A Streamlined Asymmetric Synthesis of Substituted Geissman-Waiss Lactones, Oseltamivir precursors and peptidyl hydroxylactams from (–)-Azidocyclohexenol (original) (raw)

Furan‐Derived Chiral Bicycloaziridino Lactone Synthon: Collective Syntheses of Oseltamivir Phosphate (Tamiflu), ( S )‐Pipecolic acid and its 3‐Hydroxy Derivatives

Subhash Chavan

Chemistry – An Asian Journal, 2020

View PDFchevron_right

Short Chemoenzymatic Azide-Free Synthesis of Oseltamivir ACHTUNGTRENNUNG(Tamiflu): Approaching the Potential for Process Efficiency

Lukas Werner

2010

View PDFchevron_right

Synthesis of Several Cleistrioside and Cleistetroside Natural Products via a Divergent De Novo Asymmetric Approach

George O'Doherty

Organic Letters, 2010

View PDFchevron_right

An Asymmetric Domino Three-Component Synthesis of β-Lactams

Claudio Palomo

European Journal of Organic Chemistry, 1998

View PDFchevron_right

Several Generations of Chemoenzymatic Synthesis of Oseltamivir (Tamiflu): Evolution of Strategy, Quest for a Process-Quality Synthesis, and Evaluation of Efficiency Metrics

Aleš Machara

The Journal of Organic Chemistry, 2011

View PDFchevron_right

Short Chemoenzymatic Azide-Free Synthesis of Oseltamivir (Tamiflu): Approaching the Potential for Process Efficiency

Lukas Werner

Advanced Synthesis & Catalysis, 2010

View PDFchevron_right

Enantioselective and Convergent Synthesis of the 20-Membered Lactam Aglycon of Vicenistatin Antitumor Antibiotic

Yoshitaka Matsushima

The Journal of Antibiotics, 1998

View PDFchevron_right

Catalytic Asymmetric Synthesis of trans-Configured β-Lactones: Cooperation of Lewis Acid and Ion Pair Catalysis

Jose Cabrera

Chemistry - A European Journal, 2010

View PDFchevron_right

A Multicomponent Protocol for the Synthesis of Highly Functionalized γ-Lactam Derivatives and Their Applications as Antiproliferative Agents

Edorta Martínez de Marigorta

Pharmaceuticals

View PDFchevron_right

Versatility of β-lactams in synthesis. Studies directed toward the synthesis of complex nucleoside antibiotics and some macrocyclic peptides

Claudio Palomo

Pure and Applied Chemistry, 2000

View PDFchevron_right

Facile Conversion of α-Acyloxy Amides into 3-Hydroxy-lactams

Arleta Madej

European Journal of Organic Chemistry, 2018

View PDFchevron_right

Asymmetric Synthesis of N,OHeterobicyclic Octanes and ()-GeissmanWaiss Lactone

DR MOHD TAJUDIN MOHD ALI

View PDFchevron_right

Bis-N-aryl-β-lactams: Vilsmeier Reagent as an efficient entity for the Synthesis via Alternate Cycloaddition Reaction and In vitro Biology

Rajendra S U K H A D E O R A O Dongre

2010

View PDFchevron_right

Synthesis of (-)-Geissman Waiss Lactone, cis gamma-butyrolactone derivatives and gamma-peptides

DR MOHD TAJUDIN MOHD ALI

2012

View PDFchevron_right

Insight Into Transannular Cyclization Reactions To Synthesize Azabicyclo[X.Y.Z]alkanone Amino Acid Derivatives From 8-, 9- and 10-Member Macrocyclic Dipeptide Lactams

N D Prasad Atmuri

The Journal of organic chemistry, 2015

View PDFchevron_right

Asymmetric Synthesis of a Hydroxylated Nine-membered Lactone from Tartaric Acid using the Claisen Rearrangement

Jonathan White

Australian Journal of Chemistry, 2010

View PDFchevron_right

Asymmetric synthesis of 2-alkyl-substituted 2-hydroxyglutaric acid γ-lactones

Tõnis Kanger

Tetrahedron Letters, 2006

View PDFchevron_right

Enantioselective synthesis of oseltamivir phosphate

Raghavan S, Vari Babu

Tetrahedron, 2011

View PDFchevron_right

Access to novel bicyclic fused γ-butyrolactone using [3,3]-sigmatropic rearrangement and acid-lactonization sequence as key transformation

isabelle gillaizeau

Tetrahedron Letters, 2010

View PDFchevron_right

Asymmetric Synthesis of α- and β-Benzylhydroxy-γ-butyrolactones

Rafael Chinchilla

Synlett, 2010

View PDFchevron_right

Expedient Approach to α,β-Unsaturated δ-Lactones through a Catalytic Asymmetric [2+2] Cycloaddition

Régis Guillot

European Journal of Organic Chemistry, 2017

View PDFchevron_right

Advances in the chemistry of ?-lactam and its medicinal applications

Iwao Ojima

Tetrahedron, 2012

View PDFchevron_right

Synthesis of potential γ-lactam antibiotics

Raphaël Schneider

Bioorganic & Medicinal Chemistry Letters, 1995

View PDFchevron_right

Synthetic studies directed towards (–)-Chrysanthone A: Facile synthesis of a tricyclic lactone intermediate

Biswajit Panda

2019

View PDFchevron_right

Thiol-Free Synthesis of Oseltamivir and Its Analogues via Organocatalytic Michael Additions of Oxyacetaldehydes to 2-Acylaminonitroalkenes

Štefan Toma

Synthesis, 2012

View PDFchevron_right

Three-component synthesis of functionalized five-membered ring lactones under Barbier-like conditions

Erwan Le Gall

Tetrahedron Letters, 2009

View PDFchevron_right

Stereoselective solid-phase synthesis of 3,4-substituted azetidinones as key intermediates for mono- and multicyclic β-lactam antibiotics and enzyme inhibitors

Ernesto Mata

Tetrahedron-asymmetry, 2002

View PDFchevron_right

Enantioselective syntheses of isoprostane and iridoid lactones intermediates by enzymatic transesterification

Giovanni Vidari

Tetrahedron: Asymmetry, 2001

View PDFchevron_right

Natural and Synthetic Lactones Possessing Antitumor Activities

Sandip Sengupta

International Journal of Molecular Sciences, 2021

View PDFchevron_right

Asymmetric Synthesis of Highly Substituted ?-Lactones by Nucleophile-Catalyzed [2+2] Cycloadditions of Disubstituted Ketenes with Aldehydes

Mahbub ul Alam

Angewandte Chemie International Edition, 2004

View PDFchevron_right

Asymmetric Hydroformylation of an Enantiomerically Pure Bicyclic Lactam: Efficient Synthesis of Functionalised Cyclopentylamines

Christopher Cobley

Chemistry - A European Journal, 2010

View PDFchevron_right

A Formal Total Synthesis of Virantmycin: A Modular Approach towards Tetrahydroquinoline Natural Products

Stefan Braese

European Journal of Organic Chemistry, 2006

View PDFchevron_right

Sterically guided rearrangement of 3,3-disubstited β-lactones. A rapid construction of cycloheptano trans-fused butyrolactones

Shane Eisenbeis

Tetrahedron Letters, 1990

View PDFchevron_right

Two-step Synthesis of New γ-Lactones via Cyclization of 7-Chloro-2-(methoxycarbonyl)-4-6-dimethylocta-(2 E ,4 E ,6 E )-trienoic acid

Professeur Labia

Journal of Heterocyclic Chemistry, 2015

View PDFchevron_right

Synthesis of Multicyclic β-Lactam Derivatives via Solid-Phase-Generated Ketenes

Luciana Mendez

Journal of Combinatorial Chemistry, 2010

View PDFchevron_right