original ) (raw )3-(2-Methoxytetrahydrofuran-2-yl)pyrazoles: a novel class of potent, selective cyclooxygenase-2 (COX-2) inhibitors
David Schwalb
Bioorganic & Medicinal Chemistry Letters, 2004
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Synthesis and Cyclooxygenase-2 (COX-2) Inhibiting Properties of 1,5- Diarylpyrazoles Possessing N-Substitution on the Sulfonamide (-SO2NH2) Moiety †
Venugopal Veeramaneni , Seshagiri Casturi , Parimal Misra
Letters in Drug Design & Discovery, 2005
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Synthesis, biological evaluation and molecular modeling study of pyrazole and pyrazoline derivatives as selective COX-2 inhibitors and anti-inflammatory agents. Part 2
Adel Azab
Bioorganic & medicinal chemistry, 2012
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Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)
John Talley
Journal of Medicinal Chemistry, 1997
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Parimal Misra
European Journal of Medicinal Chemistry, 2005
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Venugopal Veeramaneni
ChemInform, 2005
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shimaa Alhamaky
Bioorganic Chemistry, 2019
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yesim ozkan
Turk J Chem
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3,4-diarylpyrazoles: Potent and selective inhibitors of cyclooxygenase-2
Steven Kramer
Bioorganic & Medicinal Chemistry Letters, 1997
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Synthesis and Biologic Evaluation of Substituted 5-methyl-2-phenyl-1H-pyrazol-3(2H)-one Derivatives as Selective COX-2 Inhibitors: Molecular Docking Study
YOGESH V . USHIR
CBDD, 2014
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Synthesis and biological evaluation of a new class of acyl derivatives of 3-amino-1-phenyl-4,5-dihydro-1H-pyrazol-5-one as potential dual cyclooxygenase (COX-1 and COX-2) and human lipoxygenase (5-LOX) inhibitors
Paolo Bernardi
Il Farmaco, 2005
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Shoumyo Bhattacharya
European Journal of Medicinal Chemistry, 2014
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Mohammed Hawash
Journal of Chemistry
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Synthesis and Cyclooxygenase-2 Inhibiting Property of 1,5-Diarylpyrazoles with Substituted Benzenesulfonamide Moiety as Pharmacophore: Preparation of Sodium Salt for Injectable Formulation†
Rao Mamidi
Journal of Medicinal Chemistry, 2003
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Synthesis of 4-alkyl-1,2-diphenyl-3,5-dioxopyrazolidines possessing aryl methylsulfonyl and sulfonamide pharmacophores for evaluation as selective cyclooxygenase-2 (COX-2) inhibitors
Edward E Knaus
Journal of Heterocyclic Chemistry, 2002
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Methanesulfonamide group at position-4 of the C-5-phenyl ring of 1,5-diarylpyrazole affords a potent class of cyclooxygenase-2 (COX-2) inhibitors
Seshagiri Casturi
Bioorganic & Medicinal Chemistry Letters, 2004
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Synthesis of 1-P-SULF Am Ylphen YL-3 Trifluoromethylpyrazoles Class of CYCLOOXYGENASE-2 Inhibitors
HASSAN ALBAR
Heterocyclic Communications, 2003
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Jelena Penjišević
Bioorganic & Medicinal Chemistry Letters, 2014
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Pramod Hegde
Bioorganic & Medicinal Chemistry, 2004
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Beatrice Severino
Bioorganic & Medicinal Chemistry, 2010
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Rahmat Ali
Oriental journal of chemistry, 2015
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mohamed abdelgawad
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Design, synthesis, and biological evaluation of substituted hydrazone and pyrazole derivatives as selective COX2 inhibitors: Molecular docking study
naglaa abdel-aziz
Bioorganic & Medicinal Chemistry, 2011
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Laxman Adsul
Bioorganic & Medicinal Chemistry Letters, 2012
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2,3-Diarylpyran-4-ones: a new series of selective cyclooxygenase-2 inhibitors
Shin Chung
Bioorganic & Medicinal Chemistry Letters, 2004
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Novel Anti-inflammatory Agents Based on Pyrazole Based Dimeric Compounds; Design, Synthesis, Docking and in Vivo Activity
Ved Singh
Chemical & Pharmaceutical Bulletin, 2010
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Suchita Warangkar
Bioorganic & Medicinal Chemistry, 2010
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Design and Synthesis of Benzimidazole Analogs Endowed with Oxadiazole as Selective COX-2 Inhibitor
abuzer Ali
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Nagy Khalifa
PubMed, 2012
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Cyclooxygenase-2 inhibitors. 1, 5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/ …
Fabrizio Manetti
Journal of medicinal …, 2007
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