Agonist and Inverse Agonist Efficacy at Human Recombinant Serotonin 5-HT1A Receptors as a Function of Receptor:G-protein Stoichiometry (original) (raw)

Decreased G-protein coupling of serotonin 5-HT1A receptors in the brain of 5-HT1B knockout mouse

Ase Ase

Neuropharmacology, 2002

View PDFchevron_right

Cloning of Another Human Serotonin Receptor (5HT1F): A Fifth 5HT_1 Receptor Subtype Coupled to the Inhibition of Adenylate Cyclase

Michael Olsen

Proceedings of The National Academy of Sciences, 1993

View PDFchevron_right

Inverse Agonists and Serotonergic Transmission: From Recombinant, Human Serotonin (5HT)1B Receptors to G-Protein Coupling and Function in Corticolimbic Structures in vivo

Adrian Newman-Tancredi

Neuropsychopharmacology, 1999

View PDFchevron_right

Functional expression of the human serotonin 5-HT1A receptor in Escherichia coli. Ligand binding properties and interaction with recombinant G protein α-subunits

Stefano Marullo

Journal of Biological Chemistry

View PDFchevron_right

Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: Definition of its binding profile using agonists, antagonists and inverse agonists

Adrian Newman-Tancredi

Naunyn-Schmiedeberg's Archives of Pharmacology, 1998

View PDFchevron_right

Chromatographic Analyses of the Serotonin 5-HT 1A Receptor Solubilized from the Rat Hippocampus

S. Mestikawy

Journal of Neurochemistry, 1989

View PDFchevron_right

Preassociation between the 5‐HT 7 serotonin receptor and G protein G s : molecular determinants and association with low potency activation of adenylyl cyclase

Ornella Manfra

The FASEB Journal, 2018

View PDFchevron_right

Development and Characterization of Monoclonal Antibodies Specific to the Serotonin 5-HT2AReceptor

Jean Shih

Journal of Histochemistry and Cytochemistry, 1998

View PDFchevron_right

Pharmacological characterisation of the 5-HT1A serotonin receptor using the agonist [3H]8-OH-DPAT, and the antagonist [3H]spiperone

H. Sundaram, Adrian Newman-Tancredi

Biochemical Society transactions, 1992

View PDFchevron_right

Molecular biology of serotonin (5-HT) receptors

Jean Shih

Pharmacology Biochemistry and Behavior, 1991

View PDFchevron_right

In vitro autoradiography of serotonin 5‐HT2A2C receptor‐activated G protein: Guanosine‐5′‐(γ‐[35S]thio)triphosphate binding in rat brain

Hadassah Tamir

Journal of Neuroscience Research, 2000

View PDFchevron_right

Isolation of the serotoninergic 5-HT 4(e) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell lines

Jeanne Mialet-perez

British Journal of Pharmacology, 2000

View PDFchevron_right

Inverse agonism and constitutive activity as functional correlates of serotonin h5-HT(1B) receptor/G-protein stoichiometry

Adrian Newman-Tancredi

Molecular pharmacology, 2000

View PDFchevron_right

Serotonin autoreceptor in rat hippocampus: Pharmacological characterization as a subtype of the 5-HT1 receptor

Guido Maura

Naunyn-Schmiedeberg's Archives of Pharmacology, 1986

View PDFchevron_right

Serotonin receptors: from protein to physiological function and behavior

Prof. Youssef Sari

Neuroscience & Biobehavioral Reviews, 2004

View PDFchevron_right

Constitutive activity at serotonin 5-HT1D receptors: detection by homologous GTPγS versus [35S]-GTPγS binding isotherms

Adrian Newman-Tancredi

Neuropharmacology, 2001

View PDFchevron_right

Effect of the selective lesion of serotoninergic neurons on the regional distribution of 5-HT1A receptor mRNA in the rat brain

Magdy Riad

Molecular Brain Research, 1992

View PDFchevron_right

Differential Coupling of Serotonin 5-HT1A and 5-HT1B Receptors to Activation of ERK2 and Inhibition of Adenylyl Cyclase in Transfected CHO Cells

Jorge Antonio Mendez

Journal of Neurochemistry, 2002

View PDFchevron_right

Preassociation between the 5‐HT 7 serotonin receptor and G protein G s : molecular determinants and association with low potency activation of adenylyl cyclase

Ornella Manfra

The FASEB Journal, 2018

View PDFchevron_right

Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase

Theresa Branchek

Journal of Biological Chemistry, 1993

View PDFchevron_right

Inhibition of Serotonin 5-Hydroxytryptamine2C Receptor Function through Heterodimerization: RECEPTOR DIMERS BIND TWO MOLECULES OF LIGAND AND ONE G-PROTEIN

Joseph Mazurkiewicz

Journal of Biological Chemistry, 2005

View PDFchevron_right

Electrophysiology of 5-HT1A receptors in the rat hippocampus and cortex

Rodrigo Andrade

Drug Development Research, 1992

View PDFchevron_right

Investigation of a Novel Serotonin Receptor System in the Mammalian Brain

James Giordano

1989

View PDFchevron_right

Binding profile of the novel 5-HT1B/1D receptor antagonist, [3H]GR125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

Adrian Newman-Tancredi

European Journal of Pharmacology, 1997

View PDFchevron_right

Serotonergic modulation of neurotransmission in the rat subicular cortex in vitro: a role for 5-HT 1B receptors

Hwgm Boddeke

Naunyn-Schmiedeberg's archives of …, 1993

View PDFchevron_right