Enantioselective syntheses of (R)-3-phenyl GABA, (R)-baclofen and 4-arylpyrrolidin-2-ones (original) (raw)
Routes to 4-substituted analogues of the glycine/NMDA antagonist HA-996. Enantioselective synthesis of (3R,4R) 3-amino-1-hydroxy-4-methyl-2-pyrrolidinone (L-687, 414)
Paul D Leeson
Tetrahedron, 1992
View PDFchevron_right
Unexpected Behavior of the Reaction between 1,2-Diaza-1,3-Butadienes and 3-Dimethylaminopropenoates: A Useful Entry to New Pyrrolines, Pyrroles, and Oxazolines
Paolino Filippone
The Journal of Organic Chemistry, 2005
View PDFchevron_right
Palladium-Catalyzed Cyclization of Unsaturated β-Amino Alcohols: A New Access to Enantiopure Bicyclic Oxazolidines
Emmanuel Vrancken
Organic Letters, 2009
View PDFchevron_right
SECOND INTERNATIONAL SYMPOSIUM ON ORGANIC CHEMISTRY Sofia, Bulgaria 13 - 16 December 2008
Ali Gharib
View PDFchevron_right
Studies toward the Synthesis of 4-(2-R-ethyl)amino-2,2,5,5-tetramethyl-3-imidazoline 1-Oxyls. Nucleophilic Substitution of Bromide in the N -Alkyl Chain of the 1,2,4-Oxadiazol-2-one Precursor
Maxim Voinov
The Journal of Organic Chemistry, 2008
View PDFchevron_right
Effect of Regioisomerism on the Efficiency of 1-Phenylpyrrole-Type Atropisomeric Amino Alcohol Ligands in Enantioselective Organometallic Reactions
Ferenc Faigl
Synlett, 2018
View PDFchevron_right
Rhodium(III)-Catalyzed C–H Activation of Phenylazoles toward C–N Bond Cleavage of Diazabicyclic Olefins: A Facile Access to Mono- and Biscyclopentenyl-Functionalized Aza-Heteroaromatics
KV Radhakrishnan
Synlett, 2013
View PDFchevron_right
One-Step Preparation, Structural Assignment, and Xray Study of 2,2-Di-n-butyl- and 2,2-Diphenyl-6-aza-1,3-dioxa-2-stannabenzocyclononen-4-ones Derived from Amino Acids
Teresa Percino
Chemistry - A European Journal, 2003
View PDFchevron_right
Alkylation of Phenylglycinol-Derived Oxazolopiperidone Lactams. Enantioselective Synthesis of β-Substituted Piperidines
Rosa Griera
Journal of Organic Chemistry, 2006
View PDFchevron_right
4-Aryl-4-oxo-N-phenyl-2-aminylbutyramides as acetyl- and butyrylcholinesterase inhibitors. Preparation, anticholinesterase activity, docking study, and 3D structure–activity relationship based on molecular interaction fields
Ivan Juranic
Bioorganic & Medicinal Chemistry, 2010
View PDFchevron_right
Diastereoselective Intramolecular α-Amidoalkylation Reactions of l -DOPA Derivatives. Asymmetric Synthesis of Pyrrolo[2,1- a ]isoquinolines
Sonia Arrasate
The Journal of Organic Chemistry, 2005
View PDFchevron_right
Solution1H and13C NMR of new chiral 1,4-oxazepinium heterocycles and their intermediates from the reaction of 2,4-pentanedione with ?-L-amino acids and (R)-(?)-2-phenylglycinol
Carlos Lobato
Magnetic Resonance in Chemistry, 2003
View PDFchevron_right
Photoinduced cyclizations of mono- and dianions of N-acyl-o-chloroanilines and N-acyl-o-chlorobenzylamines as general methods for the synthesis of oxindoles and 1,4-dihydro-3(2H)-isoquinolinones
Jyothi Pisipati
Journal of the American Chemical Society, 1985
View PDFchevron_right
Functionalization of aromatic and heterocyclic systems. Regioselective introduction of 2-oxoalkyl chain or cyano functions via organoiron complexes
Ratan Chowdhury
Journal of Organic Chemistry, 1987
View PDFchevron_right
Synthesis and Chemical Reaction of 2-Oxazoline 5-Ones Derivatives
Wafaa Khl
International Journal of Chemical and Biomolecular Science, 2019
View PDFchevron_right
An expedient and facile route for the general synthesis of 3-aryl substituted 1,2,3-triazolo[1,5-a][1,4]benzodiazepin-6-ones and 1,2,3-triazolo[1,5-a][1,5]benzodiazocin-7-ones
Basudeb Achari
Organic & Biomolecular Chemistry, 2010
View PDFchevron_right
2H-1,2-Azaphosphindoles – Synthesis and Characterization
Victorio Cadierno
European Journal of Inorganic Chemistry, 2000
View PDFchevron_right
Synthesis and molecular modeling of (4′R)- and (4′S)- 4′-substituted 2′-{[(E)-androst-5-en-17-ylidene]-methyl}oxazolines
Alexander Veselovsky
Steroids, 2013
View PDFchevron_right
An asymmetric organocatalytic approach towards allylic amines and β-keto amino compounds
Lars Ransborg
Chemical Communications, 2009
View PDFchevron_right
Electrochemical generation of chiral oxazolidin-2-ones anions: a new procedure for the highly diastereoselective conjugate addition to nitroalkenes
M. Feroci
Tetrahedron: Asymmetry, 2001
View PDFchevron_right
A new chiral glycine synthon. Synthesis, x-ray structure of (−).(2S,4R)-2-ethoxycarbonyl-4-phenyl-1,3-oxazolidine and diastereoselective nucleophilic ring opening to (R)-ethyl α-amino carboxylates
Santiago García-Granda
Tetrahedron Letters, 1992
View PDFchevron_right
A Fast and Facile Synthesis of Geometric Isomers of 4-Cinnamylidene-2-Phenyl-2- Oxazolin-5-One and their Stereospecific Solvolysis Products
Priyanka Borah
IARJSET, 2021
View PDFchevron_right
Metal free stereoselective synthesis of functionalized enamides
Bilal Bhat
Org. Biomol. Chem., 2014
View PDFchevron_right
Synthesis of Tetra-, Hexa-, and Octanuclear Organozinc Ring Systems
Mark Elsegood
Angewandte Chemie International Edition, 2007
View PDFchevron_right
Oxa-ene Reaction of Enols of Amides with 4-Phenyl-1,2,4-triazoline-3,5-dione †
Ahmad Basheer
The Journal of Organic Chemistry, 2008
View PDFchevron_right
Enantiopure 4‐oxazolin‐2‐ones and 4‐methylene‐2‐oxazolidinones as chiral building blocks in a divergent asymmetric synthesis of heterocycles
Joaquín Tamariz
Chirality, 2019
View PDFchevron_right
A highly active organocatalyst for the asymmetric α-aminoxylation of aldehydes and α-hydroxylation of ketones
Miquel A. Pericàs
RSC Advances, 2012
View PDFchevron_right
Synthesis, configuration and properties of some new 3, 4, 5-substituted oxazolidin-2-ones
Anelia Mavrova
European Journal of …, 2011
View PDFchevron_right
Syntheses of 21-hydroxy-11,19-oxidopregn-4-ene-3,20-dione and 21-hydroxy- 6,19-oxidopregn-4-ene-3,20-dione
Gerardo Burton
Steroids, 1995
View PDFchevron_right
Design, synthesis, and evaluation of cyclic amide/imide-bearing hydroxamic acid derivatives as class-selective histone deacetylase (HDAC) inhibitors
Hiroyuki Miyachi
Bioorganic & Medicinal Chemistry, 2006
View PDFchevron_right
Diastereospecific synthesis of (S,S)-2-substituted-4,4-diphenyl-3, 1-oxazabicyclo[3.3.0]octanes
Jiaxi Xu
Heteroatom Chemistry, 2003
View PDFchevron_right
11.Use of 0002www.iiste.org Call_for_Paper-Ethoxy(4H)-3,1-benzoxazin-4-one as a Precursor
Alexander Decker
View PDFchevron_right
Sequential CÀN and CÀO Bond Formation in a Single Pot: Synthesis of 2H-Benzo[b][1,4]oxazines from 2,5-Dihydroxybenzaldehyde and Amino acid Precursors
Balakrishna Dulla
View PDFchevron_right
Dimethoxyethane as an Alternative Solvent for Schmidt Reactions. Preparation of Homochiral N-(5-Oxazolyl)oxazolidinones from N-Acetoacetyl Derivatives of Oxazolidinones
Tadaaki NAGAO
Tetrahedron, 1996
View PDFchevron_right
Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine
Michela Festa
European Journal of Medicinal Chemistry, 2007
View PDFchevron_right