Glutathione S -transferase (GST) inhibitors
Nisha Mathew
Expert Opinion on Therapeutic Patents, 2006
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Molecular Modeling, Synthesis, and Preliminary Biological Evaluation of Glutathione-S-Transferase Inhibitors as Potential Therapeutic Agents
Sante Cundari
Journal of Medicinal Chemistry, 2005
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A novel method for screening the glutathione transferase inhibitors
Grzegorz Węgrzyn
BMC Biochemistry, 2009
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Potent and Selective Inhibitors of Glutathione S -Transferase Omega 1 That Impair Cancer Drug Resistance
Timothy Spicer
Journal of the American Chemical Society, 2011
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Characterization of new potential anticancer drugs designed to overcome glutathione transferase mediated resistance
Miyuki Shimoji, Carolien Schophuizen
Molecular pharmaceutics, 2011
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Structural Basis for the Binding of the Anticancer Compound 6-(7-Nitro-2,1,3-Benzoxadiazol-4-Ylthio)Hexanol to Human Glutathione S-Transferases
Caccuri, Caccuri
Cancer Research, 2009
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Glutathione-S-transferase Activates Novel Alkylating Agents
Colby Caldwell
Journal of Medicinal Chemistry, 1994
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Glutathione S-transferases, structure, regulation, and therapeutic implications
Thomas Rushmore
Journal of Biological Chemistry, 1993
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Structural insights into omega-class glutathione transferases: a snapshot of enzyme reduction and identification of a non-catalytic ligandin site
Aaron Oakley
PloS one, 2013
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Design of a monomeric human glutathione transferase GSTP1, a structurally stable but catalytically inactive protein
John Tainer
Protein Engineering Design and Selection, 2002
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FDA-approved drugs and other compounds tested as inhibitors of human glutathione transferase P1-1.
yasemin aksoy
Chemico-biological ınteractions
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Structural Analysis of a Glutathione Transferase A1-1 Mutant Tailored for High Catalytic Efficiency with Toxic Alkenals
Bengt Mannervik
Biochemistry, 2009
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The Structures of Human Glutathione Transferase P1-1 In Complex With Glutathione and Various Inhibitors at High Resolution1
Aaron Oakley
Journal of molecular …, 1997
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Mutational Analysis of the Binding of Alternative Substrates and Inhibitors to the Active Site of Human Glutathione Transferase P1–1
aram ismail
Processes
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Sulphonamide-based bombesin prodrug analogues for glutathione transferase, useful in targeted cancer chemotherapy
Nikolaos Labrou
European Journal of Medicinal Chemistry, 2009
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The structures of human glutathione transferase P1-1 in complex with glutathione and various inhibitors at high resolution
Hugo Villar
Journal of Molecular Biology, 1997
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The Anti-cancer Drug Chlorambucil as a Substrate for the Human Polymorphic Enzyme Glutathione Transferase P1-1: Kinetic Properties and Crystallographic Characterisation of Allelic Variants
Aaron Oakley
Journal of Molecular Biology, 2008
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Human Theta Class Glutathione Transferase: the Crystal Structure Reveals a Sulfate-Binding Pocket Within a Buried Active Site
Aaron Oakley
Structure, 1998
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Synthesis and Biological Evaluation of 2-Substituted-5-(4-nitrophenylsulfonamido)benzoxazoles as Human GST P1-1 Inhibitors, and Description of the Binding Site Features.
yasemin aksoy
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Mechanistic evaluation and transcriptional signature of a glutathione S-transferase omega 1 inhibitor
Vladimir Yarovenko
Nature communications, 2016
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The Three-Dimensional Structure of the Human Pi Class Glutathione Transferase P1-1 in Complex with the Inhibitor Ethacrynic Acid and Its Glutathione Conjugate
Caccuri, Caccuri
Biochemistry, 1997
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Human glutathione transferase A4-4 crystal structures and mutagenesis reveal the basis of high catalytic efficiency with toxic lipid peroxidation products
Bengt Mannervik
Journal of Molecular Biology, 1999
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Synthesis and structure--activity relationship of new cytotoxic agents targeting human glutathione-S-transferases
Domenico Tarantino
European journal of medicinal chemistry, 2015
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The structures of human glutathione transferase P1-1 in complex with glutathione and various inhibitors at high resolution 1 1 Edited by R. Huber
Aaron Oakley
Journal of Molecular Biology, 1997
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Identifying and Characterizing Binding Sites on the Irreversible Inhibition of Human Glutathione S-Transferase P1-1 by S-Thiocarbamoylation
Juan Manuel Casas-Solvas
ChemBioChem, 2012
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Inhibition of human glutathione transferase P1-1 by novel benzazole derivatives | İnsan glutatyon transferaz P1-1'in benzozol türevleri tarafi{dotless}ndan inhibisyonu
Usama Hegazy
Turkish Journal of Biochemistry-Turk Biyokimya Dergisi, 2012
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Glutathione Transferases: Potential Targets to Overcome Chemoresistance in Solid Tumors
Ana Savic-Radojevic
International Journal of Molecular Sciences
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