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Rune Risgaard
Molecular Pharmacology, 2013
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Structural Determinants of Agonist Efficacy at the Glutamate Binding Site ofN-Methyl-d-Aspartate Receptors
Rune Risgaard
Molecular Pharmacology, 2013
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Structure, function, and allosteric modulation of NMDA receptors
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Journal of General Physiology, 2018
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A Glutamate N-Methyl-d-Aspartate (NMDA) Receptor Subunit 2B–Selective Inhibitor of NMDA Receptor Function with Enhanced Potency at Acidic pH and Oral Bioavailability for Clinical Use
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Journal of Pharmacology and Experimental Therapeutics, 2021
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Heteromerization of Ligand Binding Domains of N-Methyl-d-Aspartate Receptor Requires Both Coagonists, l-Glutamate and Glycine
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Biochemistry, 2015
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Influence of GluN2 subunit identity on NMDA receptor function
Giles Hardingham
Neuropharmacology, 2013
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Structure–activity relationships of N-substituted 4-(trifluoromethoxy)benzamidines with affinity for GluN2B-containing NMDA receptors
Michael Kassiou, John Tsanaktsidis, Albert Windhorst
Bioorganic & Medicinal Chemistry Letters, 2014
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Subunit arrangement and function in NMDA receptors
satinder singh
Nature, 2005
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Faculty of 1000 evaluation for Arrangement of subunits in functional NMDA receptors
Robert Peoples
F1000 - Post-publication peer review of the biomedical literature, 2011
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Subtype-Specific Agonists for NMDA Receptor Glycine Binding Sites
Papangelis Athanasios
ACS chemical neuroscience, 2017
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Faculty of 1000 evaluation for Chimeric Glutamate Receptor Subunits Reveal the Transmembrane Domain Is Sufficient for NMDA Receptor Pore Properties but Some Positive Allosteric Modulators Require Additional Domains
Robert Peoples
F1000 - Post-publication peer review of the biomedical literature
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Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity
Christian Madry
Frontiers in Pharmacology
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Faculty Opinions recommendation of Structure, function, and allosteric modulation of NMDA receptors
Robert Peoples
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
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Allosteric modulation of the glutamate site on the NMDA receptor by four novel glycine site antagonists
Alan Foster
European Journal of Pharmacology: Molecular Pharmacology, 1995
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Development of Radiolabeled Ligands Targeting the Glutamate Binding Site of the N-Methyl-d-aspartate Receptor as Potential Imaging Agents for Brain
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Journal of Medicinal Chemistry, 2016
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Structural Basis for Understanding Structure−Activity Relationships for the Glutamate Binding Site of the NMDA Receptor
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Journal of Medicinal Chemistry, 2002
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Structural Dynamics of the Glycine-binding Domain of the N -Methyl-d-Aspartate Receptor
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Journal of Biological Chemistry, 2014
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A common mechanism allows selective targeting of GluN2B subunit-containing N-methyl-D-aspartate receptors
Michael Hollmann
Communications Biology
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Ncm- d-aspartate: A novel caged d-aspartate suitable for activation of glutamate transporters and N-methyl- d-aspartate (NMDA) receptors in brain tissue
Yanhua Huang
Neuropharmacology, 2005
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MPX-004 and MPX-007: New Pharmacological Tools to Study the Physiology of NMDA Receptors Containing the GluN2A Subunit
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PloS one, 2016
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Proceedings of the National Academy of Sciences, 2001
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Glycine-glutamate interactions at the NMDA receptor: role of cysteine residues
Bodo Laube
FEBS Letters, 1993
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Synthesis and in vitro evaluation of 18F-labelled S-fluoroalkyl diarylguanidines: Novel high-affinity NMDA receptor antagonists for imaging with PET
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Bioorganic & Medicinal Chemistry Letters, 2010
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Structural determinants of the blocker binding site in glutamate and NMDA receptor channels
Antonio Ferrer
Neuropharmacology, 1998
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The bioactive protein-ligand conformation of GluN2C-selective positive allosteric modulators bound to the NMDA receptor
Gil Shaulsky
Molecular pharmacology, 2017
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Molecular Determinants of Agonist Discrimination by NMDA Receptor Subunits: Analysis of the Glutamate Binding Site on the NR2B Subunit
Hirokazu Hirai
Neuron, 1997
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Partial Agonists and Subunit Selectivity at NMDA Receptors
Rune Risgaard
Chemistry - A European Journal, 2010
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A Spatial Model of the Glycine Site of the NR1 Subunit of NMDA-Receptor and Ligand Docking
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Doklady Biochemistry and Biophysics, 2002
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A novel binding mode reveals two distinct classes of NMDA receptor GluN2B-selective antagonists
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Molecular pharmacology, 2016
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[3H]5,7-Dichlorokynurenic acid, a novel radioligand labels NMDA receptor-associated glycine binding sites
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European Journal of Pharmacology: Molecular Pharmacology, 1991
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