Investigation of Subsite Preferences in Aminopeptidase A (EC 3.4.11.7) Led to the Design of the First Highly Potent and Selective Inhibitors of This Enzyme (original ) (raw )Potent and systemically active aminopeptidase N inhibitors designed from active-site investigation
Bernard Roques
Journal of Medicinal Chemistry, 1992
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Tetrahedron, 2012
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Bioorganic & Medicinal Chemistry Letters, 1999
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Journal of Medicinal Chemistry, 1994
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Journal of Medicinal Chemistry, 2003
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Bioorganic & Medicinal Chemistry, 2014
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Bioorganic & Medicinal Chemistry, 2012
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Bioorganic & Medicinal Chemistry Letters, 2006
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C. Voltattorni
Life Sciences, 1982
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Angelo Fontana
Biochemistry, 1968
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The Journal of Organic Chemistry, 2006
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Piotr Wieczorek
Liebigs Annalen der Chemie, 1984
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Ayman El-Faham
Organic Preparations …, 2001
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Sk. Abdul Amin
Perspective, 2018
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Ayman El-Faham
ChemInform, 2012
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chi ming lee
European Journal of Biochemistry, 1981
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Advances in the evaluation of the stability and characteristics of the amino acid and amine derivatives obtained with the o-phthaldialdehyde/3-mercaptopropionic acid and o-phthaldialdehyde/N-acetyl-l-cysteine reagents
Antal CsÁmpai
Journal of Chromatography A, 2002
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Xiaozhang Zheng
Journal of Medicinal Chemistry, 2004
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Pawel Kafarski
Biochimie, 2010
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Binghe Wang
Bioorganic & Medicinal Chemistry, 2009
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Discovery and Optimization of Anthranilic Acid Sulfonamides as Inhibitors of Methionine Aminopeptidase-2: A Structural Basis for the Reduction of Albumin Binding
David Barnes
Journal of Medicinal Chemistry, 2006
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Investigation of the Active Site of Aminopeptidase A Using a Series of New Thiol-Containing Inhibitors
Sherwin Wilk
Journal of Medicinal Chemistry, 1994
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Prolyl Oligopeptidase Inhibition by N -Acyl-pro-pyrrolidine-type Molecules
Károly Kánai
Journal of Medicinal Chemistry, 2008
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Rational Design of Improved Aziridine-Based Inhibitors of Cysteine Proteases
Bernd Engels
The Journal of Physical Chemistry B, 2009
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