2- and 4-[18F]fluorotropapride, two specific D2 receptor ligands for positron emission tomography: N.C.A. syntheses and animal studies (original) (raw)

Production of fluorine-18 labeled (3-N-methyl)benperidol for PET investigation of cerebral dopaminergic receptor binding

S. Moerlein

International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1992

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Comparison of two fluorine-18 labeled benzamide derivatives that bind reversibly to dopamine D2 receptors: In vitro binding studies and positron emission tomography

Thomas Morton

Synapse, 1996

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Biodistribution of N-alkyl and N-fluoroalkyl derivatives of spiroperidol; radiopharmaceuticals for PET studies of dopamine receptors

Dae Yoon Chi

International Journal of …, 1986

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The use of [18F]4-fluorobenzyl iodide (FBI) in PET radiotracer synthesis: Model alkylation studies and its application in the design of dopamine D1 and D2 receptor-based imaging agents

Thomas Morton

Nuclear Medicine and Biology, 1993

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Synthesis, Biodistribution, and Primate Imaging of Fluorine-18 Labeled 2β-Carbo-1‘-fluoro-2-propoxy-3β-(4-chlorophenyl)tropanes. Ligands for the Imaging of Dopamine Transporters by Positron Emission Tomography

Vernon Camp

Journal of Medicinal Chemistry, 2000

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N-(3-[18F]fluoropropyl)-spiperone: The preferred 18F labeled spiperone analog for positron emission tomographic studies of the dopamine receptor

C. Dence

International Journal of Radiation Applications and Instrumentation. Part B. Nuclear Medicine and Biology, 1988

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Fluorine-18 labelled substituted benzazepines as potential radiotracers for imaging dopamine D1 receptors by positron emission tomography

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European Journal of Pharmacology, 1993

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Cyclopropyl-FLB 457: A PET Radioligand for Low Densities of Dopamine D2 Receptors

Sangram Nag

Bioorganic & medicinal …, 2008

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11C]Cyclopropyl-FLB 457: A PET radioligand for low densities of dopamine D 2 receptors

Jogeshwar Mukherjee, sankha chattopadhyay

Bioorganic & Medicinal Chemistry, 2008

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Synthesis and evaluation of an 18F-labeled dopa prodrug as a PET tracer for studying brain dopamine metabolism

Tadashi Nozaki

Nuclear Medicine and Biology, 1996

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Substituted benzamides as ligands for visualization of dopamine receptor binding in the human brain by positron emission tomography

Lars Farde

Proceedings of the National Academy of Sciences, 1985

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A Comparative PET-study of five carbon-11 or fluorine-18 labelled salicylamides. Preparation and in vitro dopamine D-2 receptor binding

Lars Farde

International Journal of Radiation Applications and Instrumentation. Part B. Nuclear Medicine and Biology, 1991

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The use of [18F] 4-fluorobenzyl iodide (FBI) in PET radiotracer synthesis: model alkylation studies and its application in the design of dopamine D1 and D2 receptor- …

Theresa Filtz

Nuclear medicine and …, 1993

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Radiodefluorination of 3-Fluoro-5-(2-(2-18F-thiazol-4-yl)ethynyl)benzonitrile ([18F]SP203), a Radioligand for Imaging Brain Metabotropic Glutamate Subtype-5 Receptors with Positron Emission Tomography, Occurs by Glutathionylation in Rat Brain

Amira Brown

Journal of Pharmacology and Experimental Therapeutics, 2008

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(−)-N-[11C]propyl-norapomorphine: a positron-labeled dopamine agonist for PET imaging of D2 receptors

Lawrence Kegeles

Nuclear Medicine and Biology, 2000

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Tissue Distribution, Autoradiography, and Metabolism of 4‐(2′‐Methoxyphenyl)‐1‐[2′‐[N‐2 ″‐Pyridinyl)‐p‐[18F] Fluorobenzamido] ethyl] piperazine (p‐[18F] MPPF), a New Serotonin 5‐HT1A Antagonist for Positron Emission Tomography

Alain Plenevaux

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Radiosynthesis and Preclinical Evaluation of 18F-F13714 as a Fluorinated 5-HT1A Receptor Agonist Radioligand for PET Neuroimaging

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Journal of Nuclear Medicine, 2012

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Synthesis of ω-[18F]fluoroalkyl analogs of YM-09151-2 for the measurement of D2-dopamine receptors with PET

Masatoshi Itoh

International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1990

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Fluorinated benzamide neuroleptics—2. Synthesis and radiosynthesis of (S)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(3-[18F]fluoropropyl)-3-substituted-2-methoxybenzamides

Jogeshwar Mukherjee

International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1991

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Binding of 5-(2′-[18F]fluoroenthyl)flumazenil to central benzodiazepine receptors measured in living baboon by positron emission tomography

S. Moerlein

European Journal of Pharmacology, 1992

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Positron labeled muscarinic acetylcholine receptor antagonist: 2- and 4-[18F]fluorodexetimide. Syntheses and biodistribution

Carmen S Dence

International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology, 1991

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Evaluation of fluorinated m-Tyrosine analogs as PET imaging agents of dopamine nerve terminals: comparison with 6-FluoroDOPA

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N-.omega.-Fluoroalkyl Analogs of (1R)-2.beta.-Carbomethoxy-3.beta.-(4-iodophenyl)tropane (.beta.-CIT): Radiotracers for Positron Emission Tomography and Single Photon Emission Computed Tomography Imaging of Dopamine Transporters

Ross Baldessarini

Journal of Medicinal Chemistry, 1994

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Iodine-125 and fluorine-18 labeled aryl-1,4-dialkylpiperazines: potential radiopharmaceuticals for in vivo study of the dopamine uptake system

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International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1992

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A Comparison of 11C-Labeled L-DOPA and L-Fluorodopa as Positron Emission Tomography Tracers for the Presynaptic Dopaminergic System

Joakim Tedroff

Journal of Cerebral Blood Flow & Metabolism, 1999

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