Palbociclib in Hormone-Receptor-Positive Advanced Breast Cancer - PubMed (original) (raw)
Clinical Trial
. 2015 Jul 16;373(3):209-19.
doi: 10.1056/NEJMoa1505270. Epub 2015 Jun 1.
Jungsil Ro, Fabrice André, Sherene Loi, Sunil Verma, Hiroji Iwata, Nadia Harbeck, Sibylle Loibl, Cynthia Huang Bartlett, Ke Zhang, Carla Giorgetti, Sophia Randolph, Maria Koehler, Massimo Cristofanilli; PALOMA3 Study Group
Collaborators, Affiliations
- PMID: 26030518
- DOI: 10.1056/NEJMoa1505270
Free article
Clinical Trial
Palbociclib in Hormone-Receptor-Positive Advanced Breast Cancer
Nicholas C Turner et al. N Engl J Med. 2015.
Free article
Abstract
Background: Growth of hormone-receptor-positive breast cancer is dependent on cyclin-dependent kinases 4 and 6 (CDK4 and CDK6), which promote progression from the G1 phase to the S phase of the cell cycle. We assessed the efficacy of palbociclib (an inhibitor of CDK4 and CDK6) and fulvestrant in advanced breast cancer.
Methods: This phase 3 study involved 521 patients with advanced hormone-receptor-positive, human epidermal growth factor receptor 2-negative breast cancer that had relapsed or progressed during prior endocrine therapy. We randomly assigned patients in a 2:1 ratio to receive palbociclib and fulvestrant or placebo and fulvestrant. Premenopausal or perimenopausal women also received goserelin. The primary end point was investigator-assessed progression-free survival. Secondary end points included overall survival, objective response, rate of clinical benefit, patient-reported outcomes, and safety. A preplanned interim analysis was performed by an independent data and safety monitoring committee after 195 events of disease progression or death had occurred.
Results: The median progression-free survival was 9.2 months (95% confidence interval [CI], 7.5 to not estimable) with palbociclib-fulvestrant and 3.8 months (95% CI, 3.5 to 5.5) with placebo-fulvestrant (hazard ratio for disease progression or death, 0.42; 95% CI, 0.32 to 0.56; P<0.001). The most common grade 3 or 4 adverse events in the palbociclib-fulvestrant group were neutropenia (62.0%, vs. 0.6% in the placebo-fulvestrant group), leukopenia (25.2% vs. 0.6%), anemia (2.6% vs. 1.7%), thrombocytopenia (2.3% vs. 0%), and fatigue (2.0% vs. 1.2%). Febrile neutropenia was reported in 0.6% of palbociclib-treated patients and 0.6% of placebo-treated patients. The rate of discontinuation due to adverse events was 2.6% with palbociclib and 1.7% with placebo.
Conclusions: Among patients with hormone-receptor-positive metastatic breast cancer who had progression of disease during prior endocrine therapy, palbociclib combined with fulvestrant resulted in longer progression-free survival than fulvestrant alone. (Funded by Pfizer; PALOMA3 ClinicalTrials.gov number, NCT01942135.).
Comment in
- Breast cancer: PALOMA-3 confirms that CDK4/6 is a key therapeutic target.
Errico A. Errico A. Nat Rev Clin Oncol. 2015 Aug;12(8):436. doi: 10.1038/nrclinonc.2015.113. Epub 2015 Jun 30. Nat Rev Clin Oncol. 2015. PMID: 26122184 No abstract available. - Palbociclib--Taking Breast-Cancer Cells Out of Gear.
Carey LA, Perou CM. Carey LA, et al. N Engl J Med. 2015 Jul 16;373(3):273-4. doi: 10.1056/NEJMe1506680. N Engl J Med. 2015. PMID: 26176385 No abstract available. - Palbociclib in Hormone-Receptor-Positive Advanced Breast Cancer.
Turner NC, Huang Bartlett C, Cristofanilli M. Turner NC, et al. N Engl J Med. 2015 Oct 22;373(17):1672-3. doi: 10.1056/NEJMc1510345. N Engl J Med. 2015. PMID: 26488700 No abstract available. - Palbociclib in Hormone-Receptor-Positive Advanced Breast Cancer.
Ozaki A, Tanimoto T, Saji S. Ozaki A, et al. N Engl J Med. 2015 Oct 22;373(17):1672-3. doi: 10.1056/NEJMc1510345. N Engl J Med. 2015. PMID: 26488701 No abstract available.
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