Differential Modification of the Interaction of Cardiac Muscarinic Cholinergic and β-Adrenergic Receptors with a Guanine Nucleotide Binding Component(s). (original) (raw)

Assessment of ternary model for the binding of agonists to neurohumoral receptors

Michael Sole

Biochemistry, 1986

View PDFchevron_right

Cardiac muscarinic receptor binding is regulated by Na+ and guanine nucleotides

William Roeske

Journal of Biological Chemistry

View PDFchevron_right

Rat brain and heart muscarinic receptors: Modification with tetranitromethane

David Gurwitz

Biochemical and Biophysical Research Communications, 1985

View PDFchevron_right

Assessment of mechanistic proposals for the binding of agonists to cardiac muscarinic receptors

Michael Sole

Biochemistry, 1986

View PDFchevron_right

The regulation of cardiac α1-adrenergic receptors by guanine nucleotides and by muscarinic cholinergic agonists

William Roeske

European Journal of Pharmacology, 1980

View PDFchevron_right

Cardiac cholinergic muscarinic receptors: changes in multiple affinity forms with down-regulation

Robert Roskoski

The Journal of pharmacology and experimental therapeutics, 1985

View PDFchevron_right

Differences in affinities of muscarinic acetylcholine receptor antagonists for brain and heart receptors

Elaine M Jagoda

Biochemical Pharmacology, 1983

View PDFchevron_right

Publication 11_Pharm Biochem Beh 29 (1988).pdf

Joseph Wettstein

View PDFchevron_right

Coupling of muscarinic receptors to adenylate cyclase in the rabbit myocardium: Effects of receptor inactivation

Frederick Ehlert

Journal of Pharmacology and Experimental Therapeutics

View PDFchevron_right

A simple method for estimation of agonist activity at GPCRs: characterization of responses elicited by M 2 and M 3 muscarinic receptors

Frederick Ehlert

The FASEB Journal, 2008

View PDFchevron_right

The muscarinic receptor of heart cell membranes Association with agonists, antagonists and antiarrhythmic agents

Michel Lazdunski

FEBS Letters, 1977

View PDFchevron_right

Molecular distinction between calf heart and brain muscarine receptors: Different N-ethylmaleimide modulation of agonist binding

Louis Kanarek

European Journal of Pharmacology, 1986

View PDFchevron_right

Problems associated with the application of the Cheng-Prusoff relationship to estimate atropine affinity constants using functional tissue responses

Roger Whiting

Life Sciences, 1989

View PDFchevron_right

Cooperativity and Oligomeric Status of Cardiac Muscarinic Cholinergic Receptors †

Paul Park

Biochemistry, 2002

View PDFchevron_right

Cardic muscarinic receptors. Biochemical identification and characterization

William Roeske

Journal of Biological Chemistry

View PDFchevron_right

Promiscuous or heterogeneous muscarinic receptors in rat atria? I. Schild analysis with simple competitive antagonists

Terry Kenakin

European Journal of Pharmacology, 1990

View PDFchevron_right

Regulation of muscarinic receptor binding by guanine nucleotides and N-ethylmaleimide

Frederick Ehlert

Journal of supramolecular structure, 1980

View PDFchevron_right

Analysis of Functional Responses at G Protein-Coupled Receptors: Estimation of Relative Affinity Constants for the Inactive Receptor Sstate

Frederick Ehlert

2011

View PDFchevron_right

Haga, K., Haga, T. & Ichiyama, A. Reconstitution of the muscarinic acetylcholine receptor. Guanine nucleotide-sensitive high affinity binding of agonists to purified muscarinic receptors reconstituted with GTP-binding proteins (Gi and Go). J. Biol. Chem. 261, 10133-10140

T. Haga

Journal of Biological Chemistry

View PDFchevron_right

Effects of an alkylating derivative of oxotremorine (BM 123A) on heart rate, muscarinic receptors and adenylate cyclase activity in the rabbit myocardium

Frederick Ehlert

Journal of Pharmacology and Experimental Therapeutics

View PDFchevron_right

Distribution of mRNA and binding sites of adrenoceptors and muscarinic receptors in the rat heart

Miklós Palkovits

Life Sciences, 2006

View PDFchevron_right

Estimation of Agonist Activity at G Protein-Coupled Receptors: Analysis of M2 Muscarinic Receptor Signaling through Gi/o,Gs, and G15

Frederick Ehlert

Journal of Pharmacology and Experimental Therapeutics, 2007

View PDFchevron_right

Efficacy of beta 1-adrenergic receptors is lower than that of beta 2-adrenergic receptors

Finn Olav Levy

Proceedings of the National Academy of Sciences, 1993

View PDFchevron_right

Graphical analysis of data from pharmacology experiments

Enric I. Canela

Pharmacological Research, 1992

View PDFchevron_right

Publication 22_Pharm Biochem Beh 41 (1992).pdf

Joseph Wettstein

View PDFchevron_right

The measurement of efficacy in the drug discovery agonist selection process

Terry Kenakin

Journal of Pharmacological and Toxicological Methods, 1999

View PDFchevron_right

Muscarinic receptor subtypes in bovine adrenal medulla

Jose Aguilar

Biochemical Pharmacology, 1986

View PDFchevron_right

Analysis of Functional Responses at G Protein-Coupled Receptors: Estimation of Relative Affinity Constants for the Inactive Receptor State

Frederick Ehlert

Journal of Pharmacology and Experimental Therapeutics, 2011

View PDFchevron_right

Guanine nucleotide-induced positive cooperativity in muscarinic-cholinergic antagonist binding

J. ADOLFO GARCÍA-SÁINZ

Biochemical and Biophysical Research Communications, 1986

View PDFchevron_right

Molecular size of muscarinic acetylcholine receptors of rat brain

T. Haga

FEBS Letters, 1980

View PDFchevron_right

Partial functional reconstitution of the cardiac muscarinic cholinergic receptor

William Roeske

Journal of Biological Chemistry

View PDFchevron_right

Evaluation of an agonist index: affinity ratio for compounds active on muscarinic cholinergic M2 receptors

Seyed Khosrow Tayebati

Journal of Autonomic Pharmacology, 1999

View PDFchevron_right

Adrenoceptors in GtoPdb v.2021.3

Douglas Eikenburg

IUPHAR/BPS guide to pharmacology CITE, 2021

View PDFchevron_right