hERG potassium channel inhibition by ivabradine requires channel gating (original) (raw)
Related papers
Biophysical Journal, 2021
Sulfonylureas blockade of neural and cardiac HERG channels
FEBS Letters, 1998
Physicochemical Features of the hERG Channel Drug Binding Site
Journal of Biological Chemistry, 2004
Potassium Channel Toxins and Transmitter Release
Annals of the New York Academy of Sciences, 1994
Lipid-dependent gating of a voltage-gated potassium channel
Nature Communications, 2011
G protein modulation of K2P potassium channel TASK-2
Pflügers Archiv - European Journal of Physiology, 2013
Modulating inhibitory ligand-gated ion channels
The AAPS Journal, 2006
The Link between Ion Permeation and Inactivation Gating of Kv4 Potassium Channels
Biophysical Journal, 2003
Glutamate receptor ion channels
Current Opinion in Neurobiology, 2005
Investigation of hERG1b influence on hERG channel pharmacology at physiological temperature
Journal of Pharmacology and Pharmacotherapeutics
14-3-3θ is a Binding Partner of Rat Eag1 Potassium Channels
PLoS ONE, 2012
Inhibition of HERG potassium channels by the antimalarial agent halofantrine
British Journal of Pharmacology, 2000
Modulation of Kir4.1 and Kir4.1-Kir5.1 channels by extracellular cations
Biochimica et Biophysica Acta (BBA) - Biomembranes, 2009
A Novel Inhibitor of Hypertonicity-Induced Cation Channels in HeLa Cells
The Journal of Physiological Sciences, 2007
Phasic GABAA-mediated inhibition
Epilepsia, 2010
Molecular Pharmacology, 2005
Migraine and Two-Pore-Domain Potassium Channels
The Neuroscientist, 2020
hERG Potassium Channel Blockade by the HCN Channel Inhibitor Bradycardic Agent Ivabradine
Journal of the American Heart Association, 2015
Potassium channels in T lymphocytes: toxins to therapeutic immunosuppressants
Toxicon, 2001
Ivabradine maintains sinus rhythm and reverses atrial tachycardia-induced cardiomyopathy
European Heart Journal Supplements, 2014
Thiazide-Induced Vasodilation in Humans Is Mediated by Potassium Channel Activation
Hypertension, 1998
Yeast Screen for Constitutively Active Mutant G Protein–Activated Potassium Channels
Neuron, 2001
Diabetologia, 2001
Crosstalk between NMDAR antagonists and potassium channels in murine and human lymphocytes
2018
Involvement of potassium channels in amitriptyline and clomipramine analgesia
Neuropharmacology, 2001
Ion Channel Involvement in Tumor Drug Resistance
Journal of Personalized Medicine, 2022
The Eag Domain Regulates the Voltage-Dependent Inactivation of Rat Eag1 K+ Channels
PLoS ONE, 2014
Potassium channel blockade restores the attenuated noradrenaline sensitivity in human endotoxemia
2005
Alam et al 2008 Braz J Pharmacog
Modulation of rat cardiac sodium channel by the stimulatory G protein alpha subunit
The Journal of Physiology, 1999
Novel Inhibitors of the Gardos Channel for the Treatment of Sickle Cell Disease
Journal of Medicinal Chemistry, 2008
TREK-1, a K+ channel involved in neuroprotection and general anesthesia
The EMBO Journal, 2004
Kv1.3 Potassium Channels: Promising Therapeutic Targets in Hematological Malignancies
Journal of Cellular Signaling, 2020
Assessing hERG Channel Inhibition Using PatchXpress
Journal of the Association for Laboratory Automation, 2005