Synthesis of enantiopure trisubstituted piperidines from a chiral epoxyaziridine and α-amino esters (original) (raw)

A Simple Stereoselective Synthesis of Enantiopure 2-Substituted Pyrrolidines and Piperidines from Chiral (R)-Phenylglycinol-Derived Bicyclic 1,3-Oxazolidines

Rafael Pedrosa

European Journal of Organic Chemistry, 2000

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Totally Selective Synthesis of Enantiopure (3 S ,5 S )- and (3 R ,5 R )-4-Amino-3,5-dihydroxypiperidines from Aminodiepoxides Derived from Serine

Santiago García-Granda

The Journal of Organic Chemistry, 2008

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Chiral Oxazolopiperidone Lactams: Versatile Intermediates for the Enantioselective Synthesis of Piperidine‐Containing Natural Products

carmen escolano

Chemistry – A European Journal, 2006

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Alkylation of Phenylglycinol-Derived Oxazolopiperidone Lactams. Enantioselective Synthesis of β-Substituted Piperidines

Oscar Lozano

Journal of Organic Chemistry, 2006

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Chiral precursors for the synthesis of enantiomerically pure piperidines. Total synthesis of (R)-(-)-coniine

Núria Llor

Tetrahedron Letters, 1994

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Synthesis of Enantiopure trans -3,4-Disubstituted Piperidines. An Enantiodivergent Synthesis of (+)- and (−)-Paroxetine

Elies Molins

The Journal of Organic Chemistry, 2000

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Synthetic approaches to a chiral 4-amino-3-hydroxy piperidine with pharmaceutical relevance

Adrian Ortiz

Organic & Biomolecular Chemistry, 2012

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Synthesis of enantiopure pyrrolidine and piperidine derivatives via ring closing metathesis

Alfred Hassner

Tetrahedron Letters, 2000

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Highly enantioselective organocatalytic synthesis of piperidines. Formal synthesis of (-)-Paroxetine

Ramon Rios

Tetrahedron Letters, 2009

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An Enantioselective Synthetic Route to cis -2,4-Disubstituted and 2,4-Bridged Piperidines

maria perez

The Journal of Organic Chemistry, 2008

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Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines

Jiří Schimer, Marek Humpl

2011

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Synthesis of 3-aminopyrrolidines and piperidines from endocyclic enamine derivatives

Robert Batey

2001

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Conjugate Addition of Organocuprates to Chiral Bicyclic δ-Lactams. Enantioselective Synthesis of cis -3,4-Disubstituted and 3,4,5-Trisubstituted Piperidines

Elies Molins

Organic Letters, 2001

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An efficient synthesis of (R)- and (S)-2-(aminomethyl)piperidine dihydrochloride

thomas moraux

Tetrahedron: Asymmetry, 2008

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Enantioselective Synthesis of 3,3-Disubstituted Piperidine Derivatives by Enolate Dialkylation of Phenylglycinol-Derived Oxazolopiperidone Lactams

Oscar Lozano

Journal of Organic Chemistry, 2007

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One-pot multiple reactions: asymmetric synthesis of 2,6-cis-disubstituted piperidine alkaloids from chiral aziridine

Giuliano Kullik

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Carbohydrate-auxiliary assisted preparation of enantiopure 1,2-oxazine derivatives and aminopolyols

Dieter Lentz

Beilstein Journal of Organic Chemistry, 2012

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Dynamic Kinetic Resolution and Desymmetrization Processes: A Straightforward Methodology for the Enantioselective Synthesis of Piperidines

Elies Molins

Chemistry: A European Journal, 2006

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Efficient Enantioselective Synthesis of Piperidines through Catalytic Asymmetric Ring-Opening/Cross-Metathesis Reactions

Richard Schrock

Angewandte Chemie International Edition, 2007

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A short enantioselective access to 2,3,6-trialkylpiperidines and 5,8-dialkylindolizidines

Yung-sing Wong

Tetrahedron, 1998

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From Amino Acids to Fused Chiral Pyrrolidines and Piperidines via the INOC Route

Hugo Gottlieb

European Journal of Organic Chemistry, 2000

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A practical asymmetric synthesis of 2,6- cis-disubstituted piperidines

Stephane Ciblat

Tetrahedron-asymmetry, 1999

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Chiral ligands containing heteroatoms. 11. Optically active 2-hydroxymethyl piperazincs as catalysts in the enantioselective addition of diethylzinc to benzaldehyde

Sandra Conti

Tetrahedron: Asymmetry, 1993

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