Fluorine-18 labelled substituted benzazepines as potential radiotracers for imaging dopamine D1 receptors by positron emission tomography (original) (raw)
Comparison of two fluorine-18 labeled benzamide derivatives that bind reversibly to dopamine D2 receptors: In vitro binding studies and positron emission tomography
Thomas Morton
Synapse, 1996
View PDFchevron_right
[11C]A-69024: A potent and selective non-benzazepine radiotracer for in vivo studies of dopamine D1 receptors
Michael Kassiou
Nuclear Medicine and Biology, 1995
View PDFchevron_right
Synthesis and evaluation in rats of homologous series of [(18)F]-labeled dopamine D 2/3 receptor agonists based on the 2-aminomethylchroman scaffold as potential PET tracers
Martin Michel
EJNMMI research, 2015
View PDFchevron_right
Iodine-125 and fluorine-18 labeled aryl-1,4-dialkylpiperazines: potential radiopharmaceuticals for in vivo study of the dopamine uptake system
Marcian Van Dort
International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1992
View PDFchevron_right
Biodistribution of N-alkyl and N-fluoroalkyl derivatives of spiroperidol; radiopharmaceuticals for PET studies of dopamine receptors
Dae Yoon Chi
International Journal of …, 1986
View PDFchevron_right
Substituted benzamides as ligands for visualization of dopamine receptor binding in the human brain by positron emission tomography
Lars Farde
Proceedings of the National Academy of Sciences, 1985
View PDFchevron_right
Production of fluorine-18 labeled (3-N-methyl)benperidol for PET investigation of cerebral dopaminergic receptor binding
S. Moerlein
International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1992
View PDFchevron_right
Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors
C. Damblon
Arkivoc, 2006
View PDFchevron_right
Synthesis of ω-[18F]fluoroalkyl analogs of YM-09151-2 for the measurement of D2-dopamine receptors with PET
Masatoshi Itoh
International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1990
View PDFchevron_right
Synthesis and evaluation of an 18F-labeled dopa prodrug as a PET tracer for studying brain dopamine metabolism
Tadashi Nozaki
Nuclear Medicine and Biology, 1996
View PDFchevron_right
Radiosynthesis and Evaluation of [ 11 C]-(+)-4-Propyl-3,4,4a,5,6,10b-hexahydro-2 H -naphtho[1,2- b ][1,4]oxazin-9-ol as a Potential Radiotracer for in Vivo Imaging of the Dopamine D2 High-Affinity State with Positron Emission Tomography
ARMANDO GARCIA
Journal of Medicinal Chemistry, 2005
View PDFchevron_right
N-(3-[18F]fluoropropyl)-spiperone: The preferred 18F labeled spiperone analog for positron emission tomographic studies of the dopamine receptor
C. Dence
International Journal of Radiation Applications and Instrumentation. Part B. Nuclear Medicine and Biology, 1988
View PDFchevron_right
Synthesis and Pharmacological Evaluation of Fluorine-Containing D3 Dopamine Receptor Ligands
Zhude Tu
Journal of Medicinal Chemistry, 2011
View PDFchevron_right
Synthesis, Biodistribution, and Primate Imaging of Fluorine-18 Labeled 2β-Carbo-1‘-fluoro-2-propoxy-3β-(4-chlorophenyl)tropanes. Ligands for the Imaging of Dopamine Transporters by Positron Emission Tomography
Vernon Camp
Journal of Medicinal Chemistry, 2000
View PDFchevron_right
N-.omega.-Fluoroalkyl Analogs of (1R)-2.beta.-Carbomethoxy-3.beta.-(4-iodophenyl)tropane (.beta.-CIT): Radiotracers for Positron Emission Tomography and Single Photon Emission Computed Tomography Imaging of Dopamine Transporters
Ross Baldessarini
Journal of Medicinal Chemistry, 1994
View PDFchevron_right
Synthesis and evaluation of fluorine-substituted 1H-pyrrolo [2, 3-b] pyridine derivatives for dopamine D4 receptor imaging
Dae Yoon Chi
Bioorganic & medicinal …, 2004
View PDFchevron_right
Quality control procedure for 6-[18F]fluoro-L-DOPA: a presynaptic PET imaging ligand for brain dopamine neurons
Robert Cohen
Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1989
View PDFchevron_right
2- and 4-[18F]fluorotropapride, two specific D2 receptor ligands for positron emission tomography: N.C.A. syntheses and animal studies
Alain Plenevaux
International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1992
View PDFchevron_right
11C-SCH 39166, a selective ligand for visualization of dopamine-D1 receptor binding in the monkey brain using PET
Lars Farde
Psychopharmacology, 1991
View PDFchevron_right
A Comparison of 11C-Labeled L-DOPA and L-Fluorodopa as Positron Emission Tomography Tracers for the Presynaptic Dopaminergic System
Joakim Tedroff
Journal of Cerebral Blood Flow & Metabolism, 1999
View PDFchevron_right
A Comparative PET-study of five carbon-11 or fluorine-18 labelled salicylamides. Preparation and in vitro dopamine D-2 receptor binding
Lars Farde
International Journal of Radiation Applications and Instrumentation. Part B. Nuclear Medicine and Biology, 1991
View PDFchevron_right
Synthesis and initial PET imaging of new potential dopamine D3 receptor radioligands (E)-4,3,2-[11C]methoxy-N-4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl-cinnamoylamides
Bruce Mock
Bioorganic & Medicinal Chemistry, 2005
View PDFchevron_right
18F]Fluoro-l-dopa for the in vivo study of intracerebral dopamine
Gunter Firnau
International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1986
View PDFchevron_right
In vivo evaluation of [123I]-8-[4-[2-(5-Iodothienyl)]-4-oxobutyl]-3-methyl-1-phenyl-1, 3, 8-triazaspiro [4.5] decan-4-one as a potential dopamine D2 receptor radioligand …
Timothy Gotsick
Nuclear medicine and …, 1998
View PDFchevron_right
4-[ 18 F]Fluoro-L-m-Tyrosine: An L-3,4-Dihydroxyphenylalanine Analog for Probing Presynaptic Dopaminergic Function with Positron Emission Tomography
Sung-cheng Huang
Journal of Neurochemistry, 1989
View PDFchevron_right
Positron emission tomography imaging of dopamine D2 receptors using a highly selective radiolabeled D2 receptor partial agonist
Jinda Fan, Suwanna Vangveravong
NeuroImage, 2013
View PDFchevron_right
Dopamine D3 receptor antagonists: The quest for a potentially selective PET ligand. Part 3: Radiosynthesis and in vivo studies
Yiyun Huang
Bioorganic & Medicinal Chemistry Letters, 2009
View PDFchevron_right
Receptor binding and selectivity of three 11C-labelled dopamine receptor antagonists in the brain of Rhesus monkeys studied with positron emission tomography
Bengt Långström
Acta Neurologica Scandinavica, 1988
View PDFchevron_right