Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives (original) (raw)

Specific inhibition of binding to benzodiazepine receptors by 1, 2, 3-triazole derivatives

Journal of Pharmaceutical Sciences, 1992

Specific inhibition of benzodiazepine receptor binding by some N-(indol-3-ylglyoxylyl)amino acid derivatives

Journal of Medicinal Chemistry, 1985

Synthesis, benzodiazepine receptor affinity and in vivo testing of 3-aryl-4,7-dihydro-6-( N 1′-alkylpyrazol-3′ - or 5′-yl)pyrazolo[1,5- a]pyrimidin-7-ones

Lucia Casilli

European Journal of Medicinal Chemistry, 1998

View PDFchevron_right

Affinity of various compounds for benzodiazepine binding sites in rat brain, heart and kidneys in vitro

Veijo Saano

Acta pharmacologica et toxicologica, 1986

View PDFchevron_right

The separation of 3H-Benzodiazepine binding sites in brain and of benzodiazepine pharmacological properties

Arnold Lippa

Pharmacology, Biochemistry and Behavior, 1983

View PDFchevron_right

Modulation of benzodiazepine receptor binding: Insight into pharmacological efficacy

William Roeske

European Journal of Pharmacology, 1982

View PDFchevron_right

Recent Structure Activity Relationship Studies of 1,4-Benzodiazepines

Peertechz Journals

View PDFchevron_right

Synthesis, receptor affinity and effect on pentylenetetrazole-induced seizure threshold of novel benzodiazepine analogues: 3-Substituted 5-(2-phenoxybenzyl)-4H-1,2,4-triazoles and 2-amino-5-(phenoxybenzyl)-1,3,4-oxadiazoles

fatemeh ahmadi

Bioorganic & Medicinal Chemistry, 2014

View PDFchevron_right

Interaction of 2,3-benzodiazepines with peripheral benzodiazepine receptors

László Gráf

Pharmacological research communications, 1987

View PDFchevron_right

New 3-, 8-disubstituted pyrazolo[5,1-c][1,2,4]benzotriazines useful for studying the interaction with the HBp-3 area (hydrogen bond point area) in the benzodiazepine site on the γ-aminobutyric acid type A (GABAA) receptor

Gabriella Guerrini

Bioorganic & Medicinal Chemistry, 2011

View PDFchevron_right

Benzodiazepine receptor ligands. III. Synthesis and biological evaluation of 2- and/or 3-substituted pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides

Gabriella Guerrini

Il Farmaco

View PDFchevron_right

Novel benzodiazepine receptor partial agonists: oxadiazolylimidazobenzodiazepines

Erik Wong

Journal of Medicinal Chemistry, 1989

View PDFchevron_right

Tricyclic heteroaromatic systems: Synthesis, [3H]flunitrazepam brain membrane binding inhibition, and structure-activity relationships of 2,3-dihydro-2-aryl-4-R-[1]benzopyrano[4,3-C]pyrazole-3-ones

Giovanna Palazzino, Vittoria Colotta

Journal of Pharmaceutical Sciences, 1989

View PDFchevron_right

Synthesis and biodistribution of an 123I labelled flunitrazepam derivative: a potential in vivo tracer for benzodiazepine receptors

Paolo Ferrario

International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1988

View PDFchevron_right

2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands

Gabriella Guerrini

Bioorganic & Medicinal Chemistry, 2001

View PDFchevron_right

Benzodiazepine Receptor Ligands. 4. Synthesis and Pharmacological Evaluation of 3-Heteroaryl-8-chloropyrazolo[5,1- c ][1,2,4]benzotriazine 5-Oxides

Gabriella Guerrini

Journal of Medicinal Chemistry, 1999

View PDFchevron_right

Binding of [3H]ethyl-β-carboline-3-carboxylate to brain benzodiazepine receptors

Kenner Rice

FEBS Letters, 1981

View PDFchevron_right

Imidazo[2,1-b]thiazoles, imidazo[2,1-b]imidazoles and Pyrrolo[1,2-c]imidazoles. synthesis, structure and evaluation of benzodiazepine receptor binding

Christa Mueller

Journal of Heterocyclic Chemistry, 2002

View PDFchevron_right

Benzodiazepine receptor binding with [3H]-Ro 15-1788

Nicholas Goeders

Life Sciences, 1985

View PDFchevron_right

Molecular basis for the different binding properties of benzodiazepines to human and bovine peripheral-type benzodiazepine receptors

Daniel Caput

FEBS Letters, 1993

View PDFchevron_right

Pharmacological evaluation of an [123I] labelled imidazopyridine-3-acetamide for the study of benzodiazepine receptors

Karine Mardon, Filomena Mattner

Life Sciences, 2006

View PDFchevron_right

New Insight into the Central Benzodiazepine Receptor–Ligand Interactions: Design, Synthesis, Biological Evaluation, and Molecular Modeling of 3-Substituted 6-Phenyl-4 H -imidazo[1,5- a ][1,4]benzodiazepines and Related Compounds

Stefano Alcaro

Journal of Medicinal Chemistry, 2011

View PDFchevron_right

Benzodiazepine Binding Site Occupancy by the Novel GABA_A Receptor Subtype-Selective Drug 7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine (TPA023) in Rats, Primates, and Humans

Bindi Sohal

Journal of Pharmacology and Experimental Therapeutics, 2009

View PDFchevron_right

Animal pharmacokinetics of selected imidazopyrimidine ligands for benzodiazepine receptors

Anne Doyle

Drug Development Research, 1991

View PDFchevron_right

Isolation of Putative Benzodiazepine Receptors from Rat Brain Membranes by Affinity Chromatography

Silvana Hrelia

Journal of Neurochemistry, 1982

View PDFchevron_right

Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives (original) (raw)

Related papers