Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor-α or Estrogen Receptor-β* (original) (raw)
Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-{alpha} or estrogen receptor-{beta}
John Katzenellenbogen
Endocrinology, 1999
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Differential estrogen receptor subtype modulators: Assessment of estrogen receptor subtype-binding selectivity and transcription-regulating properties of new …
Xanthippi Alexi
The Journal of Steroid …, 2009
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Differential estrogen receptor subtype modulators: assessment of estrogen receptor subtype-binding selectivity and transcription-regulating properties of new cycloalkyl pyrazoles
Aggeliki Meligova
The Journal of steroid biochemistry and molecular biology, 2009
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Antagonists Selective for Estrogen Receptor
John Katzenellenbogen
Endocrinology, 2002
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The nature of the ligand-binding pocket of estrogen receptor alpha and beta: The search for subtype-selective ligands and implications for the prediction of estrogenic …
Rajeev Muthyala
Pure and Applied Chemistry, 2003
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A New Series of Estrogen Receptor Modulators That Display Selectivity for Estrogen Receptor β
Shawn Williams
Journal of Medicinal Chemistry, 2002
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Selective Estrogen Receptor Modulators; Role of Side Chain in Activity Modulation
Dinesh Dikshit
Asian Journal of Pharmaceutical and Clinical Research, 2014
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Design, synthesis and bioevaluation of novel candidate selective estrogen receptor modulators
Yogesh Yadav
European Journal of Medicinal Chemistry, 2011
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Estrogen receptor β selective ligands: Discovery and SAR of novel heterocyclic ligands
Kimberly Cameron
Bioorganic & Medicinal Chemistry Letters, 2005
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Estrogen receptor ligands. Part 14: Application of novel antagonist side chains to existing platforms
Lee-Yuh Pai
Bioorganic & Medicinal Chemistry Letters, 2005
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Characterization of the Pharmacophore Properties of Novel Selective Estrogen Receptor Downregulators (SERDs)
John Katzenellenbogen
Journal of Medicinal Chemistry, 2010
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Interactions of synthetic estrogens with human estrogen receptors
Matthewos Eshete
Journal of Endocrinology, 2001
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Differential activation of wild-type and variant forms of estrogen receptor α by synthetic and natural estrogenic compounds using a promoter containing three estrogen-responsive elements
L. Pallaroni
The Journal of Steroid Biochemistry and Molecular Biology, 2001
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Estrogen receptor stereochemistry: ligand binding and hormonal responsiveness
Kenneth Korach
Steroids, 1991
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Estrogenic diazenes: heterocyclic non-steroidal estrogens of unusual structure with selectivity for estrogen receptor subtypes
viswajanani sattigeri
Bioorganic & Medicinal Chemistry, 2003
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Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism
David Agard
Nature Structural & …, 2002
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Thiophene-Core Estrogen Receptor Ligands Having Superagonist Activity
Jian Min
Journal of Medicinal Chemistry, 2013
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Deconstructing estradiol: Removal of B-ring generates compounds which are potent and subtype-selective estrogen receptor agonists
muhammad asim
Bioorganic & Medicinal Chemistry Letters, 2009
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Amphipathic Benzenes Are Designed Inhibitors of the Estrogen Receptor α/Steroid Receptor Coactivator Interaction
John Katzenellenbogen
ACS Chemical Biology, 2008
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Salicylaldoximes and anthranylaldoximes as alternatives to phenol-based estrogen receptor ligands
Tiziano Tuccinardi
Arkivoc, 2006
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3,5-Diphenylpyrazolylethanone Derivatives as Selective Estrogen Receptor Modulators: Design, Synthesis, Biological Evaluation and Docking Analysis
Vivekanand Chatpalliwar
Indo Global Journal of Pharmaceutical Sciences, 2020
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Structure-Based Approach for the Discovery of Novel Selective Estrogen Receptor Modulators
Camillo Rosano
Current Medicinal …, 2011
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Optimisation of estrogen receptor subtype-selectivity of a 4-Aryl-4H-chromene scaffold previously identified by virtual screening
Daniela Zisterer
Bioorganic & Medicinal Chemistry, 2019
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Triaryl-Substituted Schiff Bases Are High-Affinity Subtype-Selective Ligands for the Estrogen Receptor
Chune Dong
Journal of Medicinal Chemistry, 2014
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Lead identification of a potent benzopyranone selective estrogen receptor modulator
Deborah Mortensen
Bioorganic & Medicinal Chemistry Letters, 2004
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Estrogen receptor β ligands: Recent advances and biomedical applications
Filippo Minutolo
Medicinal Research Reviews, 2009
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