Sphingosine-1-phosphate receptor therapies: Advances in clinical trials for CNS-related diseases (original) (raw)

Sphingosine 1-Phosphate Receptors and Metabolic Enzymes as Druggable Targets for Brain Diseases

Paola Giussani

Frontiers in Pharmacology

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Sphingosine 1-Phosphate Receptor Modulators and Drug Discovery

F. Dahlke

Biomolecules & therapeutics, 2017

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Sphingosine 1-phosphate – A double edged sword in the brain

Gerhild van Echten-Deckert

Biochimica Et Biophysica Acta - Biomembranes, 2017

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The role of sphingosine 1-phosphate metabolism in brain health and disease

Gerhild van Echten-Deckert

Review, 2023

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Sphingosine 1-phosphate receptor modulator fingolimod (FTY720) does not promote remyelination in vivo

Giuseppe Faggian

Molecular and Cellular Neuroscience, 2011

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Sphingosine kinase 1/sphingosine-1-phosphate receptors dependent signalling in neurodegenerative diseases. The promising target for neuroprotection in Parkinson’s disease

Joanna B Strosznajder

Pharmacological Reports, 2018

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Sphingosine-1-Phosphate (S1P) and S1P Signaling Pathway Modulators, from Current Insights to Future Perspectives

René Robles-Cedeño

Cells

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Sphingosine-1-Phosphate Receptors: Zooming in on Ligand-Induced Intracellular Trafficking and Its Functional Implications

Dennis Verzijl

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Sphingosine-1-phosphate receptors mediate neuromodulatory functions in the CNS

Leslie Satin

Journal of Neurochemistry, 2009

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Sphingosine 1-phosphate Receptor Modulator Therapy for Multiple Sclerosis: Differential Downstream Receptor Signalling and Clinical Profile Effects

Samuel F Hunter

Drugs

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Emerging biology of sphingosine-1-phosphate: its role in pathogenesis and therapy

timothy hla

The Journal of clinical investigation, 2015

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Implication of sphingosine-1-phosphate signaling in diseases: molecular mechanism and therapeutic strategies

rahat ali

Journal of Receptors and Signal Transduction, 2017

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An update on sphingosine-1-phosphate receptor 1 modulators

Robin Polt

Bioorganic & Medicinal Chemistry Letters, 2018

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Sphingosine 1-Phosphate Receptor 1 Signaling in Mammalian Cells

Nigel Pyne

Molecules, 2017

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Sphingosine-1-Phosphate: Boon and Bane for the Brain

Gerhild van Echten-Deckert

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FTY720 (fingolimod) efficacy in an animal model of multiple sclerosis requires astrocyte sphingosine 1-phosphate receptor 1 (S1P1) modulation

yun yung

Proceedings of the National Academy of Sciences, 2011

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Sphingosine 1-Phosphate Receptor 1 (S1P1) Upregulation and Amelioration of Experimental Autoimmune Encephalomyelitis by an S1P1 Antagonist

Pedro Gonzalez-Cabrera

Molecular Pharmacology, 2012

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Sphingosin-1-phosphate Receptor 1: a Potential Target to Inhibit Neuroinflammation and Restore the Sphingosin-1-phosphate Metabolism

Leila Dargahi

The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques, 2015

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Immunohistochemical detection of sphingosine-1-phosphate receptor 1 in vascular and lymphatic endothelial cells

Rosanna Pescini Gobert

Journal of Molecular Histology, 2008

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Benefit–Risk Profile of Sphingosine-1-Phosphate Receptor Modulators in Relapsing and Secondary Progressive Multiple Sclerosis

Ian Williams

Drugs, 2017

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Regulation and functions of sphingosine kinases in the brain

Laurens Bryan

Biochimica Et Biophysica Acta-molecular and Cell Biology of Lipids, 2008

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Sphingosine 1-phosphate pathway therapeutics: a lipid ligand–receptor paradigm

jiayu liao

Current Opinion in Chemical Biology, 2003

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Immunohistochemical Detection of Sphingosine-1-Phosphate and Sphingosine Kinase-1 in Human Tissue Samples and Cell Lines

Roger Sabbadini

Methods in molecular biology, 2017

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Identification of Sphingosine 1-Phosphate Receptor Subtype 1 (S1P1) as a Pathogenic Factor in Transient Focal Cerebral Ischemia

arjun sapkota

Molecular neurobiology, 2017

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Functional antagonism of sphingosine-1-phosphate receptor 1 prevents cuprizone-induced demyelination

narjes dahmardeh

Glia, 2018

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Loss of the neuroprotective factor Sphingosine 1-phosphate early in Alzheimer's disease pathogenesis

J. Kril

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Cis-4-methylsphingosine is a sphingosine-1-phosphate receptor modulator

Dagmar zu Heringdorf, Bianca Hegen, Sandra Labocha, Gerhild van Echten-Deckert

Biochemical Pharmacology, 2011

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Modulators of the Sphingosine 1-phosphate receptor 1

miguel angel davila guerrero

Bioorganic & Medicinal Chemistry Letters, 2013

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Activation of sphingosine 1-phosphate receptor-1 by SEW2871 improves cognitive function in Alzheimer's disease model rats

Abolhassan Ahmadiani

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Sphingosine-1-Phosphate Receptors Modulators Decrease Signs of Neuroinflammation and Prevent Parkinson’s Disease Symptoms in the 1-Methyl-4-Phenyl-1,2,3,6-Tetrahydropyridine Mouse Model

Tim Jalinier

Frontiers in Pharmacology

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Sphingolipid Metabolism: A New Therapeutic Opportunity for Brain Degenerative Disorders

Alba Di Pardo

Frontiers in neuroscience, 2018

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Overexpression of sphingosine-1-phosphate receptors on reactive astrocytes drives neuropathology of multiple sclerosis rebound after fingolimod discontinuation

Fabio Bandini

Multiple Sclerosis Journal, 2018

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Selectivity and Specificity of Sphingosine-1-Phosphate Receptor Ligands: Caveats and Critical Thinking in Characterizing Receptor-Mediated Effects

Salvatore Salomone

Frontiers in Pharmacology, 2011

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Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate-1 Receptor

Jaimie Rueter

ACS medicinal chemistry letters, 2014

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