Structure-based design of six novel classes of nonpeptide antagonists of the bradykinin B2 receptor (original) (raw)

Structure activity relationships of non-peptide bradykinin B2 receptor antagonists

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Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists

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α-Hydroxy amides as a novel class of bradykinin B1 selective antagonists

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Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides

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Alpha-hydroxy amides as a novel class of bradykinin B1 selective antagonists

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2,3-Diaminopyridine Bradykinin B1 Receptor Antagonists

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Rationally designed non-peptides: Variously substituted piperazine libraries for the discovery of bradykinin antagonists and other G-protein-coupled receptor ligands

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Conformational properties of a cyclic peptide bradykinin B2 receptor antagonist using experimental and theoretical methods

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Discovery of dihydroquinoxalinone acetamides containing bicyclic amines as potent Bradykinin B1 receptor antagonists

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Further pharmacological evaluation of a novel synthetic peptide bradykinin B2 receptor agonist

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