Critical Molecular Determinants of α7 Nicotinic Acetylcholine Receptor Allosteric Activation (original) (raw)
Critical molecular determinants of α7 nicotinic acetylcholine receptor allosteric activation: separation of direct allosteric activation and positive allosteric modulation
Ganesh Chaturbhuj
Journal of Biological Chemistry, 2016
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Molecular blueprint of allosteric binding sites in a homologue of the agonist-binding domain of the α7 nicotinic acetylcholine receptor
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ACS Chemical Biology, 2012
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Steven m. M Sine
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Critical Elements Determining Diversity in Agonist Binding and Desensitization of Neuronal Nicotinic Acetylcholine Receptors
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1998
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Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant β Subunits Acquire Sensitivity to α7-Selective Positive Allosteric Modulators
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LY2087101 and dFBr share transmembrane binding sites in the (α4)3(β2)2 Nicotinic Acetylcholine Receptor
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A Novel Pharmatope Tag Inserted into the 4 Subunit Confers Allosteric Modulation to Neuronal Nicotinic Receptors
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