original ) (raw )Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands
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Bioorganic & Medicinal Chemistry Letters, 2010
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Novel cyclohexyl amides as potent and selective D 3 dopamine receptor ligands
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Bioorganic & Medicinal Chemistry Letters, 1997
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A solid phase parallel synthesis of diverse amides as dopamine D 3 receptor ligands
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Journal of Enzyme Inhibition and Medicinal Chemistry, 2008
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New generation dopaminergic agents. 5. heterocyclic bioisosteres that exploit the 3-OH-N1-phenylpiperazine dopaminergic template
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Bioorganic & Medicinal Chemistry Letters, 1998
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Bioorganic & Medicinal Chemistry, 2013
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MedChemComm, 2013
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Enantiospecific synthesis and receptor binding of novel dopamine receptor ligands employing natural 4-hydroxyproline as a practical and flexible building block
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Tetrahedron: Asymmetry, 2003
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Synthesis and evaluation of several cathechol bioisosteres as potential dopamine receptor ligands
Vukic Soskic
Bioorganic & Medicinal Chemistry Letters, 1991
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Novel Heterocyclic Trans Olefin Analogues of N-{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as Selective Probes with High Affinity for the Dopamine D3 Receptor
Christina bennett
Journal of Medicinal Chemistry, 2005
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Synthesis and dopaminergic properties of the two enantiomers of 3-(3,4-dimethylphenyl)-1-propylpiperidine, a potent and selective dopamine D4 receptor ligand
Filippo Minutolo
Bioorganic & Medicinal Chemistry Letters, 2001
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4-N-linked-heterocyclic piperidine derivatives with high affinity and selectivity for human dopamine D4 receptors
Paul D Leeson
Bioorganic & Medicinal Chemistry Letters, 1999
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Substituted 4-Aminopiperidines Having High In Vitro Affinity and Selectivity for the Cloned Human Dopamine D4 Receptor
Arthur Lopez
European journal of …, 1997
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Analogs of the dopamine D4 receptor ligand FAUC 113 with planar- and central-chirality
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Tetrahedron: Asymmetry, 2002
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Synthesis and SAR study of a novel series of dopamine receptor agonists
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Bioorganic & Medicinal Chemistry, 2014
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DOPAMINE D2 RECEPTOR ANTAGONIST ACTIVITY AND MOLECULAR MODELING OF CERTAIN NEW CYCLOHEXANE DERIVED ARYLCARBOXAMIDES …
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chalcogen.ro
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Synthesis and biological investigations of dopaminergic partial agonists preferentially recognizing the D4 receptor subtype
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Bioorganic & Medicinal Chemistry Letters, 2006
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New N - n -Propyl-Substituted 3Aryl and 3-Cyclohexylpiperidines as Partial Agonists at the D 4 Dopamine Receptor
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Journal of Medicinal Chemistry, 2003
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Functionally Selective Dopamine D 2 /D 3 Receptor Agonists Comprising an Enyne Moiety
Peter Gmeiner
Journal of Medicinal Chemistry, 2013
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Design and Synthesis of Bitopic 2Phenylcyclopropylmethylamine (PCPMA) Derivatives as Selective Dopamine D3 Receptor Ligands
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Fancy Bioisosteres: Novel Paracyclophane Derivatives As Super-Affinity Dopamine D3 Receptor Antagonists
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Journal of Medicinal Chemistry, 2006
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ChemInform Abstract: Heterocyclic Congeners of PD 128,907 with a Partially Hydrogenated Benzomorpholine Moiety as Potential Dopamine D3-Receptor Ligands
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Cheminform, 2010
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Tetrahedron, 1998
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Heterocyclic congeners of PD 128,907 with a partially hydrogenated benzomorpholine moiety as potential dopamine D3-receptor ligands
Holger Stark
European Journal of Medicinal Chemistry, 1999
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N - n -Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding Studies 1
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Journal of Medicinal Chemistry, 1998
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Discovery of selective dopamine D4 receptor antagonists: 1-Aryloxy-3-(4-aryloxypiperidinyl)-2-propanols
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Bioorganic & Medicinal Chemistry Letters, 1997
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Analogues of doxanthrine reveal differences between the dopamine D1 receptor binding properties of chromanoisoquinolines and hexahydrobenzo[a]phenanthridines
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N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 Receptor Selectivity
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Journal of Medicinal Chemistry, 2011
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Further Definition of the D1 Dopamine Receptor Pharmacophore: Synthesis of trans-6,6a,7,8,9,13b-Hexahydro-5H-benzo[d]naphth[2,1-b]azepines as Rigid Analogues of β-Phenyldopamine
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Journal of Medicinal Chemistry, 1997
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Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps
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Bioorganic & Medicinal Chemistry Letters, 1999
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Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligands
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Bioorganic & Medicinal Chemistry Letters, 2009
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