Side Reaction of Significance in Preparation of Peptide- or Peptidomimetic-Based Hydroxamate Enzyme Inhibitors (original) (raw)

Hydroxamate inhibitors of the matrix metallo-proteinases (MMPs) containing novel P1′ heteroatom based modifications

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Bioorganic & Medicinal Chemistry Letters, 1997

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Journal of Medicinal Chemistry, 1995

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M. Caldarelli

Bioorganic & Medicinal Chemistry Letters, 1999

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Bioorganic & Medicinal Chemistry Letters, 2001

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László Patthy

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Protease Inhibitors: Synthesis of Bacterial Collagenase and Matrix Metalloproteinase Inhibitors Incorporating Succinyl Hydroxamate and Iminodiacetic Acid Hydroxamate Moieties

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Sérgio Marques

Bioorganic & Medicinal Chemistry, 2006

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Application of epimerisation-free amide coupling conditions to the synthesis of matrix metalloprotease inhibitor intermediates

Jonathan Fray

Tetrahedron, 1998

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