NNC-711: An Inhibitor of GAB A Uptake with Selective Affinity to GAT-1 (original) (raw)

NNC-711 is detailed as a selective inhibitor of GABA uptake, specifically targeting the GAT-1 transporter, which is crucial in regulating GABAergic neurotransmission in the mammalian brain. The study explores the pharmacological effects of NNC-711 in various neurological models, showcasing its potential in modulating GABA levels and influencing neurological disorders. Furthermore, the research provides a comprehensive receptor-binding profile, highlighting the selectivity of NNC-711 across multiple neurotransmitter systems.