New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists (original) (raw)
1-Aryl-3,5-dihydro-4 H -2,3-benzodiazepin-4-ones: Novel AMPA Receptor Antagonists
Giovambattista Sarro
Journal of Medicinal Chemistry, 1997
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Synthesis and anticonvulsant activity of N-3 substituted 2,3-benzodiazepines
Giovambattista Sarro
Il Farmaco, 2004
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Synthesis of 7,8-(Methylenedioxy)-1-phenyl-3,5-dihydro-4 H -2,3-benzodiazepin- 4-ones as Novel and Potent Noncompetitive AMPA Receptor Antagonists
Sui Cai
Journal of Medicinal Chemistry, 1998
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New non competitive AMPA antagonists
István Tarnawa
Bioorganic & Medicinal Chemistry, 2000
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Discovery of a Novel and Highly Potent Noncompetitive AMPA Receptor Antagonist
Laura Luca
Journal of Medicinal Chemistry, 2003
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The non-competitive AMPA/kainate receptor antagonist, GYKI 52466, potentiates the anticonvulsant activity of conventional antiepileptics
Stanisław Czuczwar, Kinga Borowicz
European Journal of Pharmacology, 1995
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Comparative anticonvulsant activity of some 2,3-benzodiazepine derivatives in rodents
Giovambattista Sarro
Pharmacology Biochemistry and Behavior, 2003
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AMPA Receptor Antagonists as Potential Anticonvulsant Drugs
Laura Luca
Current Topics in Medicinal Chemistry, 2005
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Synthesis, Chiral Resolution, and Enantiopharmacology of a Potent 2,3Benzodiazepine Derivative as Noncompetitive AMPA Receptor Antagonist
Frank Menniti, Giovambattista Sarro
Journal of Medicinal Chemistry, 2006
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Synthesis and Evaluation of Some New (1,2,4) Triazolo(4,3-a)Quinoxalin-4(5H)-one Derivatives as AMPA Receptor Antagonists
adel ghiaty, Hamada S Abulkhair
Journal of Heterocyclic Chemistry, 2013
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Synthesis and Evaluation of Some New (1,2,4) Triazolo(4,3-a) Quinoxalin-4(5H)-one Derivatives as AMPA Receptor Antagonists Vol 50
Hamada S Abulkhair, adel ghiaty
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Quinazolinedione sulfonamides: A novel class of competitive AMPA receptor antagonists with oral activity
Joerg Kallen, Yves Auberson
Bioorganic & Medicinal Chemistry Letters, 2011
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Phthalazine-1,4-dione derivatives as non-competitive AMPA receptor antagonists: design, synthesis, anticonvulsant evaluation, ADMET profile and molecular docking
Khaled El Adl
Molecular Diversity, 2018
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Synthesis and anticonvulsant activity of novel and potent 1-aryl-7,8-methylenedioxy-1,2,3,5-tetrahydro-4 H-2,3-benzodiazepin-4-ones
Magdy Gineinah, Giovambattista Sarro
Bioorganic & Medicinal Chemistry Letters, 2001
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Neuroprotective and anticonvulsant effects of EGIS-8332, a non-competitive AMPA receptor antagonist, in a range of animal models
Adriana Rodrigues
British Journal of Pharmacology, 2007
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Influence of LY 300164, an AMPA/kainate receptor antagonist upon the anticonvulsant action of antiepileptic drugs against aminophylline-induced seizures in mice
Stanisław Czuczwar
2003
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Synthesis and anticonvulsant properties of 2,3,3a,4-tetrahydro-1H-pyrrolo[1,2-a]benzimidazol-1-ones
Giovambattista Sarro
Journal of Medicinal Chemistry, 1989
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Effects of some AMPA receptor antagonists on the development of tolerance in epilepsy-prone rats and in pentylenetetrazole kindled rats
Luca Gallelli
European Journal of Pharmacology, 1999
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New AMPA antagonists in epilepsy
Giovambattista Sarro
Expert Opinion on Investigational Drugs, 2012
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Competitive AMPA receptor antagonists
Daniela Catarzi, Flavia Varano, Vittoria Colotta
Medicinal Research Reviews, 2007
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Anticonvulsant Activity and Plasma Level of 2,3-Benzodiazepin-4-ones (CFMs) in Genetically Epilepsy-Prone Rats
Giovambattista Sarro
Pharmacology Biochemistry and Behavior, 1999
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Azirino[1, 2-d][1, 4]benzodiazepine derivatives and related 1,4-benzodiazepines as anticonvulsant agents in DBA/2 mice
Giovambattista Sarro
General Pharmacology: The Vascular System, 1996
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