santos MM, Moreira R. Santos MM, et al. Mini Rev Med Chem. 2007 Oct;7(10):1040-50. doi: 10.2174/138955707782110105. Mini Rev Med Chem. 2007. PMID: 17979807 Review.
Cited by
- Clickable Probes for Pathogen Proteasomes: Synthesis and Applications.
Liu LJ, Lucero B, Manriquez-Rodriguez C, Francisco KR, Teixeira TR, Yohannan DJ, Ballatore C, Myers SA, O'Donoghue AJ, Caffrey CR. Liu LJ, et al. ACS Omega. 2024 Aug 2;9(32):34829-34840. doi: 10.1021/acsomega.4c04316. eCollection 2024 Aug 13. ACS Omega. 2024. PMID: 39157084 Free PMC article. - The clinical significance of cathepsin S expression in human astrocytomas.
Flannery T, Gibson D, Mirakhur M, McQuaid S, Greenan C, Trimble A, Walker B, McCormick D, Johnston PG. Flannery T, et al. Am J Pathol. 2003 Jul;163(1):175-82. doi: 10.1016/S0002-9440(10)63641-3. Am J Pathol. 2003. PMID: 12819022 Free PMC article. - Schistosomiasis mansoni: novel chemotherapy using a cysteine protease inhibitor.
Abdulla MH, Lim KC, Sajid M, McKerrow JH, Caffrey CR. Abdulla MH, et al. PLoS Med. 2007 Jan;4(1):e14. doi: 10.1371/journal.pmed.0040014. PLoS Med. 2007. PMID: 17214506 Free PMC article. - Synthesis of macrocyclic trypanosomal cysteine protease inhibitors.
Chen YT, Lira R, Hansell E, McKerrow JH, Roush WR. Chen YT, et al. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5860-3. doi: 10.1016/j.bmcl.2008.06.012. Epub 2008 Jun 10. Bioorg Med Chem Lett. 2008. PMID: 18585034 Free PMC article. - Synthesis and SAR study of novel peptide aldehydes as inhibitors of 20S proteasome.
Ma Y, Xu B, Fang Y, Yang Z, Cui J, Zhang L, Zhang L. Ma Y, et al. Molecules. 2011 Sep 5;16(9):7551-64. doi: 10.3390/molecules16097551. Molecules. 2011. PMID: 21894088 Free PMC article.
MeSH terms
Substances
LinkOut - more resources
Other Literature Sources
Chemical Information