An Efficient Synthesis of the Taxane-Derived Anticancer Agent ABT-271 (original) (raw)
Preface, Brief History of the Discovery and Development of Taxane Anticancer Agents ( 1-3 )
Iwao Ojima
ACS Symposium Series, 1994
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William Rose
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IUBMB Life (International Union of Biochemistry and Molecular Biology: Life), 2002
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Michael Rasmussen
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Maria Aparecida Nicoletti
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International Journal of Cancer, 1997
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A ready synthesis of intermediates containing the A-ring substructure of taxol: a Diels-Alder route to the B-seco taxane series. [Erratum to document cited in CA117(3):26833h]
William Bornmann
J Org Chem, 1993
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ChemInform Abstract: New Strategy for the Synthesis of the Taxane Diterpenes: Formation of the BC-Rings of Taxol via a (5 + 2) Pyrylium Ylide-Alkene Cyclization, Ring Expansion Strategy
Jim Tarrant
ChemInform, 2010
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Ezio Bombardelli
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Synthetic studies on taxane diterpenes X-ray structure of a key intermediate
Isaac Hanna
Tetrahedron, 1984
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Evaluation of 2-Bromocyclohexenone Acetals as Vehicles for the Introduction of C-7 Oxygen Preliminary to the Synthesis of Taxane Diterpenes
Francis Montgomery
The Journal of Organic Chemistry, 1995
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A convergent synthesis of functionalized B-seco taxane skeletons
Christian Montalbetti
Tetrahedron Letters, 1995
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A ready synthesis of intermediates containing the A-ring substructure of taxol: a Diels-Alder route to the B-seco taxane series
William Bornmann
The Journal of Organic Chemistry, 1992
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TaxKB: a knowledge base for new taxane-related drug discovery
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BioData Mining, 2015
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Taxol Semisynthesis: A Highly Enantio- and Diastereoselective Synthesis of the Side Chain and a New Method for Ester Formation at C-13 Using Thioesters
Nicola Mongelli
The Journal of Organic Chemistry, 1997
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Second Generation Taxanes: from the Natural Framework to the Challenge of Drug Resistance
E. Bombardelli, M. Distefano
Current Medicinal Chemistry-Anti-Cancer Agents, 2003
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A Novel Hydroxylation Step in the Taxane Biosynthetic Pathway: A New Approach to Paclitaxel Production by Synthetic Biology
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Frontiers in Bioengineering and Biotechnology, 2020
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Taxane diterpenes 5: Synthesis of the A- and C-rings: An unusual rearrangement of an N-hydroxyimino lactone
Patrick Linnane
Tetrahedron, 1999
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Facile access to the ABC ring system of the taxane diterpenes via anionic oxy-Cope rearrangements
James White
Tetrahedron, 1995
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The Chemistry of the Taxane Diterpene: Stereoselective Reductions of Taxanes
Dinah Dutta
Journal of Organic Chemistry, 1998
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Site-specific enzymatic hydrolysis of taxanes at C-10 and C-13
Ramesh Patel
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Anticancer regimens containing third generation taxanes SB-T-121605 and SB-T-121606 are highly effective in resistant ovarian carcinoma model
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Antitumour activity of novel taxanes that act at the same time as cytotoxic agents and P-glycoprotein inhibitors
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British Journal of Cancer, 2000
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