Selective glycosidase inhibitors: A patent review (2012-present) (original) (raw)
Tetrahedron report number 773 a-and b-Glucosidase inhibitors: chemical structure and biological activity
man U
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and β-Glucosidase inhibitors: chemical structure and biological activity
Eduardo Melo
Tetrahedron, 2006
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α- and β-Glucosidase Inhibitors: Chemical Structure and Biological Activity
Ivone Carvalho
ChemInform, 2007
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Back to (non-)Basics: An Update on Neutral and Charge-Balanced Glycosidase Inhibitors
Todd Houston
Mini reviews in medicinal chemistry, 2017
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TARGETING GLYCOSYLATION AS A THERAPEUTIC APPROACH
Nicole Zitzmann
Nature Reviews Drug Discovery, 2002
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Back to (non)-Basics: Recent Developments in Neutral and Charge- Balanced Glycosidase Inhibitors
Todd Houston
Mini-Reviews in Medicinal Chemistry, 2003
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Sugar-mimic glycosidase inhibitors: natural occurrence, biological activity and prospects for therapeutic application
George Fleet
Tetrahedron: Asymmetry, 2000
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Iminosugars as glycosyltransferase inhibitors
Alberto Marra
Organic & Biomolecular Chemistry, 2021
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Synthesis of new six-and seven-membered 1-N-iminosugars as promising glycosidase inhibitors
Sanjay Chavan
Bioorganic & Medicinal …, 2011
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Synthesis of Hybrids of D‐Glucose and D‐Galactose with Pyrrolidine‐Based Iminosugars as Glycosidase Inhibitors
Girish Rawal
European Journal of …, 2008
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Glycosidase inhibitors from the roots of Glyphaea brevis
Abdulmagid Magid, Dominique Harakat
Phytochemistry, 2015
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The Two Faces of Iminoalditols: Powerful Inhibitors Trigger Glycosidase Activation
Current Enzyme Inhibition
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Enzyme Inhibitors as Therapeutic Tools
Mahmoud Balbaa
Biochemistry & Physiology: Open Access, 2012
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Synthesis and evaluation of sulfamide-type indolizidines as glycosidase inhibitors
José Fernández, Anne Wadouachi
Bioorganic & Medicinal Chemistry Letters, 2008
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A drug targeting motif for glycosidase inhibitors: an iminosugar–boronate shows unexpectedly selective β-galactosidase inhibition
Todd Houston
Tetrahedron Letters, 2002
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Synthetic studies in butenonyl C-glycosides: Preparation of polyfunctional alkanonyl glycosides and their enzyme inhibitory activity
Rama P Tripathi
Bioorganic & Medicinal Chemistry Letters, 2009
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Enzyme inhibition by iminosugars: Analysis and insight into the glycosidase–iminosugar dependency of pH
Mikael Bols
Bioorganic & Medicinal Chemistry, 2013
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Glycosidase Inhibition: An Assessment of the Binding of 18 Putative Transition-State Mimics
Andrea Vasella
Journal of the American Chemical Society, 2007
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Cyclic Guanidino-Sugars with Low p K a as Transition-State Analog Inhibitors of Glycosidases: Neutral Instead of Charged Species Are the Active Forms
Jin-hyun Jeong
Journal of the American Chemical Society, 1996
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Solid-phase enzyme-linked assay for the screening of glycosidase activities and inhibitors
Charles Tellier
Biotechnology Techniques
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Glycosyltransferase and Glypiation Inhibitors
Ishtiaq Ahmad
Current Organic Chemistry, 2007
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4-C-Me-DAB and 4-C-Me-LAB—enantiomeric alkyl-branched pyrrolidine iminosugars—are specific and potent α-glucosidase inhibitors; acetone as the sole protecting group
George Fleet
Tetrahedron Letters, 2011
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Improved cellular inhibitors for glycoprotein processing α-glucosidases: biological characterisation of alkyl- and arylalkyl-N-substituted deoxynojirimycins
raymond dwek
Tetrahedron: Asymmetry, 2009
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Potential role of glycosidase inhibitors in industrial biotechnological applications
Laura Camardella
Biochimica Et Biophysica Acta-proteins and Proteomics, 2004
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The Structural Basis of Glycosidase Inhibition by Five‐Membered Iminocyclitols: The Clan A Glycoside Hydrolase Endoglycoceramidase as a Model System
Andrea Vasella
Angewandte Chemie International Edition, 2007
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Synthesis and evaluation as glycosidase inhibitors of 2,5-imino-d-glucitol and 1,5-imino-d-mannitol related derivatives
Matthias Böhm
Bioorganic & Medicinal Chemistry, 2000
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A novel class of glycosidase inhibitors: structures related to australine, lentiginosine, salacinol and swainsonine
Sharwan Kumar
2007
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Synthesis and evaluation of d-gluco-pyranocyclopropyl amines as potential glucosidase inhibitors
Martijn D P Risseeuw
Bioorganic & Medicinal Chemistry Letters, 2009
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Synthesis and evaluation of a bicyclic deo×ymannojirimycin derivative as a potential glycosidase inhibitor
Kelly Tanaka
Canadian Journal of Chemistry-revue Canadienne De Chimie, 1998
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