[3H] pirenzepine selectively identifies a high affinity population of muscarinic cholinergic receptors in the rat cerebral cortex (original) (raw)

Comparison Between Purified Cerebral and Atrial Muscarinic Acetylcholine Receptors: Pirenzepine Binding and the Effect of Sulfhydryl Reagents

Gabriel Berstein

Biomedical Research, 1989

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Characterization of agonist and antagonist binding to muscarinic cholinergic receptors solubilized from rat cerebral cortex

Agneta Nordberg

Journal of Neural Transmission, 1988

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Inverse agonist activity of pirenzepine at M 2 muscarinic acetylcholine receptors

Fabien Schmidlin

British Journal of Pharmacology, 1999

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Loss of pirenzepine regional selectivity following solubilization and partial purification of the putative M1 and M2 muscarinic receptor subtypes

Elliot Gershon

Molecular Brain Research, 1987

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Interaction of Psychotropic Drugs with Brain Muscarinic Cholinoceptors: Similarities of Biperiden with Pirenzepine in Receptor Binding Properties

Erkka Syvälahti

Pharmacology & Toxicology, 1987

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Autoradiographic localization of peripheral M1 muscarinic receptors using [3H]pirenzepine

Noel J Buckley

Brain Research, 1986

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Functional and biochemical basis for multiple muscarinic acetylcholine receptors

William Roeske

Progress in Neuro-Psychopharmacology and Biological Psychiatry, 1985

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Pirenzepine-insensitive muscarinic autoreceptors regulate acetylcholine release in human neocortex

Mario Marchi

Brain Research, 1990

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The properties of cholinergic muscarinic receptor sites from bovine atria reconstituted after solubilization

Jose Aguilar

Neurochemistry International, 1987

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High-affinity [3H]pirenzepine binding to putative M1 muscarinic sites in the neuroblastoma × glioma hybrid cell line (NG 108-15)

William Roeske

Biochemical and Biophysical Research Communications, 1984

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Autoradiography of muscarinic cholinergic receptors in cortical and subcortical brain regions of C57BL/6 and DBA/2 mice

Alberto Oliverio

Neurochemical Research, 1992

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Assessment of Novel Muscarinic Acetylcholine Receptors in Rat Cerebral Cortex by a Tissue Segment Binding Method

Atsushi Nishimune

Journal of Pharmacological Sciences, 2010

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The N4 nitrogen of pirenzepine is responsible for selective binding of the M1 subtype human muscarinic receptor

Nicholas Murgolo

Bioorganic & Medicinal Chemistry Letters, 1996

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Evidence for Multiple Muscarinic Receptor Subtypes in Human Brain

Martin Rossor

Journal of Neurochemistry, 1984

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Agonist and Antagonist Binding of Muscarinic Acetylcholine Receptors Purified from Porcine Brain: Interconversion of High- and Low-Affinity Sites by Sulfhydryl Reagents

T. Haga

Journal of Neurochemistry, 1988

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Muscarinic receptors on cultured cells of rat hippocampus: cholinergic regulation and presence of subtypes

Flavio Keller

European Journal of Pharmacology, 1989

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Mapping muscarinic receptors in human and baboon brain using [N-11C-methyl]-benztropine

Jonathan Brodie

Synapse, 1990

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Functional and direct binding studies using subtype selective muscarinic receptor antagonists

Roger Whiting

British Journal of Pharmacology, 1988

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Degradation of Rat Brain Cholinergic Muscarinic Receptors In Vitro: Enhancement by Agonists and Inhibition by Antagonists

Robert Roskoski

Journal of Neurochemistry, 1985

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Muscarinic cholinergic receptors in the rat deep cerebellar nuclei: a quantitative autoradiographic study

A. Beitz

Neuroscience letters, 1984

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[3H]Pirenzepine identifies putative M1 muscarinic receptors in human stellate ganglia

William Roeske

Brain Research, 1984

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Calcium-dependent pirenzepine-sensitive muscarinic response in the rat hippocampal slice

Bradley Alger

Neuroscience Letters, 1988

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Partial functional reconstitution of the cardiac muscarinic cholinergic receptor

William Roeske

Journal of Biological Chemistry

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Differences in affinities of muscarinic acetylcholine receptor antagonists for brain and heart receptors

Elaine M Jagoda

Biochemical Pharmacology, 1983

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Cardiac cholinergic muscarinic receptors: changes in multiple affinity forms with down-regulation

Robert Roskoski

The Journal of pharmacology and experimental therapeutics, 1985

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Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors

Vladimír Doležal

Scientific Reports

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Effects of (±)-huprine Y and (±)-huprine Z, two new anticholinesterasic drugs, on muscarinic receptors

Diego Muñoz-torrero

Neuroscience Letters, 2005

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Modulation of Muscarinic Cholinergic Receptor Affinity for Antagonists in Rat Heart

McHardy Smith

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Quantitative distribution of muscarinic receptors and choline acetyltransferase in rat medulla: examination of transmitter-receptor mismatch

Paul Ernsberger

Brain research, 1988

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Pirenzepine Promotes the Dimerization of Muscarinic M1 Receptors through a Three-step Binding Process

Raja Chinnappan

Journal of Biological Chemistry, 2009

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Repeated effects of asenapine on adrenergic and cholinergic muscarinic receptors

Erik Wong

The International …, 2010

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Cooperativity and Oligomeric Status of Cardiac Muscarinic Cholinergic Receptors †

Paul Park

Biochemistry, 2002

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