Regulation of Androgen Receptor Activity by Transient Interactions of Its Transactivation Domain with General Transcription Regulators (original) (raw)

Increased androgen receptor transcription: a cause of castration-resistant prostate cancer and a possible therapeutic target

Masaki Shiota

Journal of Molecular …, 2011

View PDFchevron_right

The Androgen Receptor Induces a Distinct Transcriptional Program in Castration-Resistant Prostate Cancer in Man

Stewart MacArthur

Cancer Cell, 2013

View PDFchevron_right

Small molecule screening reveals a transcription-independent pro-survival function of androgen receptor in castration-resistant prostate cancer

Inna Shyshynova

Cell Cycle, 2009

View PDFchevron_right

Androgen receptors in early and castration resistant prostate cancer: friend or foe?

Efstathios Stathopoulos

HORMONES, 2013

View PDFchevron_right

Regression of Castrate-Recurrent Prostate Cancer by a Small-Molecule Inhibitor of the Amino-Terminus Domain of the Androgen Receptor

Simon Haile, Iain McEwan

Cancer Cell, 2010

View PDFchevron_right

Ligand-independent Androgen Receptor Activity Is Activation Function-2-independent and Resistant to Antiandrogens in Androgen Refractory Prostate Cancer Cells

Yingming Li

Journal of Biological Chemistry, 2006

View PDFchevron_right

Androgen Receptor Cofactors in Prostate Cancer: Potential Therapeutic Targets of Castration-Resistant Prostate Cancer

Akira Yokomizo

Current Cancer Drug Targets, 2011

View PDFchevron_right

Development of an Androgen Receptor Inhibitor Targeting the N-Terminal Domain of Androgen Receptor for Treatment of Castration Resistant Prostate Cancer

Hisham Mohammed

Cancers, 2021

View PDFchevron_right

Recent Discoveries in the Androgen Receptor Pathway in Castration-Resistant Prostate Cancer

Asish Pati

Frontiers in Oncology, 2020

View PDFchevron_right

Androgen Receptor Signaling Pathway in Prostate Cancer: From Genetics to Clinical Applications

Alessia Cimadamore

Cells

View PDFchevron_right

Mechanisms of androgen receptor repression in prostate cancer

Vikash Reebye

Biochemical Society Transactions, 2006

View PDFchevron_right

Suppression of Androgen Receptor Signaling in Prostate Cancer Cells by an Inhibitory Receptor Variant

Carmela Ricciardelli

Molecular Endocrinology, 2006

View PDFchevron_right

Inhibiting androgen receptor nuclear entry in castration-resistant prostate cancer

scott lawrence

Nature Chemical Biology, 2016

View PDFchevron_right

Posttranslational Modification of the Androgen Receptor in Prostate Cancer

Donald Tindall

International Journal of Molecular Sciences, 2013

View PDFchevron_right

A detailed characterization of stepwise activation of the androgen receptor variant 7 in prostate cancer cells

Marcelo Roggero

Oncogene, 2020

View PDFchevron_right

A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance

Eva Estébanez-Perpiñá

Science Advances

View PDFchevron_right

Androgen receptor regulates a distinct transcription program in androgen-independent prostate cancer

Mathieu Lupien

Cell, 2009

View PDFchevron_right

Eighty Years of Targeting Androgen Receptor Activity in Prostate Cancer: The Fight Goes on

Eva Estébanez-Perpiñá

Cancers

View PDFchevron_right

Global analysis of transcription in castration-resistant prostate cancer cells uncovers active enhancers and direct androgen receptor targets

Einari Niskanen

Scientific Reports, 2016

View PDFchevron_right

Engineered repressors are potent inhibitors of androgen receptor activity

Simak Ali

Oncotarget, 2014

View PDFchevron_right

Agonist and antagonist switch DNA motifs recognized by human androgen receptor in prostate cancer

Pearlly Yan

The EMBO journal, 2014

View PDFchevron_right

The Androgen Receptor in Prostate Cancer: Effect of Structure, Ligands and Spliced Variants on Therapy

Maria Mudryj

Biomedicines

View PDFchevron_right

Targeting androgen receptor activation function-1 with EPI to overcome resistance mechanisms in castration-resistant prostate cancer

Iain McEwan

Clinical cancer research : an official journal of the American Association for Cancer Research, 2016

View PDFchevron_right

Clinical relevance of androgen receptor alterations in prostate cancer

Pernilla Wikström

Endocrine Connections, 2017

View PDFchevron_right

Increased Expression of Androgen Receptor Sensitizes Prostate Cancer Cells to Low Levels of Androgens

Olli Jänne

Cancer Research, 2009

View PDFchevron_right

Modulation of Androgen Receptor Signaling in Hormonal Therapy-Resistant Prostate Cancer Cell Lines

Wilfred van IJcken

PLoS ONE, 2011

View PDFchevron_right