Characterization in Rats of the Anxiolytic Potential of ELB139 [1-(4-Chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-on], a New Agonist at the Benzodiazepine Binding Site of the GABAA Receptor
Shahram Akbarzadeh
Journal of Pharmacology and Experimental Therapeutics, 2005
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Benzodiazepine Binding Site Occupancy by the Novel GABAA Receptor Subtype-Selective Drug 7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine (TPA023) in Rats, Primates, and Humans
Bindi Sohal
Journal of Pharmacology and Experimental Therapeutics, 2009
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Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series
Frederic Knoflach
Bioorganic & Medicinal Chemistry Letters, 2009
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Sh-I-048A, an in vitro non-selective super-agonist at the benzodiazepine site of GABAA receptors: The approximated activation of receptor subtypes may explain behavioral effects
Bojan Markovic
Brain Research, 2014
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Are GABAA Receptors Containing α5 Subunits Contributing to the Sedative Properties of Benzodiazepine Site Agonists?
Dubravko Bokonjic
Neuropsychopharmacology, 2008
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Benzodiazepine Binding Site Occupancy by the Novel GABAA Receptor Subtype-Selective Drug 7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine (TPA023) in Rats, Primates, and Humans
sandra sanabria
Journal of Pharmacology and Experimental Therapeutics, 2010
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Interaction of SQ 20009 and GABA-like drugs as modulators of benzodiazepine receptor binding
Porntip Supavilai
European Journal of Pharmacology, 1980
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Beyond classical benzodiazepines: novel therapeutic potential of GABAA receptor subtypes
Uwe Rudolph
Nature Reviews Drug Discovery, 2011
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A Review of the Updated Pharmacophore for the Alpha 5 GABA(A) Benzodiazepine Receptor Model
Michael Poe
International Journal of Medicinal Chemistry, 2015
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benzodiazepine receptor ligands a patent review (2006-2012).pdf
Gabriella Guerrini
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Benzodiazepine receptor ligands: a patent review (2006 – 2012)
Gabriella Guerrini
Expert Opinion on Therapeutic Patents, 2013
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Inhibition of γ-aminobutyric acid stimulated [3H]diazepam binding by benzodiazepine receptor ligands
Phil Skolnick
Biochemical Pharmacology, 1981
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Gaba Receptors and Benzodiazepines
Colin Goodchild
BJA: British Journal of Anaesthesia, 1993
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Modulation of benzodiazepine receptor binding: Insight into pharmacological efficacy
William Roeske
European Journal of Pharmacology, 1982
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Actions of two GABAA receptor benzodiazepine-site ligands that are mediated via non-γ2-dependent modulation
Holger Rabe, Hartmut Lüddens
European Journal of Pharmacology, 2011
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Chronic treatment with diazepam or the inverse benzodiazepine receptor agonist FG 7142 causes differential changes in the effects of GABA receptor stimulation
Dai Stephens
Epilepsy Research, 1988
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Chronic exposure of cells expressing recombinant GABAA receptors to benzodiazepine antagonist flumazenil enhances the maximum number of benzodiazepine …
Dubravka Švob Štrac
Life sciences, 2004
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Biological function of GABAA/benzodiazepine receptor heterogeneity
Hartmut Lüddens
Journal of Psychiatric Research, 1995
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Computer-aided design of selective ligands of the benzodiazepine-binding site of the GABAA receptor
Vladimir Chupakhin
Doklady Chemistry, 2008
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Triazolam is more efficacious than diazepam in a broad spectrum of recombinant GABAA receptors
Stefano Vicini
European Journal of Pharmacology: Molecular Pharmacology, 1993
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Chronic exposure of cells expressing recombinant GABAA receptors to benzodiazepine antagonist flumazenil enhances the maximum number of benzodiazepine binding sites
Dubravka Švob Štrac
Life Sciences, 2004
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6-Methyl-3′-bromoflavone, a High-Affinity Ligand for the Benzodiazepine Binding Site of the GABAA Receptor with Some Antagonistic Properties
Luciana Izquierdo
Biochemical and Biophysical Research Communications, 1999
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