A Novel Protecting/Activating Strategy for β-Hydroxy Acids and Its Use in Convergent Peptide Synthesis † (original) (raw)

Synthesis and application of acid labile anchor groups for the synthesis of peptide amides by Fmoc-solid-phase peptide synthesis

Jochen Knolle

International journal of peptide and protein research, 1989

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An Improved Procedure for N- to C-Directed (Inverse) Solid-Phase Peptide Synthesis

Gunnar Lindeberg

Journal of Combinatorial Chemistry, 2000

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Preparation and Applications of Xanthenylamide (XAL) Handles for Solid-Phase Synthesis of C-Terminal Peptide Amides under Particularly Mild Conditions1-3

George Barany

The Journal of Organic Chemistry, 1996

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Facile solid-phase synthesis of C-terminal peptide aldehydes and hydroxamates from a common Backbone Amide-Linked (BAL) intermediate*†

Sharon Gazal, Larry R . Masterson

The Journal of Peptide Research, 2008

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Application of N-(tert-butyloxycarbonyl)amino acid N-carboxyanhydrides in solid-phase peptide synthesis

Fred Naider

The Journal of Organic Chemistry, 1993

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Facile solid-phase synthesis of C-terminal peptide aldehydes and hydroxamates from a common Backbone Amide-Linked (BAL) intermediate*†: Synthesis of peptide aldehydes and hydroxamates

Larry R . Masterson

Journal of Peptide Research, 2008

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Synthesis of 5-(((R,S)-5-((9-Fluorenylmethoxycarbonyl)amino)-10,11-dihydrodibenzo[a,d]cyclohepten-2-yl)oxy)valeric Acid (CHA) and 5-(((R,S)-5-((9-Fluorenylmethoxycarbonyl)amino)dibenzo[a,d]-cyclohepten-2-yl)oxy)valeric Acid (CHE) Handles for the Solid-Phase Synthesis of C-Terminal Peptide Amides ...

Kiyoshi Nokihara

The Journal of Organic Chemistry, 1994

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Fundamentals of Modern Peptide Synthesis

Jean-alain Fehrentz

ChemInform, 2006

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Cyclohexyloxycarbonyl based orthogonal solid phase peptide synthesis in Boc chemistry

Ferenc Hudecz

Tetrahedron, 1998

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A new flourene-derived anchor for solid-phase synthesis of protected peptides

Francesc Rabanal

Tetrahedron Letters, 1992

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Tetrahydropyranyl: A Non-aromatic, Mild-Acid-Labile Group for Hydroxyl Protection in Solid-Phase Peptide Synthesis

Hortensia Maria Rodriguez Cabrera

ChemistryOpen, 2017

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Direct cleavage of peptides from a solid support into aqueous buffer. Application in simultaneous multiple peptide synthesis

Rhonda Campbell

The Journal of Organic Chemistry, 1991

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Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C-Terminal-Modified and Cyclic Peptides1,2,3

George Barany

Journal of the American Chemical Society, 1998

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Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides

Walter Cabri

ACS Sustainable Chemistry & Engineering, 2019

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Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C-Terminal-Modified and Cyclic Peptides 1 , 2 , 3

Josef Vagner

Journal of the American Chemical Society, 1998

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Aqueous solid-phase peptide synthesis (ASPPS): A novel concept of peptide synthesis

Sascha Knauer

2020

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4-Alkoxy-2-hydroxybenzaldehyde (AHB): A Versatile Aldehyde Linker for Solid-Phase Synthesis of C-Terminal Modified Peptides and Peptidomimetics †

Victor Hruby

Organic Letters, 2000

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A New Strategy To Produce β-Peptides: Use of Alicyclic β-Lactams

Ferenc Fülöp

Organic Letters, 2004

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Direct access to side chain N,N′-diaminoalkylated derivatives of basic amino acids suitable for solid-phase peptide synthesis

Predrag Cudic

Amino Acids, 2013

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2-(2,4-DINITROPHENYL)ETHYLOXYCARBONYL-AMINO Acids, New Base Labile Protected Derivatives Suitable for Solid-Phase Peptide Synthesis

Ramon Eritja

Tetrahedron Letters, 1992

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Synthesis of peptides with α,β-dehydroamino acids, VI. Synthesis ofN-benzyloxycarbonyl andN-trifluoroacetyl dipeptides of α,β-dehydro-butyrine, -valine, -leucine, and -isoleucine

Piotr Wieczorek

Liebigs Annalen der Chemie, 1988

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N-2-(2,4-Dinitrophenyl)ethyloxycarbonyl Amino Acids, New Base Labile Protected Derivatives Suitable for Solid-Phase Peptide Synthesis

Ramon Eritja

Cheminform, 1993

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Synthesis of N-carboxyalkyl and N-aminoalkyl functionalized dipeptide building units for the assembly of backbone cyclic peptides

Diana Imhof

Journal of Peptide Research, 1999

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Acetophenone-based linker for solid-phase peptide synthesis

thao nguyen

Journal of Peptide Science, 2000

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Selective deprotection of the N.alpha.-tert-butyloxycarbonyl group in solid phase peptide synthesis with chlorotrimethylsilane in phenol

Francis Picart

Journal of Organic Chemistry, 1993

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The synthesis of ‘difficult’ peptides using 2-hydroxy-4-methoxybenzyl or pseudoproline amino acid building blocks: a comparative study

Nicholas Ede

Journal of Peptide Science, 1999

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High Throughput Synthesis of Peptides and Peptidomimetics

Victor Hruby is to

ChemInform, 2007

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