Design, synthesis and evaluation of 2,4-disubstituted pyrimidines as cholinesterase inhibitors (original) (raw)

New Pyrimidine and Pyridine Derivatives as Multitarget Cholinesterase Inhibitors: Design, Synthesis, and In Vitro and In Cellulo Evaluation

ACS Chemical Neuroscience, 2021

View PDFchevron_right

Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors

Annarita Stringaro

Pharmaceuticals

View PDFchevron_right

Cholinesterase Inhibition by Derivatives of 2-Amino-4,6-Dimethylpyridine

Journal of Enzyme Inhibition and Medicinal Chemistry, 1997

View PDFchevron_right

Design, Synthesis and Cholinesterase Inhibitory Activity of New Dispiro Pyrrolidine Derivatives

Social Science Research Network, 2022

View PDFchevron_right

Microwave assisted synthesis, cholinesterase enzymes inhibitory activities and molecular docking studies of new pyridopyrimidine derivatives

Bioorganic & Medicinal Chemistry, 2013

View PDFchevron_right

Synthesis and discovery of highly functionalized mono- and bis-spiro-pyrrolidines as potent cholinesterase enzyme inhibitors

Bioorganic & Medicinal Chemistry Letters, 2014

View PDFchevron_right

Synthesis, cytotoxicity and molecular modelling studies of new phenylcinnamide derivatives as potent inhibitors of cholinesterases

European Journal of Medicinal Chemistry, 2014

View PDFchevron_right

Synthesis and cholinesterase inhibitory activity of some phenylacetamide derivatives bearing 1H-pyrazole and 1H-1,2,4-triazole

MARMARA PHARMACEUTCAL JOURNAL, 2015

View PDFchevron_right

Synthesis, Biological Evaluation and Molecular Docking Study of Hydrazone-Containing Pyridinium Salts as Cholinesterase Inhibitors

Chemical & Pharmaceutical Bulletin, 2016

View PDFchevron_right

Sulfonamide Derivatives of 2-Amino-1-phenylethane as Suitable Cholinesterase Inhibitors

Dr. Shahid Rasool

Tropical Journal of Pharmaceutical Research, 2014

View PDFchevron_right

New multifunctional agents and their inhibitory effects on the acetyl cholinesterase enzyme

Macedonian Journal of Chemistry and Chemical Engineering

View PDFchevron_right

Synthesis and molecular modeling studies of cholinesterase inhibitor dispiro[indoline-3,2′-pyrrolidine-3′,3′′-pyrrolidines]

RSC Advances

View PDFchevron_right

Acetylcholinesterase enzyme inhibitor activity of some novel pyrazinamide condensed 1,2,3,4-tetrahydropyrimidines

Biotechnology Reports, 2015

View PDFchevron_right

Preparation, in vitro evaluation and molecular modelling of pyridinium–quinolinium/isoquinolinium non-symmetrical bisquaternary cholinesterase inhibitors

View PDFchevron_right

Synthesis, biological evaluation, QSAR study and molecular docking of novel N-(4-amino carbonylpiperazinyl) (thio)phosphoramide derivatives as cholinesterase inhibitors

View PDFchevron_right

2-Phenitidine derivatives as suitable inhibitors of butyrylcholinesterase

Dr. Muhammad Athar Abbasi

Brazilian Journal of Pharmaceutical Sciences, 2013

View PDFchevron_right

Synthesis and Acetylcholinesterase/Butyrylcholinesterase Inhibition Activity of 4-Amino-2, 3-diaryl-5, 6, 7, 8-tetrahydrofuro(and thieno)[2, 3-b]-quinolines, and 4-Amino-5, 6, 7, 8, 9-pentahydro-2, 3-diphenylcyclohepta[e]furo(and thieno)-[2, 3-b]pyridines

Maria C D C S A Carreiras

Archiv der Pharmazie, 2002

View PDFchevron_right