Synthesis of Stable and Potent δ/μ Opioid Peptides: Analogues of H-Tyr- c [ d -Cys-Gly-Phe- d -Cys]-OH by Ring-Closing Metathesis
Luisa Mannina
Journal of Medicinal Chemistry, 2007
View PDFchevron_right
Structure–activity relationships of bifunctional cyclic disulfide peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors
Victor Hruby is to
Peptides, 2008
View PDFchevron_right
Conformation-activity relationships of cyclo -constrained µ/δ opioid agonists derived from the N -terminal tetrapeptide segment of dermorphin/deltorphin
Cezary Czaplewski
Journal of Peptide Science, 2008
View PDFchevron_right
Cyclic Opioid Peptide Agonists and Antagonists Obtained Via Ring-Closing Metathesis
Peter Schiller
Chemical Biology & Drug Design, 2009
View PDFchevron_right
Opioid receptor affinity and selectivity effects of second residue and carboxy terminal residue variation in a cyclic disulfide-containing opioid tetrapeptide
Henry I. Mosberg
International Journal of Peptide and Protein Research, 2009
View PDFchevron_right
Synthesis and activity profiles of novel cyclic opioid peptide monomers and dimers
Peter Schiller
Journal of Medicinal Chemistry, 1985
View PDFchevron_right
Peptides opioides: synthèse et propriétés biologiques d'hexapeptides apparents à la dermorphine
Gianfranco Balboni
European Journal of Medicinal Chemistry, 1990
View PDFchevron_right
Cyclization in Opioid Peptides
Anna Janecka
Current Drug Targets, 2013
View PDFchevron_right
In Vivo Cleavability of a Disulfide-Based Chimeric Opioid Peptide in Rat Brain
Ulrich Bickel
Bioconjugate Chemistry, 1995
View PDFchevron_right
Opioid peptides. Synthesis and biological properties of dermorphin related hexapeptides
Roberto Tomatis
View PDFchevron_right
Translation of structure-activity relationships from cyclic mixed efficacy opioid peptides to linear analogues
Jessica Anand
Biopolymers, 2014
View PDFchevron_right
Cyclic, disulfide- and dithioether-containing opioid tetrapeptides: Development of a ligard with high delta opioid receptor selectivity and affinity
Henry I. Mosberg
Life Sciences, 1988
View PDFchevron_right
New paradigm for drug design: Design and synthesis of novel biologically active peptides that are agonists at opioid receptors and antagonists at cholecystokinin receptors
Richard Agnes
2003
View PDFchevron_right
Conformational analysis of enkephalin analogs contaIntng a disulfide bond Models for delta- and mu-receptor opioid agonists
Victor Hruby
International Journal of Peptide and Protein Research, 2009
View PDFchevron_right
Bifunctional μ/δ Opioid Peptides: Variation of the Type and Length of the Linker Connecting the Two Components
Peter Schiller
Chemical Biology & Drug Design, 2012
View PDFchevron_right
Design, Synthesis and Functional Analysis of Cyclic Opioid Peptides with Dmt-Tic Pharmacophore
Arijit Sarkar
Molecules, 2020
View PDFchevron_right
Development of Centrally Acting Peptide Analogs: Structure-Transport Studies and Pharmacological Evaluation of Analogs of the Opioid Peptide Dynorphin A
Amanda Carey
View PDFchevron_right
Opioid peptides: synthesis and biological properties of [(N?-glucosyl,N?-methoxy)-?,?-diamino-(S)-butanoyl]4-deltorphin-1-neoglycopeptide and related analoguesWith the exception of d-Ala the amino acid residues are of l-configuration. Standard abbreviations for amino acid derivatives and peptides...
elisa giannini
Organic & Biomolecular Chemistry, 2003
View PDFchevron_right
Recent developments in the design of receptor specific opioid peptides
Victor Hruby is to
Medicinal Research Reviews, 1989
View PDFchevron_right
δ Opioidmimetic Antagonists: Prototypes for Designing a New Generation of Ultraselective Opioid Peptides
Delia Picone
Molecular Medicine, 1995
View PDFchevron_right
Design and Comprehensive Conformational Studies of Tyr 1 -cyclo( d Pen 2 Gly 3 -Phe 4 - l -3-Mpt 5 ) and Tyr 1 -cyclo( d Pen 2 Gly 3 -Phe 4 - d -3-Mpt 5 ): Novel Conformationally Constrained Opioid Peptides
Steve Kolodziej, Garland Marshall
Cheminform, 2010
View PDFchevron_right
Recent Progress Towards Pharmaceutical Applications of Disulfide-Rich Cyclic Peptides
Christina Schroeder, Joakim Swedberg
Current Protein & Peptide Science, 2013
View PDFchevron_right
Combined use of NMR, distance geometry and MD calculations for the conformational analysis of opioid peptides of the type [D(L)Cys2, D(L)Cys5]enkephalin
Fritz Andreae
International Journal of Peptide and Protein Research, 2009
View PDFchevron_right
δ-Selective Opioid Peptides Containing a Single Aromatic Residue in the Message Domain: An NMR Conformational Analysis
Delia Picone
Journal of Peptide Science, 1996
View PDFchevron_right
Conformational analysis of enkephalin analogs containing a disulfide bond. Models for delta- and mu-receptor opioid agonists
Victor Hruby is to
International journal of peptide and protein research, 1989
View PDFchevron_right
Opioid peptides: synthesis and biological properties of [(Nγ-glucosyl,Nγ-methoxy)-α,γ-diamino-(S)-butanoyl]4-deltorphin-1-neoglycopeptide and related analogues
elisa giannini
Organic Biomolecular Chemistry, 2003
View PDFchevron_right
Novel Opioid Peptide Derived Antagonists Containing (2 S )-2-Methyl-3-(2,6-dimethyl-4-carbamoylphenyl)propanoic Acid [(2 S )-Mdcp]
Peter Schiller
Journal of Medicinal Chemistry, 2008
View PDFchevron_right