Halogenated triazinediones behave as antagonist of PKR1: in -vitro and in-vivo pharmacological characterization (original) (raw)

Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization

Cenzo Congiu, Valentina Onnis

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A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

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Orally Active Peptidic Bradykinin B1 Receptor Antagonists Engineered from a Cyclotide Scaffold for Inflammatory Pain Treatment

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Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel

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Recent advances in neurokinin-3 receptor antagonists

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Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

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Selective agonists for substance P and neurokinin receptors

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Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework

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Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics

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Prokineticin receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

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