18 F-Fluorothiols: A New Approach To Label Peptides Chemoselectively as Potential Tracers for Positron Emission Tomography † (original) (raw)
18F-Labeling of Peptides by means of an Organosilicon-Based Fluoride Acceptor
Ralf Schirrmacher, Klaus Jurkschat
Angewandte Chemie International Edition, 2006
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Using 5-deoxy-5-[18F]fluororibose to glycosylate peptides for positron emission tomography
Anne Roivainen
Nature Protocols, 2013
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Sulfonyl Fluoride-Based Prosthetic Compounds as Potential 18 F Labelling Agents
Samia Ait-mohand
Chemistry - A European Journal, 2012
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One-step synthesis of 18F labeled [18F]-N-succinimidyl 4-(fluoromethyl)benzoate for protein labeling
William Eckelman
Applied Radiation and Isotopes, 1994
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Synthesis and Application of [ 18 F]FDG-Maleimidehexyloxime ([ 18 F]FDG-MHO): A [ 18 F]FDG-Based Prosthetic Group for the Chemoselective 18 F-Labeling of Peptides and Proteins
Ralf Bergmann
Bioconjugate Chemistry, 2008
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Use of 3-[ 18 F]fluoropropanesulfonyl chloride as a prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamides
Martin Köckerling
Beilstein Journal of Organic Chemistry, 2013
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Arylfluoroborates and Alkylfluorosilicates as Potential PET Imaging Agents: High-Yielding Aqueous Biomolecular 18 F-Labeling
Thomas Ruth
Journal of the American Chemical Society, 2005
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para -Functionalized Aryl-di- tert -butylfluorosilanes as Potential Labeling Synthons for 18 F Radiopharmaceuticals
Ralf Schirrmacher, Klaus Jurkschat
Chemistry - A European Journal, 2009
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1-[3-(2-[ 18 F]Fluoropyridin-3-yloxy)propyl]pyrrole-2,5-dione: Design, Synthesis, and Radiosynthesis of a New [ 18 F]Fluoropyridine-Based Maleimide Reagent for the Labeling of Peptides and Proteins
Raphaël Boisgard, Frédéric Dollé, Bertrand Tavitian
Bioconjugate Chemistry, 2005
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3,4,6-Tri- O -acetyl-2-deoxy-2-[ 18 F]fluoroglucopyranosyl Phenylthiosulfonate: A Thiol-Reactive Agent for the Chemoselective 18 F-Glycosylation of Peptides
Peter Gmeiner
Bioconjugate Chemistry, 2007
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Automated radiochemical synthesis of [18F]FBEM: A thiol reactive synthon for radiofluorination of peptides and proteins
Lixin Lang
Applied Radiation and Isotopes, 2011
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Kit-Like 18 F-Labeling of Proteins: Synthesis of 4-(Di- tert -butyl[ 18 F]fluorosilyl)benzenethiol (Si[ 18 F]FA-SH) Labeled Rat Serum Albumin for Blood Pool Imaging with PET
Klaus Jurkschat
Bioconjugate Chemistry, 2009
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Novel ( 18 F)Fluorinated Prosthetic Groups for the Labelling of Peptides for Positron Emission Tomography (PET)
Dag Erlend Olberg
2000
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Rapid and high-yielding cysteine labelling of peptides with N-succinimidyl 4-[18F]fluorobenzoate
Santiago Rojas
Chemical Communications, 2012
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Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase: a comparative study
Torsten Kniess
Amino Acids, 2012
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Oxalic Acid Supported Si– 18 F-Radiofluorination: One-Step Radiosynthesis of N -Succinimidyl 3-(Di- tert -butyl[ 18 F]fluorosilyl)benzoate ([ 18 F]SiFB) for Protein Labeling
Klaus Jurkschat
Bioconjugate Chemistry, 2012
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Radiosynthesis and Analysis of (S)-4-(3-[18F]Fluoropropyl)-L-Glutamic Acid
Dmitry Soloviev
Molecular Imaging and Biology, 2022
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One-step radiosynthesis of the MCTs imaging agent [18F]FACH by aliphatic 18F-labelling of a methylsulfonate precursor containing an unprotected carboxylic acid group
Masoud Sadeghzadeh
Scientific Reports
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Sulfonium Salts as Leaving Groups for Aromatic Labelling of Drug-like Small Molecules with Fluorine-18
Mark Lythgoe
Scientific Reports, 2015
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Fast and reliable method for the preparation of ortho-and para-[18 F] fluorobenzyl halide derivatives: key intermediates for the preparation of no-carrier-added PET aromatic radiopharmaceuticals
Alain Plenevaux
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The facile synthesis of a pyrimidinyl sulfonamide (N,N,N,6-tetramethyl-2-(4-nitrophenylsulfonamido)pyrimidin-4-ammonium chloride) as a PET tracer precursor
Hans-peter Saluz
Arkivoc, 2012
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Synthesis of 4-[18F]fluorobenzoyllisinopril: A radioligand for angiotensin converting enzyme (ACE) imaging with positron emission tomography
William Eckelman
Journal of Labelled Compounds and Radiopharmaceuticals, 2001
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A new precursor for the preparation of 6-[18F]Fluoro-l-m-tyrosine ([18F]FMT): efficient synthesis and comparison of radiolabeling
Alex Hoepping
Applied Radiation and Isotopes, 2004
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Use of Diethylaminosulfur Trifluoride in an Efficient Synthesis of (S)-N-[(1-Ethyl-2-Pyrrolidinyl)Methyl]-5-(3-Fluoropropyl-2-Methoxybenzamide
Jogeshwar Mukherjee
Journal of Fluorine Chemistry, 1990
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Synthesis of the positron-emitting radiotracer [18F]-2-fluoro-2-deoxy-d-glucose from resin-bound perfluoroalkylsulfonates
Alex Jackson
Organic & Biomolecular Chemistry, 2009
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A Rapid and Efficient Method for the Fluoroalkylation of Amines and Amides. Development of a Method Suitable for Incorporation of the Short-Lived Positron Emitting …
Dae Yoon Chi
The Journal of …, 1987
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One-step radiosynthesis of 4-nitrophenyl 2-[ 18 F]fluoropropionate ([ 18 F]NFP); improved preparation of radiolabeled peptides for PET imaging
Craig Hutton
Journal of Labelled Compounds and Radiopharmaceuticals, 2013
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N-(4-(di- tert-butyl[ 18F]fluorosilyl)benzyl)-2-hydroxy-N,N-dimethylethylammonium bromide ([ 18F]SiFAN +Br −): A novel lead compound for the development of hydrophilic SiFA-based prosthetic groups for 18F-labeling
Klaus Jurkschat
Journal of Fluorine Chemistry, 2011
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Fluorinated Diaryl Sulfides as Serotonin Transporter Ligands: Synthesis, Structure−Activity Relationship Study, and in Vivo Evaluation of Fluorine-18-Labeled Compounds as PET Imaging Agents
Yiyun Huang
Journal of Medicinal Chemistry, 2005
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First 18F-Labeled Tracer Suitable for Routine Clinical Imaging of sst Receptor-Expressing Tumors Using Positron Emission Tomography
Horst Kessler
Clinical Cancer Research, 2004
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A Simple On-column Preparation of [^<18>F]Fluorocholine from [^<18>F]Fluoromethyl Triflate
Claudio Pascali
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