Synthesis of conformationally constrained potential inhibitors of mammalian metalloproteinases
Andrew Griffin
Bioorganic & Medicinal Chemistry Letters, 1997
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In silico scaffold evaluation and solid phase approach to identify new gelatinase inhibitors
Franco Minissi
Bioorganic & Medicinal Chemistry, 2012
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Design and synthesis of novel inhibitors of gelatinase B
Charles Craik
Bioorganic & Medicinal Chemistry Letters, 2002
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X-ray Absorption Studies of Human Matrix Metalloproteinase-2 (MMP-2) Bound to a Highly Selective Mechanism-based Inhibitor. COMPARISON WITH THE LATENT AND ACTIVE FORMS OF THE ENZYME
Oded Kleifeld
Journal of Biological Chemistry, 2001
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Amino Acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors
Ermelinda Vernieri, Alessia Bertamino, Isabel Gomez-monterrey, Armando Rossello
Journal of amino acids, 2013
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Conformational analyses of thiirane-based gelatinase inhibitors
Dusan Hesek, Jed Fisher
Bioorganic & Medicinal Chemistry Letters, 2008
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Insights into the Complex Formed by Matrix Metalloproteinase-2 and Alloxan Inhibitors: Molecular Dynamics Simulations and Free Energy Calculations
Gianluca Lattanzi
PloS one, 2011
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Pharmacophore identification for matrix metalloproteinases by in silico investigations
Carmen Cotrutz
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Extra Binding Region Induced by Non-Zinc Chelating Inhibitors into the S 1 ′ Subsite of Matrix Metalloproteinase 8 (MMP-8) †
Fernando Mazza
Journal of Medicinal Chemistry, 2009
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A Rationalization of the Acidic pH Dependence for Stromelysin-1 (Matrix Metalloproteinase-3) Catalysis and Inhibition
Chiu-Fai Man, Adam Johnson
Journal of Biological Chemistry, 2000
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Purification of Active Matrix Metalloproteinase Catalytic Domains and Its Use for Screening of Specific Stromelysin-3 Inhibitors
Marc Ruff
Protein Expression and Purification, 1999
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Synthesis of an array of potential matrix metalloproteinase inhibitors using a sequence of polymer-supported reagents
M. Caldarelli
Bioorganic & Medicinal Chemistry Letters, 1999
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A study on quantitative structure–activity relationship and molecular docking of metalloproteinase inhibitors based on L-tyrosine scaffold
Fatemeh Ramezani
DARU Journal of Pharmaceutical Sciences, 2015
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Structural Basis for Potent Slow Binding Inhibition of Human Matrix Metalloproteinase-2 (MMP-2)
gabriel rosenblum
Journal of Biological Chemistry, 2003
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Structure of matrix metalloproteinase-3 with a platinum-based inhibitor
Giovanni Natile
Chemical Communications, 2013
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Crystal Structures of MMP-9 Complexes with Five Inhibitors: Contribution of the Flexible Arg424 Side-chain to Selectivity
Wolfram Bode, Anna Tochowicz, Peter Goettig, K. Maskos
Journal of Molecular Biology, 2007
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Specificity of Binding with Matrix Metalloproteinases
VAISHALI MANIKRAO PATIL
Matrix Metalloproteinase Inhibitors, 2012
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Structural characterizations of nonpeptidic thiadiazole inhibitors of matrix metalloproteinases reveal the basis for stromelysin selectivity
Eric Baldwin
Protein Science, 1998
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X-ray structure of human stromelysin catalytic domain complexed with nonpeptide inhibitors: Implications for inhibitor selectivity
Christine Humblet
Protein Science, 1999
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Hydroxamate inhibitors of the matrix metallo-proteinases (MMPs) containing novel P1′ heteroatom based modifications
Bruce Tomczuk, Arup Ghose
Bioorganic & Medicinal Chemistry Letters, 1995
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QM/MM Studies of the Matrix Metalloproteinase 2 (MMP2) Inhibition Mechanism of (S)-SB-3CT and its Oxirane Analogue
Jed Fisher
Journal of Chemical Theory and Computation, 2010
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X-ray structure of a hydroxamate inhibitor complex of stromelysin catalytic domain and its comparison with members of the zinc metalloproteinase superfamily
Christine Humblet
Structure, 1996
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Pharmacomodulation of Broad Spectrum Matrix Metalloproteinase Inhibitors Towards Regulation of Gelatinases
János Sápi
Enzyme Inhibition and Bioapplications, 2012
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Design and synthesis of novel metalloproteinases inhibitors
Armando Rossello
2009
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New bifunctional metalloproteinase inhibitors: an integrated approach towards biological improvements and cancer therapy
Elisa Nuti, Armando Rossello
Journal of Inorganic Biochemistry, 2013
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Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies
Elisabetta Orlandini
Journal of medicinal chemistry, 2018
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