original ) (raw )Synthesis of hexahydro[2]benzopyrano[3,4-c]pyrroles as serotonin 5-HT2C receptor agonists via intramolecular hetero Diels–Alder reactions
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Tetrahedron Letters, 2011
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Tetrahedron Letters, 2011
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ACS Medicinal Chemistry Letters, 2015
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Journal of Medicinal Chemistry, 1996
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SYNTHESIS AND FUNCTIONALIZATION OF THE PYRAZOLO [3,4-b]PYRIDIN-3-ONES RESEARCH OF THE SEROTONINERGIC ACTIVITY
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Moroccan Journal of Heterocyclic Chemistry, 2021
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3,4-Dihydro-3-amino-2H-1-benzopyran Derivatives as 5-HT1A Receptor Ligands and Potential Anxiolytic Agents. 1. Synthesis and Structure-Activity Relationship Studies
Tchao Podona
Journal of Medicinal Chemistry, 1994
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Substituted hexahydrobenzodipyrans as 5-HT2A/2C receptor probes
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Bioorganic & Medicinal Chemistry, 2002
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Martha Ramirez
2003
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Bioorganic & Medicinal Chemistry, 2009
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2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists
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European Journal of Medicinal Chemistry, 2011
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Synthesis and Structure Activity Relationship of Rigidized Indolyl Pyrrolidine Derivatives as 5-HT6 Receptor Ligands
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Asian Journal of Chemistry, 2013
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Novel and Selective Partial Agonists of 5-HT3 Receptors. 2. Synthesis and Biological Evaluation of Piperazinopyridopyrrolopyrazines, Piperazinopyrroloquinoxalines, and Piperazinopyridopyrroloquinoxalines
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Journal of Medicinal Chemistry, 1997
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Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT 6 Receptor Ligands
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ChemMedChem, 2013
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Journal of medicinal chemistry, 2011
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One-step synthesis of aminopyrimidines from 5Oxo4 H -benzopyrans
Estael Ochoa
Journal of Heterocyclic Chemistry, 2004
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Synthesis and Biological Evaluation of Novel 5,8-Disubstituted-2-methyl-2,3,4,5-tetrahydro-1 H -pyrido[4,3- b ] indoles as 5HT 6 and H 1 Receptors Antagonists
Maha Soltan
Archiv Der Pharmazie, 2009
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Design and Discovery of Functionally Selective Serotonin 2C (5-HT2C) Receptor Agonists
alan kozikowski
Journal of medicinal chemistry, 2016
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N 0 -(Arylsulfonyl)pyrazoline-1-carboxamidines as Novel, Neutral 5-Hydroxytryptamine 6 Receptor (5-HT 6 R) Antagonists with Unique Structural Features
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Monatshefte für Chemie - Chemical Monthly, 2009
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Bioorganic & Medicinal Chemistry, 2010
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Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT 2A receptor ligands
Lucjan Strekowski
Journal of Heterocyclic Chemistry, 2009
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Journal of Medicinal Chemistry, 1998
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Diastereoselective Synthesis of Some Novel Benzopyranopyridine Derivatives
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Beilstein Journal of …
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Further Structural Exploration of Trisubstituted Asymmetric Pyran Derivatives (2 S ,4 R ,5 R )-2-Benzhydryl-5-benzylamino-tetrahydropyran-4-ol and Their Corresponding Disubstituted (3 S ,6 S ) Pyran Derivatives: A Proposed Pharmacophore Model for High-Affinity Interaction with the Dopamine, Sero...
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Journal of Medicinal Chemistry, 2006
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Identification of 4-methyl-1,2,3,4,10,10a- hexahydropyrazino[1,2-a]indoles as 5-HT 2C receptor agonists
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One‐pot synthesis of 2‐amino‐4,8‐dihydropyrano[3,2‐b]pyranes and pyridopyrimidines under mild conditions
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Journal of the Chinese Chemical Society, 2018
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Novel benzopyrano[3,4-c]pyrrole derivatives as potent and selective dopamine D3 receptor antagonists
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Bioorganic & Medicinal Chemistry Letters, 1999
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Three-component condensation of diethyl 2,4,6-trioxoheptanedicarboxylate with salicylaldehyde and ammonium acetate as a new method for the synthesis of the [1]benzopyrano[4,3-b]pyridine system
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Russian Chemical Bulletin, 2005
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Preparation and Biological Evaluation of Some New 2-Amino-6- Aryl-3-Cyano 4-(M-Phenoxy Phenyl)-Pyridines
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Oriental journal of chemistry, 2001
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A New Class of Arylpiperazine Derivatives: the Library Synthesis on SynPhase Lanterns and Biological Evaluation on Serotonin 5-HT 1A and 5-HT 2A Receptors
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Journal of Combinatorial Chemistry, 2004
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