Metabotropic glutamate receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database (original) (raw)

Metabotropic glutamate receptors in GtoPdb v.2021.3

Francesco Ferraguti

IUPHAR/BPS Guide to Pharmacology CITE, 2021

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Metabotropic glutamate receptors in GtoPdb v.2023.1

Francesco Ferraguti

IUPHAR/BPS guide to pharmacology CITE, 2023

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Comparative analysis of the ligand-binding sites of the metabotropic glutamate receptors mGluR1-mGluR8

Igor Baskin

Doklady. Biochemistry and biophysics

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The G Protein-Coupling Profile of Metabotropic Glutamate Receptors, as Determined with Exogenous G Proteins, Is Independent of Their Ligand Recognition Domain

Jean-philippe Pin

Molecular Pharmacology, 1998

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Dynamics and modulation of metabotropic glutamate receptors

Philippe Rondard

Current opinion in pharmacology, 2015

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Metabotropic glutamate receptors as drug targets: what's new?

R. Ngomba, Roberto Gradini

Current Opinion in Pharmacology, 2015

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Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein coupling

R. Rahmeh, Pauline Scholler

Proceedings of the National Academy of Sciences, 2012

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Molecular modeling and mutagenesis of the ligand-binding pocket of the mGlu3 subtype of metabotropic glutamate receptor

David Hampson

Journal of Neurochemistry, 2003

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Amino-Pyrrolidine Tricarboxylic Acids Give New Insight into Group III Metabotropic Glutamate Receptor Activation Mechanism

Nicolas Triballeau

Molecular Pharmacology, 2006

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Allosteric Binding Site and Activation Mechanism of Class C G-Protein Coupled Receptors: Metabotropic Glutamate Receptor Family

Guanxing Hu

The AAPS Journal, 2015

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Constitutive activity of metabotropic glutamate receptors: Role of the intracellular interacting proteins, Homer

Laurent Prézeau

European Neuropsychopharmacology, 2002

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Sensing conformational changes in metabotropic glutamate receptors

Marie-Laure RIVES

Proceedings of the National Academy of Sciences, 2013

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Membrane Topology of a Metabotropic Glutamate Receptor

Farzana Karim

Journal of Biological Chemistry, 2003

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Inverse agonists to explore the mechanisms of metabotropic glutamate receptor activity

Laurent Prézeau

International Congress Series, 2003

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Pharmacology and Functions of Metabotropic Glutamate Receptors

faisal soomro

Annual Review of Pharmacology and …, 1997

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A new binding mode of competitive antagonists to metabotropic glutamate receptors exemplified by the mGluR1-receptor antagonist AIDA (RS-aminoindan-1,5-dicarboxylic acid)

Igor Baskin

Doklady. Biochemistry and biophysics

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Transposition of Three Amino Acids Transforms the Human Metabotropic Glutamate Receptor (mGluR)-3-Positive Allosteric Modulation Site to mGluR2, and Additional Characterization of the mGluR2-Positive Allosteric Modulation Site

Hervé Schaffhauser

Journal of Pharmacology and Experimental Therapeutics, 2008

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Closure of the Venus flytrap module of mGlu8 receptor and the activation process: Insights from mutations converting antagonists into agonists

Philippe Rondard

Proceedings of the National Academy of Sciences, 2002

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Identification of essential residues involved in the glutamate binding pocket of the group II metabotropic glutamate receptor

Vincent Mutel

Molecular Pharmacology, 2001

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The C Terminus of the Metabotropic Glutamate Receptor Subtypes 2 and 7 Specifies the Receptor Signaling Pathways

Gustavo Gutierrez

Journal of Biological Chemistry, 2001

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Allosteric modulation of metabotropic glutamate receptors: Structural insights and therapeutic potential

Jeffrey Conn

Neuropharmacology, 2011

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Cloning, Distribution and Functional Expression of the Human mGlu6 Metabotropic Glutamate Receptor

B. Sommer

Neuropharmacology, 1997

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Metabotropic Glutamate Receptors: Physiology, Pharmacology, and Disease

Jeffrey Conn

Annual Review of Pharmacology and Toxicology, 2010

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Metabotropic Glutamate 1 Receptor: Current Concepts and Perspectives

Francesco Ferraguti

Pharmacological Reviews, 2008

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Metabotropic glutamate receptors

Katarzyna Ossowska

Amino Acids, 2007

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Molecular Pharmacology and Physiology of Glutamate Receptors

Raymond Dingledine

Glutamate and Addiction, 2002

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Functional identification of Gd3+ binding site of metabotropic glutamate receptor 1α

Hideki Abe

FEBS Letters, 2003

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Allosteric modulators of metabotropic glutamate receptors: lessons learnt from mGlu1, mGlu2 and mGlu5 potentiators and antagonists

Melvin Baez

Biochemical Society Transactions, 2004

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The Second Intracellular Loop of Metabotropic Glutamate Receptor 1 Cooperates with the Other Intracellular Domains to Control Coupling to G-proteins

Jean-philippe Pin

Journal of Biological Chemistry, 1996

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Transposition of Three Amino Acids Transforms the Human Metabotropic Glutamate Receptor (mGluR)-3-Positive Allosteric Modulation Site to mGluR2, and Additional Characterization of the mGluR2-Positive Allosteric Modulation Site □ S

Blake Rowe

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