Y-26763: ATP-sensitive K+ channel activation and the inhibition of insulin release from human pancreatic β-cells (original) (raw)

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The antidiabetic sulfonylurea glibenclamide is a potent blocker of the ATP-modulated K+ channel in insulin secreting cells

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A Novel Enhancer of Insulinotrophic Action by High Glucose (JTT-608) Stimulates Insulin Secretion from Pancreatic β-Cells via a New Cellular Mechanism

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Antidiabetic sulfonylurea stimulates insulin secretion independently of plasma membrane KATP channels

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PIP2 and ATP cooperatively prevent cytosolic Ca2+-induced modification of ATP-sensitive K+ channels in rat pancreatic beta-cells

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ATP-Sensitive K+ Channel-Dependent Regulation of Glucagon Release and Electrical Activity by Glucose in Wild-Type and SUR1-/- Mouse -Cells

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3-(Alkylamino)-4H-pyrido[4,3-e]1,2,4-thiadiazine 1,1-dioxides as powerful inhibitors of insulin release from rat pancreatic B-cells: a new class of potassium channel openers?

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Mechanism of Cloned ATP-sensitive Potassium Channel Activation by Oleoyl-CoA

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3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-Dioxides as ATP-Sensitive Potassium Channel Openers: Effect of 6,7-Disubstitution on Potency and Tissue Selectivity

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Structural Nucleotide Analogs Are Potent Activators/Inhibitors of Pancreatic Cell KATP Channels: An Emerging Mechanism Supporting Their Use as Antidiabetic Drugs

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The Imidazoline RX871024 Stimulates Insulin Secretion in Pancreatic β-Cells from Mice Deficient in KATP Channel Function

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Sulfonylurea Blockade of KATP Channels Unmasks a Distinct Type of Glucose-Induced Ca2+ Decrease in Pancreatic β-Cells

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2006, ATP-Sensitive K+ Channels Current and Putative Target for the Prevention

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Characterization of ATP-Sensitive Potassium Channel-Blocking Activity of ZENECA ZM 181,037, a Eukalemic Diuretic

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Beneficial effects of K-ATP channel openers in diabetes: an update on mechanisms and clinical experiences

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Concentration-dependent effects of tolbutamide, meglitinide, glipizide, glibenclamide and diazoxide on ATP-regulated K+ currents in pancreatic B-cells

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Y-26763: ATP-sensitive K+ channel activation and the inhibition of insulin release from human pancreatic β-cells (original) (raw)

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