New conformationally homogeneous β‐turn antagonists of the human B2 kinin receptor (original) (raw)

New conformationally homogeneous ?-turn antagonists of the human B2 kinin receptor

Andrea Madami

Journal of Peptide Science, 2001

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Structure-based design of six novel classes of nonpeptide antagonists of the bradykinin B2 receptor

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Bioorganic & Medicinal Chemistry Letters, 2000

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Structure activity relationships of non-peptide bradykinin B2 receptor antagonists

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Bioorganic & Medicinal Chemistry Letters, 1995

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Synthesis and Characterization of Bradykinin B 2 Receptor Agonists Containing Constrained Dipeptide Mimics

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In Vitro Pharmacological Profile of a New Small Molecule Bradykinin B2 Receptor Antagonist

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2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists

Cuyue Tang

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The nonpeptide WIN 64338 is a bradykinin B2 receptor antagonist

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Proceedings of the National Academy of Sciences, 1994

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Novel Subtype-Selective Nonpeptide Bradykinin Receptor Antagonists FR167344 and FR173657

Hitoshi Kojo

Molecular Pharmacology, 1997

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Synthesis and biological activity of new bradykinin pseudopeptide B1 receptor agonists containing alkylic spacers

Mariella Tancredi

Bioorganic & Medicinal Chemistry Letters, 1997

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Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide series

Christina Marco

Bioorganic & Medicinal Chemistry Letters, 2007

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A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity

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Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile

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Bioorganic & Medicinal Chemistry Letters, 2008

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Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides

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Journal of Medicinal Chemistry, 2007

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A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor

Jean-Philippe Fortin

International Immunopharmacology, 2003

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A Proposed Model of Bradykinin Bound to the Rat B2 Receptor and Its Utility for Drug Design

Sarvajit Chakravarty

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Synthesis and structure–Activity relationships of aroylpyrrole alkylamide bradykinin (B 2) antagonists

Scott Dax

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Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. Synthesis and structure-relationships of α,α-tetrahydropyranylglycine

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α-Hydroxy amides as a novel class of bradykinin B1 selective antagonists

Scott Mosser

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2,3-Diaminopyridine Bradykinin B1 Receptor Antagonists

Cuyue Tang

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Discovery of dihydroquinoxalinone acetamides containing bicyclic amines as potent Bradykinin B1 receptor antagonists

Ben Askew

Bioorganic & Medicinal Chemistry Letters, 2008

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Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists

Alessandro Giolitti, Francesca Bellucci

Biochemical Pharmacology, 2004

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Alpha-hydroxy amides as a novel class of bradykinin B1 selective antagonists

Scott Mosser

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Aspartic acid scaffold in bradykinin B1 antagonists

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Potent bradykinin B1 receptor antagonists: 4-Substituted phenyl cyclohexanes

Cuyue Tang

Bioorganic & Medicinal Chemistry Letters, 2007

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MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization

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European Journal of Pharmacology, 2005

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