Antiapoptotic BCL-2 proteins determine sorafenib/regorafenib resistance and BH3-mimetic efficacy in hepatocellular carcinoma (original) (raw)

Regorafenib Alteration of the BCL-xL/MCL-1 Ratio Provides a Therapeutic Opportunity for BH3-Mimetics in Hepatocellular Carcinoma Models

Loreto Boix

Cancers, 2020

View PDFchevron_right

Apoptotic blocks and chemotherapy resistance: strategies to identify Bcl2 protein signatures

Ozgur Gul

Briefings in Functional Genomics and Proteomics, 2008

View PDFchevron_right

Bcl-2 inhibitors: small molecules with a big impact on cancer therapy

Martin Dyer

Cell Death and Differentiation, 2009

View PDFchevron_right

Targeting the differential addiction to anti-apoptotic BCL-2 family for cancer therapy

Paul Jeng

Nature Communications, 2017

View PDFchevron_right

Unlocking the Therapeutic Potential of BCL-2 Associated Protein Family: Exploring BCL-2 Inhibitors in Cancer Therapy

Yasser Bustanji

Biomolecules & therapeutics, 2024

View PDFchevron_right

BH3-only protein expression determines hepatocellular carcinoma response to sorafenib-based treatment

Frank Essmann

Cell Death & Disease

View PDFchevron_right

Down-regulation of apoptosis-related bcl-2 but not bcl-xL or bax proteins in multidrug-resistant MCF-7/Adr human breast cancer cells

B. Ogretmen

International Journal of Cancer, 1996

View PDFchevron_right

Bax/Bak-independent mitochondrial depolarization and reactive oxygen species induction by sorafenib overcome resistance to apoptosis in renal cell carcinoma

Robert Preissner

The Journal of biological chemistry, 2017

View PDFchevron_right

Endogenous Bak inhibitors Mcl-1 and Bcl-xL: differential impact on TRAIL resistance in Bax-deficient carcinoma

Robert Preissner

Journal of Experimental Medicine, 2010

View PDFchevron_right

BCL-2 Family Inhibitors Enhance Histone Deacetylase Inhibitor and Sorafenib Lethality via Autophagy and Overcome Blockade of the Extrinsic Pathway to Facilitate Killing

Roland Reinehr

Molecular Pharmacology, 2009

View PDFchevron_right

Mitochondrial Bcl-2 Family Dynamics Define Therapy Response and Resistance in Neuroblastoma

Susan Peirce

Cancer Research, 2012

View PDFchevron_right

The Stress Protein BAG3 Stabilizes Mcl-1 Protein and Promotes Survival of Cancer Cells and Resistance to Antagonist ABT-737

Mariana Boiani

Journal of Biological Chemistry, 2013

View PDFchevron_right

Inhibition of Bcl-2 antiapoptotic members by obatoclax potently enhances sorafenib-induced apoptosis in human myeloid leukemia cells through a Bim-dependent process

Andrea Ferreira-Gonzalez

Blood, 2012

View PDFchevron_right

Bcl-2 Inhibition to Overcome Resistance to Chemo- and Immunotherapy

Marilina García Aranda

International Journal of Molecular Sciences, 2018

View PDFchevron_right

BCL-2 protein family: attractive targets for cancer therapy

deeksha kaloni

Apoptosis

View PDFchevron_right

Protect and serve: Bcl-2 proteins as guardians and rulers of cancer cell survival

Philippe Juin

Cell Cycle, 2013

View PDFchevron_right

Sensitizing non-small cell lung cancer to BCL-xL-targeted apoptosis

maricela ramirez

Cell death & disease, 2018

View PDFchevron_right

ABT-263 sensitizes TRAIL-resistant hepatocarcinoma cells by downregulating the Bcl-2 family of anti-apoptotic protein

Guan Wang

Cancer Chemotherapy and Pharmacology, 2011

View PDFchevron_right

Sorafenib sensitizes hepatocellular carcinoma cells to physiological apoptotic stimuli

Patricia Sancho, Isabel Fabregat, Conrado Rodriguez

Journal of Cellular Physiology, 2012

View PDFchevron_right

Preclinical Development The Bcl-2 / Bcl-XL / Bcl-w Inhibitor , Navitoclax , Enhances the Activity of Chemotherapeutic Agents In Vitro and In Vivo

Bernard Liu

2011

View PDFchevron_right

Cisplatin overcomes Bcl-2-mediated resistance to apoptosis via preferential engagement of Bak: critical role of Noxa-mediated lipid peroxidation

Maria Shoshan

Carcinogenesis, 2009

View PDFchevron_right

Targeting Bcl-2 Family of Proteins: An Important Strategy in Cancer Therapeutics

RAKESH R SOMANI

View PDFchevron_right

The Bcl-2 family: roles in cell survival and oncogenesis

David Huang

Oncogene, 2003

View PDFchevron_right

Bcl-2/Bcl-xL Inhibition Increases the Efficacy of MEK Inhibition Alone and in Combination with PI3 Kinase Inhibition in Lung and Pancreatic Tumor Models

Karen Williams

Molecular Cancer Therapeutics, 2013

View PDFchevron_right

Sorafenib induces apoptosis of AML cells via Bim-mediated activation of the intrinsic apoptotic pathway

Michael Andreeff

Leukemia, 2008

View PDFchevron_right

Proapoptotic BH3-Only BCL-2 Family Protein BIM Connects Death Signaling from Epidermal Growth Factor Receptor Inhibition to the Mitochondrion

Geoffrey Shapiro

Cancer Research, 2007

View PDFchevron_right

Co‐expression of Bcl‐2 protein and vascular endothelial growth factor in hepatocellular carcinomas treated by chemoembolization

Aditi Agarwal

Liver, 1999

View PDFchevron_right

Breast Cancer Cells Can Evade Apoptosis-Mediated Selective Killing by a Novel Small Molecule Inhibitor of Bcl-2

Zaneta Nikolovska-Coleska

Cancer Research, 2004

View PDFchevron_right

Downregulation of Bcl-xL and Mcl-1 is sufficient to induce cell death in mesothelioma cells highly refractory to conventional chemotherapy

Elena Varin

Carcinogenesis, 2010

View PDFchevron_right

Overexpression of Bcl-xs Sensitizes MCF-7 Cells to Chemotherapy-induced Apoptosis1

Venil N Sumantran

View PDFchevron_right

Integrated analysis of multiple receptor tyrosine kinases identifies Axl as a therapeutic target and mediator of resistance to sorafenib in hepatocellular carcinoma

Jamie Beaumont

British Journal of Cancer

View PDFchevron_right

The Bcl-2/Bcl-XL/Bcl-w Inhibitor, Navitoclax, Enhances the Activity of Chemotherapeutic Agents in vitro and in vivo

Bernard Liu

Molecular Cancer …, 2011

View PDFchevron_right

Small-molecule inhibitors of Bcl-2 family proteins as therapeutic agents in cancer

Anton-Scott Goustin

Recent patents on anti-cancer drug discovery, 2008

View PDFchevron_right

Synergistic induction of apoptosis by the Bcl-2 inhibitor ABT-737 and imatinib mesylate in gastrointestinal stromal tumor cells

David Mendiola Reynoso

Molecular Oncology, 2010

View PDFchevron_right

Targeting BCL-2 in Cancer: Advances, Challenges, and Perspectives

Mohamed Rahmani

Cancers, 2021

View PDFchevron_right