Novel 18F-labelled triazine derivatives for PET imaging of phosphodiesterase 2A (original) (raw)
Synthesis, 18F-Radiolabelling and Biological Characterization of Novel Fluoroalkylated Triazine Derivatives for in Vivo Imaging of Phosphodiesterase 2A in Brain via Positron Emission Tomography
Susann Schröder, Rodrigo Teodoro
Molecules, 2015
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Development of a fluorine-18-labeled benzoimidazotriazine-based radioligand for the imaging of phosphodiesterase 2A in the brain with positron emission tomography
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2020
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Preclinical Evaluation of 18F-PF-05270430, a Novel PET Radioligand for the Phosphodiesterase 2A Enzyme
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Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2016
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Radiosynthesis and Biological Investigation of a Novel Fluorine-18 Labeled Benzoimidazotriazine- Based Radioligand for the Imaging of Phosphodiesterase 2A with Positron Emission Tomography
RIEN RITAWIDYA
Molecules
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Synthesis and In Vitro Evaluation of 8-Pyridinyl-Substituted Benzo[e]imidazo[2,1-c][1,2,4]triazines as Phosphodiesterase 2A Inhibitors
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{"__content__"=>"Investigation of anF-labelled Imidazopyridotriazine for Molecular Imaging of Cyclic Nucleotide Phosphodiesterase 2A.", "sup"=>{"__content__"=>"18"}}
Rodrigo Carvalho Teodoro
Molecules (Basel, Switzerland), 2018
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Discovery and development of 11C-Lu AE92686 as a radioligand for PET imaging of phosphodiesterase10A in the brain
Claus Christoffersen
Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2014
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The Discovery of a Novel Phosphodiesterase (PDE) 4B-Preferring Radioligand for Positron Emission Tomography (PET) Imaging
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The Journal of Nuclear Medicine, 2014
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Carbon-11 and Fluorine-18 Radiolabeled Pyridopyrazinone Derivatives for Positron Emission Tomography (PET) Imaging of Phosphodiesterase-5 (PDE5)
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Journal of medicinal chemistry, 2016
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First-in-Human Evaluation of18F-PF-06445974, a PET Radioligand That Preferentially Labels Phosphodiesterase-4B
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Fluorine-Containing 6,7-Dialkoxybiaryl-Based Inhibitors for Phosphodiesterase 10 A: Synthesis and in vitro Evaluation of Inhibitory Potency, Selectivity, and Metabolism
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Journal of Nuclear Medicine, 2014
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Pyrido[4,3- e ][1,2,4]triazolo[4,3- a ]pyrazines as Selective, Brain Penetrant Phosphodiesterase 2 (PDE2) Inhibitors
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ACS Medicinal Chemistry Letters, 2015
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Synthesis, in vitro and in vivo evaluation of [O-methyl-11C] 2-{4-[4-(3-methoxyphenyl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]-triazine-3,5-dione: A novel agonist 5-HT1A receptor PET ligand
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