2-Amino-4-pyrrolidinothieno[2,3- d ]pyrimidine-6-carboxylic Acid as an N -Terminal Surrogate in Amino Acid and Peptide Analogues (original) (raw)

Recent Advances in the Synthesis of Some Bioactive Peptides and Peptidomimetics

Javed Iqbal

Current Pharmaceutical Biotechnology, 2006

View PDFchevron_right

Design, Synthesis and Pharmacological properties of peptidomimetics

Ahmad Junaid

View PDFchevron_right

High Throughput Synthesis of Peptides and Peptidomimetics

Victor Hruby is to

ChemInform, 2007

View PDFchevron_right

Therapeutic importance of peptidomimetics in medicinal chemistry

Prabodh Sharma

View PDFchevron_right

Synthesis and conformational analysis of peptidomimetics containing unnatural amino acids based on a piperazinone and g-butyrolactone scaffolds

D. Scherman

2009

View PDFchevron_right

Peptidomimetics, a synthetic tool of drug discovery

Victor Hruby is to

Current Opinion in Chemical Biology, 2008

View PDFchevron_right

Synthesis of Conformational Restricted Amino Acids and Their Use in the Preparation of Biologically Active Peptides and Peptidomimetics

Cristian Cattaneo

2015

View PDFchevron_right

Synthesis and Conformational Studies of Peptidomimetics Containing Furanoid Sugar Amino Acids and a Sugar Diacid

Marco Crisma

The Journal of Organic Chemistry, 2000

View PDFchevron_right

Synthesis of heterocyclic β-amino acids. A convenient preparation of β-amino-5-pyrimidinepropanoic acid and derivatives

Joseph Rico

Tetrahedron Letters, 1993

View PDFchevron_right

Development of 5-(aminomethyl)pyrrole-2-carboxylic acid as a constrained surrogate of Gly-ΔAla and its application in peptidomimetic studies

Kiran Singarapu

Tetrahedron Letters, 2002

View PDFchevron_right

Non-Canonical Amino Acids as Building Blocks for Peptidomimetics: Structure, Function, and Applications

Tarsila Castro

Biomolecules

View PDFchevron_right

Solid-Phase Synthesis of Multiple Classes of Peptidomimetics from Versatile Resin-Bound Aldehyde Intermediates

John Huffman

Journal of the American Chemical Society, 2007

View PDFchevron_right

Solid-Phase Synthesis of “Mixed” Peptidomimetics Using Fmoc-Protected Aza-β 3 -amino Acids and α-Amino Acids

Lanrong Bi

The Journal of Organic Chemistry, 2005

View PDFchevron_right

An efficient approach for solid-phase synthesis of peptidomimetics based on 4-imidazolidinones

Richard Siahaan

Tetrahedron letters, 2002

View PDFchevron_right

Conformationally Constrained Histidines in the Design of Peptidomimetics: Strategies for the χ-Space Control

Ivana Cacciatore

International Journal of Molecular Sciences, 2011

View PDFchevron_right

Proficient synthesis of bioactive annulated pyrimidine derivatives: A review

ajmal bhat

Journal of Taibah University for Science

View PDFchevron_right

A proposed bioactive form of peptide T and the design of peptidomimetics

Margarita Calafell

Letters in Peptide Science, 1998

View PDFchevron_right

Chemo- and Regioselective Syntheses of Enantiopure Aminopyrrolidinones as Building Blocks for Constrained Peptidomimetics

Peter Gmeiner

HETEROCYCLES, 1999

View PDFchevron_right

Application of the Ugi reaction with multiple amino acid-derived components: synthesis and conformational evaluation of piperazine-based minimalist peptidomimetics

Michael Christodoulou

Organic & biomolecular chemistry, 2015

View PDFchevron_right

Peptide, peptidomimetic, and organic synthetic combinatorial libraries

Jutta Eichler

Medicinal Research Reviews, 1995

View PDFchevron_right

Synthesis of Novel Pyrimidine Derivative and Its Biological Evaluation

Anshu Chaudhary

2011

View PDFchevron_right

Synthesis of ‘difficult’ peptides free of aspartimide and related products, using peptoid methodology

Corrado Guarnaccia, Sándor Pongor

Tetrahedron Letters, 2006

View PDFchevron_right

Synthesis of a Chloroalkene Dipeptide Isostere-Containing Peptidomimetic and Its Biological Application

Kentaro Hozumi

ACS Medicinal Chemistry Letters, 2018

View PDFchevron_right

4-Alkoxy-2-hydroxybenzaldehyde (AHB): A Versatile Aldehyde Linker for Solid-Phase Synthesis of C-Terminal Modified Peptides and Peptidomimetics †

Victor Hruby

Organic Letters, 2000

View PDFchevron_right

Advances in Development of Antimicrobial Peptidomimetics as Potential Drugs

Henrik Franzyk

Molecules

View PDFchevron_right

Peptidomimetic Synthesis by Way of Diastereoselective Iodoacetoxylation and Transannular Amidation of 7–9-Membered Lactams

N D Prasad Atmuri

Organic Letters, 2017

View PDFchevron_right